Results 91 to 100 of about 1,394 (176)

Distinct Inhibition Modes of New Delhi Metallo-β-lactamase-1 Revealed by NMR Spectroscopy. [PDF]

JACS Au, 2023
Cheng K, Wu Q, Yao C, Chai Z, Jiang L, Liu M, Li C.   +6 more
europepmc   +1 more source

Prediction of Phytochemicals for Their Potential to Inhibit New Delhi Metallo β-Lactamase (NDM-1). [PDF]

Pharmaceuticals (Basel), 2023
Bibi Z, Asghar I, Ashraf NM, Zeb I, Rashid U, Hamid A, Ali MK, Hatamleh AA, Al-Dosary MA, Ahmad R, Ali M.   +10 more
europepmc   +1 more source

New Borane-Protected Derivatives of α-Aminophosphonous Acid as Anti-Osteosarcoma Agents: ADME Analysis and Molecular Modeling, In Vitro Studies on Anti-Cancer Activities, and NEP Inhibition as a Possible Mechanism of Anti-Proliferative Activity. [PDF]

Int J Mol Sci, 2022
Mizerska-Kowalska M, Sowa S, Donarska B, Płaziński W, Sławińska-Brych A, Tomasik A, Ziarkowska A, Łączkowski KZ, Zdzisińska B.   +8 more
europepmc   +1 more source

Oxygen-Controlled Assembly of Chiral [7]-Helicene on ZnO Surfaces. [PDF]

Langmuir
Hakimi Raad N, Lyutakov O, Yang PQ, Hsu HS, Rezek B, Ukraintsev E.   +5 more
europepmc   +1 more source

Mutation of an active site-adjacent residue in VIM indirectly dictates interactions with and blunts inhibition by D-captopril. [PDF]

J Inorg Biochem
Silwal SB, Wamsley B, Wang Z, Gung BW, Nix JC, Page RC.   +5 more
europepmc   +1 more source

Spectroscopic and biochemical characterization of metallo-β-lactamase IMP-1 with dicarboxylic, sulfonyl, and thiol inhibitors. [PDF]

Bioorg Med Chem, 2021
Zhang H, Yang K, Cheng Z, Thomas C, Steinbrunner A, Pryor C, Vulcan M, Kemp C, Orea D, Paththamperuma C, Chen AY, Cohen SM, Page RC, Tierney DL, Crowder MW.   +14 more
europepmc   +1 more source

Chemically tailored anionic antibiotic adjuvants targeting divalent cations to overcome carbapenem resistance in gram-negative bacteria. [PDF]

Sci Adv
Tang H, Zhao X, Sun M, Qi J, Huang Z, Zhu Y, Zeng Y, Xia Y, Luo Z, Jiang X.   +9 more
europepmc   +1 more source

Tripchlorolide attenuates β-amyloid generation by inducing NEP activity in N2a/APP695 cells. [PDF]

Transl Neurosci, 2021
Zeng Y, Li Y, Shen H, Lin N, Zhang J.
europepmc   +1 more source

Étude de l'effet de divers inhibiteurs de protéases sur l'activité biologique de peptides in vitro

, 1989
La présente étude traite de la stabilité des neurokinines, des kinines et des angiotensines, sur des tissus isolés très sensibles à ces peptides. La stabilité a été évaluée de façon indirecte par la mesure des activités biologiques de ces peptides sur ...
Rouissi, Noureddine
core  

Fluorescently Modified NDM-1: A Versatile Drug Sensor for Rapid In Vitro β-Lactam Antibiotic and Inhibitor Screening. [PDF]

ACS Omega
Chung SF, Tam SY, Wong WT, So PK, Cheong WL, Mak CW, Lee LM, Chan PH, Wong KY, Leung YC.   +9 more
europepmc   +1 more source