Results 1 to 10 of about 7,635 (110)

Transdermal Permeation of Curcumin Promoted by Choline Geranate Ionic Liquid: Potential for the Treatment of Skin Diseases [PDF]

open access: yesSaudi Pharmaceutical Journal, 2022
The transdermal permeation of curcumin aided by choline and geranic acid ionic liquid (CAGE-IL) was addressed as a potential treatment for skin diseases.
Marta M D C Vila, Victor M Balcão
exaly   +4 more sources

Performance of Choline Geranate Deep Eutectic Solvent as Transdermal Permeation Enhancer: An in Vitro Skin Histological Study [PDF]

open access: yesPharmaceutics, 2021
In the present research work, we addressed the changes in skin by which deep eutectic solvents (DES) enhanced transdermal permeation of bioactive compounds and propose a rationale for this mechanism. Several studies showed that these unusual liquids were
Thaïs J Oliveira   +2 more
exaly   +4 more sources

Mechanism and Application of Chitosan and Its Derivatives in Promoting Permeation in Transdermal Drug Delivery Systems: A Review

open access: yesPharmaceuticals, 2022
The mechanisms and applications of chitosan and its derivatives in transdermal drug delivery to promote drug permeation were reviewed in this paper.
Jinqian Ma, Yuchen Wang, Rong Lu
exaly   +3 more sources

A melatonin textile transdermal patch based on physicochemical synergistic permeation-enhancement strategy for circadian rhythm regulation [PDF]

open access: yesFrontiers in Bioengineering and Biotechnology
Melatonin, an endogenous circadian rhythm-regulating hormone, has faced challenges in achieving prolonged exogenous regulation due to its low oral bioavailability and short half-life.
Juyang Zhao   +9 more
doaj   +2 more sources

Novel Chemical Permeation Enhancers for Transdermal Drug Delivery

open access: yesAsian Journal of Pharmaceutical Sciences, 2014
Transdermal drug delivery has been accepted as a potential non-invasive route of drug administration, with advantages of prolonged therapeutic action, decreased side effect, easy use and better patient compliance.
Yang Chen, Xiaochang Liu, Peng Quan
exaly   +3 more sources

Transdermal Permeation and Anti-Inflammation Activities of Novel Sinomenine Derivatives

open access: yesMolecules, 2016
Sinomenine is extracted from Sinomenii caulis (a traditional Chinese medicine), and it is used as the active ingredient in rheumatic arthritis treatments. It has been used in clinical applications for decades.
Jian-Cheng Wang, Chang Zhao, Jing Xiao
exaly   +3 more sources

Usefulness of Low-Resistance Electrodes Used in Iontophoresis to Enhance Skin Permeability of Drugs [PDF]

open access: yesMolecules
This study investigated how electrode design and electrical conditions influence iontophoretic transdermal drug delivery. A low-resistance silver electrode (Ag*) was developed to reduce interfacial resistance and improve the delivery of lidocaine ...
Takeshi Oshizaka   +6 more
doaj   +2 more sources

EFFECT OF ESSENTIAL OILS ON TRANSDERMAL PERMEATION OF METOPROLOL SUCCINATE [PDF]

open access: yesBulletin of Pharmaceutical Sciences. Assiut University, 2021
The objective of the present study was to prepare a matrix-type transdermal drug delivery system containing metoprolol succinate and to evaluate the effect of essential oils on transdermal permeation of drug.
B. N. Suhagia   +5 more
doaj   +1 more source

The enantioselective enhancing effect and mechanistic insights of chiral enhancers in transdermal drug delivery

open access: yesAsian Journal of Pharmaceutical Sciences, 2023
Overlook of chiral consideration in transdermal drug delivery increases administrated dose and risk of side effects, decreasing therapeutical effects. To improve the transdermal delivery efficiency of eutomer, this work focused on investigating the law ...
Yang Zhang   +9 more
doaj   +1 more source

Enhanced Transdermal Delivery of Bisoprolol Hemifumarate via Combined Effect of Iontophoresis and Chemical Enhancers: Ex Vivo Permeation/In Vivo Pharmacokinetic Studies

open access: yesPharmaceutics, 2021
Bisoprolol hemifumarate (BH) is an antihypertensive drug that is used as first-line treatment for chronic hypertension and angina pectoris. Our study was performed to enhance the transdermal delivery of BH, a hydrophilic drug active with high molecular ...
Mahmoud H. Teaima   +5 more
doaj   +1 more source

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