Results 31 to 40 of about 13,481 (259)

Greener Selective Cycloalkane Oxidations with Hydrogen Peroxide Catalyzed by Copper-5-(4-pyridyl)tetrazolate Metal-Organic Frameworks [PDF]

, 2015
Microwave assisted synthesis of the Cu(I) compound [Cu(µ4-4-ptz)]n [1, 4-ptz = 5-(4-pyridyl)tetrazolate] has been performed by employing a relatively easy method and within a shorter period of time compared to its sister compounds.
Martins, Luisa, Mobin, Shaikh, Mukhopadhyay, Suman, Nasani, Rajendar, Pombeiro, Armando, Saha, Manideepa   +5 more
core   +6 more sources

Crystal structure of poly[di-μ-aqua-{5-[(1Z)-2-(4-chlorophenyl)-1-cyanoethenyl]-1,2,3,4-tetrazol-1-ido-κN1}sodium]

Acta Crystallographica Section E: Crystallographic Communications, 2015
In the title compound, [Na(C10H5ClN5)(H2O)2]n, infinite chains of [Na(H2O)2]+ cations having a diamond-shaped cross-section and running parallel to the b axis are formed.
Joel T. Mague, Shaaban K. Mohamed, Mehmet Akkurt, Ahmed M. M. El-Saghier, Mustafa R. Albayati   +4 more
doaj   +1 more source

Safe and Efficient Tetrazole Synthesis in a Continuous Flow Microreactor [PDF]

, 2011
Safer flow: The synthesis of 5-substituted tetrazoles in flow (see scheme) is safe, efficient, scalable, requires no metal promoter, and uses a near-equimolar amount of NaN[subscript 3], yet nonetheless displays a broad substrate scope.
Jamison, Timothy F., Palde, Prakash B.
core   +1 more source

3-(1,2,3-Triazol-4-yl)-β-Carbolines and 3-(1H-Tetrazol-5-yl)-β-Carbolines: Synthesis and Evaluation as Anticancer Agents

Pharmaceuticals, 2022
Herein, the synthesis and anticancer activity evaluation of a series of novel β-carbolines is reported. The reactivity of nitrosoalkenes towards indole was explored for the synthesis of novel tryptophan analogs where the carboxylic acid was replaced by a
João L. P. Ribeiro, Joana B. Loureiro, Susana M. M. Lopes, Lucília Saraiva, Teresa M. V. D. Pinho e Melo   +4 more
doaj   +1 more source

Synthesis of tetrazole analogs of amino acids using Fmoc chemistry: isolation of amino free tetrazoles and their incorporation into peptides [PDF]

, 2007
An efficient synthesis of tetrazole analogs of amino acids starting from Nα-​Fmoc amino acid (Fmoc = 9-​fluorenylmethoxycarbonyl) in a three-​step protocol is reported.
Chennakrishnareddy, G., Shankar Naik, A., Sureshbabu, V.V., Venkataramanarao, R.   +3 more
core   +2 more sources

Selective synthesis of ureas and tetrazoles from amides controlled by experimental conditions using conventional and microwave irradiation

Journal of Saudi Chemical Society, 2018
An efficient synthetic procedure has been achieved for selective synthesis of 1,5-disubstituted tetrazoles and diaryl ureas from secondary amides in situ in the presence of NaN3 and POCl3 as solvent, both by conventional and microwave methods.
Rajendran Sribalan, Andiappan Lavanya, Maruthan Kirubavathi, Vediappen Padmini   +3 more
doaj   +1 more source

Iridium-catalysed ortho-H/D and -H/T exchange under basic conditions : C-H activation of unprotected tetrazoles [PDF]

, 2016
The first examples of selective ortho-directed C-H activation with unprotected 2-aryltetrazoles are described. A new base-assisted protocol for iridium (I) hydrogen isotope exchange catalysis allows access to ortho-deuterated and tritiated tetrazoles ...
Atzrodt, Jens, Derdau, Volker, Kerr, William J., Lindsay, David M., Reid, Marc, Rojahn, Patrick, Weck, Remo   +6 more
core   +1 more source

Synthesis of New C- and N-β-d-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase

Molecules, 2018
The aim of the present study was to broaden the structure-activity relationships of C- and N-β-d-glucopyranosyl azole type inhibitors of glycogen phosphorylase.
Sándor Kun, Éva Bokor, Ádám Sipos, Tibor Docsa, László Somsák   +4 more
doaj   +1 more source

Zn/MeOH-Mediated Practical and Easy Detritylation of Protected 1-Trityltetrazoles [PDF]

, 2016
A practical and low-cost method for the detritylation of 1-titryltetrazoles using zinc and methanol is described. This procedure is versatile and efficient in the deprotection of several protected tetrazoles bearing aliphatic, aromatic, and ...
Behloul, Cherif, Benseghir, Saadia, Bouchelouche, Kenza, Guijarro, David, Hadji, Yasmine, Nájera, Carmen, Yus, Miguel   +6 more
core   +2 more sources

New endoperoxides highly active in vivo and in vitro against artemisinin-resistant Plasmodium falciparum [PDF]

, 2018
Background: The emergence and spread of Plasmodium falciparum resistance to artemisinin-based combination therapy in Southeast Asia prompted the need to develop new endoperoxide-type drugs.
A Gómez-Zavaglia, A Ismael, A Ismael, A Paulo, A Siriwardana, AM Dondorp, AM Dondorp, António Sebastião Rodrigues, B Weniger, B Witkowski, B Witkowski, Bruno Guerreiro, C Amaratunga, C Amaratunga, D Ménard, EA Ashley, ES Schaffert, F Ariey, F Nogueira, F Teuscher, Fatima Nogueira, FG Baptista, H Noedl, H Noedl, H Singh, HM Ismail, I Fernández, J Adamec, J Jourdan, J Straimer, J Straimer, J Straimer, J Straimer, JL Vennerstrom, K Chauhan, K Chauhan, K Chotivanich, KM Tun, L Lobo, LH Carvalho, Lis Lobo, Lília I. L. Cabral, M Drąg-Zalesińska, M Machado, M Mota, M Tukulula, MA Fügi, Maria Inês Sena, Maria L. S. Cristiano, MD Spring, N Thuy-Nhien, NCP Araújo, PB Mohite, PM O’Neill, PN Soh, RJ Herr, RS Upadhayaya, S Arulmurugan, S Chaorattanakawee, S Nwaka, S Takala-Harrison, S Takala-Harrison, SA Santos, SD Fontaine, T Yang, TNC Wells, Valter Ferreira de Andrade-Neto, VS de Sena Pereira, W Peters, WA Kite, World Health Organization, X Fan, Y Lubell, Y Tang, Z Li, Z Wang   +75 more
core   +2 more sources