Results 91 to 100 of about 1,836 (178)

New Borane-Protected Derivatives of α-Aminophosphonous Acid as Anti-Osteosarcoma Agents: ADME Analysis and Molecular Modeling, In Vitro Studies on Anti-Cancer Activities, and NEP Inhibition as a Possible Mechanism of Anti-Proliferative Activity. [PDF]

Int J Mol Sci, 2022
Mizerska-Kowalska M, Sowa S, Donarska B, Płaziński W, Sławińska-Brych A, Tomasik A, Ziarkowska A, Łączkowski KZ, Zdzisińska B.   +8 more
europepmc   +1 more source

Spectroscopic and biochemical characterization of metallo-β-lactamase IMP-1 with dicarboxylic, sulfonyl, and thiol inhibitors. [PDF]

Bioorg Med Chem, 2021
Zhang H, Yang K, Cheng Z, Thomas C, Steinbrunner A, Pryor C, Vulcan M, Kemp C, Orea D, Paththamperuma C, Chen AY, Cohen SM, Page RC, Tierney DL, Crowder MW.   +14 more
europepmc   +1 more source

Tripchlorolide attenuates β-amyloid generation by inducing NEP activity in N2a/APP695 cells. [PDF]

Transl Neurosci, 2021
Zeng Y, Li Y, Shen H, Lin N, Zhang J.
europepmc   +1 more source

Enhancement of Anti-Tumoral Immunity by β-Casomorphin-7 Inhibits Cancer Development and Metastasis of Colorectal Cancer. [PDF]

Int J Mol Sci, 2021
Mori S, Fujiwara-Tani R, Kishi S, Sasaki T, Ohmori H, Goto K, Nakashima C, Nishiguchi Y, Kawahara I, Luo Y, Kuniyasu H.   +10 more
europepmc   +1 more source

Mutation of an active site-adjacent residue in VIM indirectly dictates interactions with and blunts inhibition by D-captopril. [PDF]

J Inorg Biochem
Silwal SB, Wamsley B, Wang Z, Gung BW, Nix JC, Page RC.   +5 more
europepmc   +1 more source

Ovarian cancer G protein-coupled receptor 1 inhibits A549 cells migration through casein kinase 2α intronless gene and neutral endopeptidase. [PDF]

BMC Cancer, 2022
Sharma AL, Meitei PM, Machathoibi TC, Singh NT, Singh TR, Singh LS.   +5 more
europepmc   +1 more source

Chemically tailored anionic antibiotic adjuvants targeting divalent cations to overcome carbapenem resistance in gram-negative bacteria. [PDF]

Sci Adv
Tang H, Zhao X, Sun M, Qi J, Huang Z, Zhu Y, Zeng Y, Xia Y, Luo Z, Jiang X.   +9 more
europepmc   +1 more source

Anti-Colorectal Cancer Chemotherapy-Induced Diarrhoea: Current Treatments and Side-Effects [PDF]

, 2014
Bornstein, Joel C, McQuade, Rachel, Nurgali, Kulmira   +2 more
core   +2 more sources

Fluorescently Modified NDM-1: A Versatile Drug Sensor for Rapid In Vitro β-Lactam Antibiotic and Inhibitor Screening. [PDF]

ACS Omega
Chung SF, Tam SY, Wong WT, So PK, Cheong WL, Mak CW, Lee LM, Chan PH, Wong KY, Leung YC.   +9 more
europepmc   +1 more source

GPR35 agonists inhibit TRPA1-mediated colonic nociception through suppression of substance P release. [PDF]

Pain
Gupta RA, Higham JP, Pearce A, Urriola-Muñoz P, Barker KH, Paine L, Ghooraroo J, Raine T, Hockley JRF, Rahman T, St John Smith E, Brown AJH, Ladds G, Suzuki R, Bulmer DC.   +14 more
europepmc   +1 more source