Results 131 to 140 of about 40,557 (208)

Synergism of a Novel 1,2,4-oxadiazole-containing Derivative with Oxacillin against Methicillin-Resistant Staphylococcus aureus. [PDF]

Antibiotics (Basel), 2021
Buommino E, De Marino S, Sciarretta M, Piccolo M, Festa C, D'Auria MV.   +5 more
europepmc   +1 more source

Design, Synthesis and Herbicidal Activity of 1,2,4-Oxadiazole Compounds as Novel Light-Dependent Protochlorophyllide Oxidoreductase Inhibitors. [PDF]

Molecules
Hu X, Miao J, Tian Y, Luo W, Shang J, Liu R, Lu H.   +6 more
europepmc   +1 more source

Radiolabeling and evaluation of ⁶⁴⁺⁶⁷Cu-2,2'-(1,2,4-Oxadiazole-3,5-diyl)di aniline as a theranostic agent for solid tumors. [PDF]

Sci Rep
Gizawy MA, Ayoup MS, Kodous AS, Abdelrahman MT, Motaleb MA.   +4 more
europepmc   +1 more source

Discovery of <i>N</i>-Acetyltransferase 8-Like (NAT8L) inhibitors based on a <i>N</i>-Acylated (Piperidin-3-ylmethyl)-1,2,4-Oxadiazole Scaffold. [PDF]

ACS Med Chem Lett
Nayeen MJ, Thomas AG, Kundu B, Carlyle E, Hin N, Hin P, Pal A, Paule J, Rais R, Slusher BS, Tsukamoto T.   +10 more
europepmc   +1 more source

Structure-Based Bioisosterism Design, Synthesis, Biological Activity and Toxicity of 1,2,4-Oxadiazole Substituted Benzamides Analogues Containing Pyrazole Rings. [PDF]

Molecules, 2022
Tu MT, Shao YY, Yang S, Sun BL, Wang YY, Tan CX, Wang XD.   +6 more
europepmc   +1 more source

Design, synthesis, and apoptotic antiproliferative activity of novel dihydropyrimidine-5-carbonitrile/1,2,4-oxadiazole hybrids as dual EGFR/VEGFR-2 inhibitors endowed with antioxidant activity. [PDF]

RSC Adv
Al-Wahaibi LH, Mohamed AM, Abou-Zied HA, Abdullah Alzahrani AY, Bräse S, Youssif BGM.   +5 more
europepmc   +1 more source

New 1,2,4-oxadiazole derivatives as potential multifunctional agents for the treatment of Alzheimer's disease: design, synthesis, and biological evaluation. [PDF]

BMC Chem
Ayoup MS, Ghanem M, Abdel-Hamid H, Abu-Serie MM, Masoud A, Ghareeb DA, Hawsawi MB, Sonousi A, Kassab AE.   +8 more
europepmc   +1 more source

Design and synthesis of new 1,2,4-oxadiazole/quinazoline-4-one hybrids with antiproliferative activity as multitargeted inhibitors. [PDF]

Front Chem
Mohamed AM, Abou-Ghadir OMF, Mostafa YA, Dahlous KA, Bräse S, Youssif BGM.   +5 more
europepmc   +1 more source

Novel 1,2,4-oxadiazole derivatives as selective butyrylcholinesterase inhibitors: Design, synthesis and biological evaluation. [PDF]

EXCLI J, 2021
Nazari M, Rezaee E, Hariri R, Akbarzadeh T, Tabatabai SA.   +4 more
europepmc   +1 more source

Development of Diphenyl-1,2,4-Oxadiazole Analogues as Allosteric Modulators of the RXFP3 Receptor: Evaluation of Importance of the N-Substituted-2-Pyrrolidone Moiety in RLX-33. [PDF]

J Med Chem
Guan D, Chaminda Lakmal HH, Bender BN, Rahman MT, Gay EA, Barrus DG, Mosera AM, Kerr AT, Besheer J, Jin C.   +9 more
europepmc   +1 more source