Results 151 to 160 of about 44,050 (359)

Tackling Microbial Resistance with Isatin-Decorated Thiazole Derivatives: Design, Synthesis, and in vitro Evaluation of Antimicrobial and Antibiofilm Activity

Drug Design, Development and Therapy, 2022
Refaie M Kassab,1 Sami A Al-Hussain,2 Nooran S Elleboudy,3 Amgad Albohy,4 Magdi EA Zaki,2 Khaled AM Abouzid,5,6 Zeinab A Muhammad7 1Department of Chemistry, Faculty of Science, Cairo University, Giza, 12613, Egypt; 2Department of Chemistry, Faculty of ...
Kassab RM, Al-Hussain SA, Elleboudy NS, Albohy A, Zaki MEA, Abouzid KAM, Muhammad ZA   +6 more
doaj  

A Comprehensive Review of Magnetic Nanocatalysts for C−S, C−Se Bond Formation

ChemistryOpen, EarlyView.
This review manuscript provides an exhaustive examination of magnetic nanocatalysts and their pivotal role in the formation of carbon‐sulfur (C−S) and carbon‐selenium (C−Se) bonds. The study delves into the latest advancements in the synthesis, characterization, and application of magnetic nanocatalysts, highlighting their unique advantages, including ...
Radwan Ali, Jianlin Han, Mosstafa Kazemi, Ramin Javahershenas   +3 more
wiley   +1 more source

Thiazole Effect on Phycomyces [PDF]

Proceedings of the National Academy of Sciences, 1941
William J. Robbins, Frederick Kavanagh
openaire   +3 more sources

Synthesis, Anticancer Evaluation, and Molecular Docking of Novel Thiazolobenzimidazole–Thiazole Hybrids as Potent Colon Cancer Inhibitors

ChemistryOpen, EarlyView.
Novel benzimidazothiazole–thiazole hybrids are synthesized and evaluated for anticancer activity against HCT‐116 colon cancer cells. Compound 16b shows superior cytotoxicity over doxorubicin. Molecular docking confirms strong binding to 6MTU protein, and ADMET profiling indicates favorable pharmacokinetics and low toxicity.
Bader Huwaimel, Amr S. Abouzied, Magdi E. A. Zaki, Abdulwahab Alamri, Basant Farag, Saad Alqarni, Sobhi M. Gomha   +6 more
wiley   +1 more source

Design, Synthesis, In Silico Absorption, Distribution, Metabolism, and Elimination and Molecular Docking Studies of Thiazole‐Based Furan Derivatives, and Their Biological Evaluation for Alzheimer Disease Therapy

ChemistryOpen, EarlyView.
GA: Oxidative stress plays a critical role in Alzheimer's disease (AD) by promoting Aβ plaque accumulation and tau pathology, accelerating neurodegeneration. Elevated reactive oxygen species contribute to cognitive decline through extensive oxidative damage.
Abdüllatif Karakaya, Ulviye Acar Çevik, Betül Kaya, Bilge Çiftçi, Adem Necip, Mesut Işık, Şükrü Beydemir, Yusuf Özkay, Zafer Asım Kaplancıklı   +8 more
wiley   +1 more source

Synthesis of 1,3,5-Triazepines and Benzo[f][1,3,5]triazepines and Their Biological Activity: Recent Advances and New Approaches

Molecules
This review article discusses the recent progress in synthesizing seven-membered ring 1,3,5-triazepine and benzo[f][1,3,5]triazepine derivatives. These derivatives can be either unsaturated, saturated, fused, or separated.
Ameen Ali Abu-Hashem, Othman Hakami, Nasser Amri, Yousef E. Mukhrish, Ahmed A. M. Abdelgawad   +4 more
doaj   +1 more source

The continuing significance of chiral agrochemicals

Pest Management Science, Volume 81, Issue 4, Page 1697-1716, April 2025.
In the time frame 2018–2023, around 43% of the 35 chiral agrochemicals introduced to the market (herbicides, fungicides, insecticides, acaricides, and nematicides) contain one or more stereogenic centers in the molecule, and almost 69% of them have been marketed as racemic mixtures of enantiomers or stereoisomers.
Peter Jeschke
wiley   +1 more source

Chlorination of 2-Amino Thiazoles and the Use of Chlorinated Thiazoles as Possible Fungicides

, 1975
Department of Chemistry, Ravenshaw College, Cuttack·3 Manuscript received 9 September 1971, accepted 19 April 1975 Chlorination of 2-Amino Thiazoles and the Use of Chlorinated Thiazoles as Possible Fungicides.
H. TRIPATHY, G. N. MAHAPATRA
openaire   +2 more sources

Green synthesis of novel coumarin derivatives via grinding approach and their antimicrobial evaluation

Green Chemistry Letters and Reviews
Herein, a rapid, clean, less expensive and environmentally friendly route to a novel series of coumarins bearing thiazoles or 1,3,4-thiadiazoles was developed via grinding method under solvent conditions.
Anhar Abdel-Aziem
doaj   +1 more source

Low‐Background His‐Tag‐Targeting Probes for Turn‐On Fluorescence Detection of Cell Surface Proteins and Their Binding Interactions

Small, EarlyView.
Conjugating a tri‐nitrilotriacetic acid unit to quinoline‐based cyanine dyes generated probes that fluoresce upon binding to His‐tagged proteins on cell surfaces. Using the thiazole orange‐bearing probe, the binding of the receptor binding domain (RBD) of the SARS‐CoV‐2 virus to host cells is readily detected, enabling the straightforward ...
Pragati Kishore Prasad, Suraj Toraskar, Suman Khan, Tom Granot, Yael Fridmann Sirkis, Eliane Hadas Yardeni, Shira Albeck, Tamar Unger, Ekaterina Petrovich‐Kopitman, Yoseph Addadi, Rakesh Raigawali, Saurabh Anand, Sharath S. Vishweshwara, Chethan D. Shanthamurthy, Noa Oppenheimer‐Low, Raghavendra Kikkeri, Ori Avinoam, Leila Motiei, David Margulies   +18 more
wiley   +1 more source