Results 121 to 130 of about 31,516 (214)

Synthesis and Bioactivity Evaluation of a Novel 1,2,4-Oxadiazole Derivative in vitro and in 3×Tg Mice. [PDF]

Drug Des Devel Ther, 2022
Luo Z, Wang Y, Pang S, Gao S, Liu N, Gao X, Zhang L, Qi X, Yang Y, Zhang L.   +9 more
europepmc   +1 more source

Discovery of 3-phenyl-1,2,4-oxadiazole derivatives as a new class of SARS-CoV-2 main protease inhibitors. [PDF]

Bioorg Med Chem Lett, 2023
Guo N, Huang C, Qiao J, Li Y, Wang Y, Xia A, Zhang G, Fang Z, You J, Li L.   +9 more
europepmc   +1 more source

Design, Synthesis, and Biological Activity of Novel Chalcone Derivatives Containing an 1,2,4-Oxadiazole Moiety. [PDF]

Front Chem, 2022
Luo L, Liu D, Lan S, Gan X.
europepmc   +1 more source

Investigation of 3,5-diamino-1,2,4-oxadiazole as a precursor for energetic salts [PDF]

1,2,4-Oxadiazole is an attractive backbone for energetic materials as it shows a positive impact on the oxygen balance compared to other heterocycles like imidazole or triazole. The suitability of 1,2,4-oxadiazole as a cation in energetic salts should be
Lieber, Patrick, Klapötke, Thomas M., Schaller, Uwe   +2 more
core  

3D-QSAR Studies of 1,2,4-Oxadiazole Derivatives as Sortase A Inhibitors. [PDF]

Biomed Res Int, 2021
Shakour N, Hadizadeh F, Kesharwani P, Sahebkar A.   +3 more
europepmc   +1 more source

Expanding the Library of 1,2,4-Oxadiazole Derivatives: Discovery of New Farnesoid X Receptor (FXR) Antagonists/Pregnane X Receptor (PXR) Agonists. [PDF]

Molecules, 2023
Finamore C, Festa C, Fiorillo B, Leva FSD, Roselli R, Marchianò S, Biagioli M, Spinelli L, Fiorucci S, Limongelli V, Zampella A, De Marino S.   +11 more
europepmc   +1 more source

Benzamides Substituted with Quinoline-Linked 1,2,4-Oxadiazole: Synthesis, Biological Activity and Toxicity to Zebrafish Embryo. [PDF]

Molecules, 2022
Sun BL, Wang YY, Yang S, Tu MT, Shao YY, Hua Y, Zhou Y, Tan CX.   +7 more
europepmc   +1 more source

Synthesis of Some 3-Aryl-1,2,4-oxadiazoles Carrying a Protected L-Alanine Side Chain

Journal of the Brazilian Chemical Society, 1998
The synthesis of some 1,2,4-oxadiazole derivatives (4a-d) starting from arylamidoximes 1a-d and N-t-butoxycarbonyl-O-benzyl-L-aspartic acid is described. The structures of these new products have been determined by spectroscopic methods.
Melo Sebastião J. de, Sobral Antônio D., Lopes Heron de Lima, Srivastava R.M.   +3 more
doaj  

Development of 1,2,4-Oxadiazole Antimicrobial Agents to Treat Enteric Pathogens within the Gastrointestinal Tract. [PDF]

ACS Omega, 2022
Pitcher NP, Harjani JR, Zhao Y, Jin J, Knight DR, Li L, Putsathit P, Riley TV, Carter GP, Baell JB.   +9 more
europepmc   +1 more source

Synthesis, biological activity and toxicity to zebrafish of benzamides substituted with pyrazole-linked 1,2,4-oxadiazole. [PDF]

RSC Adv, 2022
Shao Y, Tu M, Yang S, Wang Y, Sun B, Shi J, Tan C, Wang X.   +7 more
europepmc   +1 more source