Results 141 to 150 of about 157,767 (395)

Modular Synthesis of Dendritic Oligo‐Glycerol Cationic Surfactants for Enhanced Antibacterial Efficacy

open access: yesAngewandte Chemie International Edition, EarlyView.
An orthogonal click chemistry approach was used to synthesize a series of cationic surfactants. The results show that an optimal balance between positive charges and hydrophobicity is a crucial factor for the improvement of antibacterial properties.
Natalie Hanheiser   +8 more
wiley   +1 more source

5-(5-Aryl-1,3,4-oxadiazole-2-carbonyl)furan-3-carboxylate and New Cyclic <em>C</em>-Glycoside Analogues from Carbohydrate Precursors with MAO-B, Antimicrobial and Antifungal Activities

open access: yesMolecules, 2012
Cyclization of acyclic <em>C</em>-glycoside derivatives <strong>1a,b</strong> to <strong>2a,b</strong> as the major isomers, and <strong>4a,b</strong> as the minor isomers were carried out.
Nagwa Said Abd El-Dayem   +3 more
doaj   +1 more source

Insights into the Nature of Synergistic Effects in Proton-Conducting 4,4−1H,1H-Bitriazole-Poly(ethylene oxide) Composites [PDF]

open access: yes, 2009
A nitrogen-containing heterocycle (NCH), 4,4-1H-1H-bi-1,2,3-triazole (bitriazole), capable of mimicking the hydrogen bonding of water in the solid state is synthesized and its ability to conduct protons in the presence of poly(ethylene oxides) under ...
Alabi, Christopher A.   +3 more
core   +1 more source

General properties and comparison of the corrosion inhibition efficiencies of the triazole derivatives for mild steel

open access: yesCorrosion reviews, 2018
Mild steel (MS) corrosion is a worldwide issue that greatly affects the industrial and natural environment. To extend the lifespan of appliances, the control of MS corrosion is necessary.
M. Faisal   +8 more
semanticscholar   +1 more source

1-[(1-{[(1S,2R,6R,8R,9S)-4,4,11,11-Tetramethyl-3,5,7,10,12-pentaoxatricyclo[7.3.0.02,6]dodecan-8-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1H-indole-2,3-dione

open access: yesIUCrData, 2017
The title compound,C23H26N4O7, adopts a Z-shaped conformation, with a dihedral angle between the mean planes of the dihydroindole and triazole rings of 70.36 (7)°.
Fatima-Zahrae Qachchachi   +5 more
doaj   +1 more source

Extensive structure‐activity relationship study of albicidin’s C‐terminal dipeptidic p‐aminobenzoic acid moiety [PDF]

open access: yes, 2019
Albicidin is a recently described natural product that strongly inhibits bacterial DNA gyrase. The pronounced activity, particularly against Gram‐negative bacteria, turns it into a promising lead structure for an antibacterial drug.
Behroz, Iraj   +7 more
core   +1 more source

Emerging threat of triazole-resistant Aspergillus fumigatus

open access: yesJournal of Antimicrobial Chemotherapy, 2018
Invasive aspergillosis is a leading cause of morbidity and mortality among immunocompromised populations and is predicted to cause more than 200 000 life-threatening infections each year. Aspergillus fumigatus is the most prevalent pathogen isolated from
J. Rybak, J. Fortwendel, P. Rogers
semanticscholar   +1 more source

Convergent Assembly of Homo‐ and Heterotypic Ubiquitin Chains from Functionalized, Expressed Monomers via Thiol‐Ene Chemistry

open access: yesAngewandte Chemie International Edition, EarlyView.
Generating functionalized ubiquitin building blocks via expression in E. coli paves the way to different di‐, tri‐, and tetra‐ubiquitin chains. Light‐induced thiol‐ene click reactions, combined with a masking and protection strategy, are harnessed to establish controlled ubiquitin chain assembly and to allow the semisynthesis of site‐selectively ...
Moritz Urschbach   +6 more
wiley   +1 more source

Synthesis, antimicrobial and cytotoxicity evaluation of new cholesterol congeners

open access: yesBeilstein Journal of Organic Chemistry, 2015
3β-Azidocholest-5-ene (3) and (3β)-3-(prop-2-yn-1-yloxy)cholest-5-ene (10) were prepared as substrates to synthesize a variety of three-motif pharmacophoric conjugates through CuAAC.
Mohamed Ramadan El Sayed Aly   +2 more
doaj   +1 more source

Towards Water Soluble Mitochondria-Targeting Theranostic Osmium(II) Triazole-Based Complexes

open access: yesMolecules, 2016
The complex [Os(btzpy)2][PF6]2 (1, btzpy = 2,6-bis(1-phenyl-1,2,3-triazol-4-yl)pyridine) has been prepared and characterised. Complex 1 exhibits phosphorescence (λem = 595 nm, τ = 937 ns, φem = 9.3% in degassed acetonitrile) in contrast to its known ...
Salem A. E. Omar   +5 more
doaj   +1 more source

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