Results 21 to 30 of about 8,060 (204)
Corrosion Inhibition Effect of Substituted Thiadiazoles on Brass
International Journal of Electrochemical Science, 2011 The corrosion inhibition of thiadiazole derivatives for brass in natural seawater has been evaluated by potentiodynamic polarisation and electrochemical impedance spectroscopic techniques.
X. Joseph Raj, N. Rajendran
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Identification of a novel BCL2-specific inhibitor that binds predominantly to the BH1 domain [PDF]
, 2016 The antiapoptotic protein BCL 2 is overexpressed in several cancers and contributes to prolonged cell survival and chemoresistance, lending itself as an excellent target for cancer therapy.
Anderson +57 more
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1,3,4-Thiadiazoles Effectively Inhibit Proliferation of Toxoplasma gondii [PDF]
Cells, 2021 Congenital and acquired toxoplasmosis caused by the food- and water-born parasite Toxoplasma gondii (T. gondii) is one of the most prevalent zoonotic infection of global importance. T. gondii is an obligate intracellular parasite with limited capacity for extracellular survival, thus a successful, efficient and robust host cell invasion process is ...
Lidia Węglińska +7 more
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Journal of Advanced Pharmaceutical Technology & Research, 2014 The presence of heterocyclic structures in diverse types of compounds, this is strongly indicative of the profound effect like structure exerts on physiologic activity, and recognition of this is abundantly reflected in efforts to find useful synthetic ...
Dilipkumar Pal +3 more
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Electrochemical Oxidation of 2,5-Dimercapto-1,3,4-thiadiazole on Carbon Electrodes Modified with Ru(III) Schiff Base Complex [PDF]
Kemija u Industriji, 2021 The thiol compound 2,5-dimercapto-1,3,4-thiadiazole is a potential cathode material. The redox reactions of the mentioned thiol compound are slow at room temperature but can be enhanced using electron transfer mediators.
Mirha Pazalja
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Formation of Pyrazol-1,3,4-Thiadiazoles through 1,3-Dipolar Cycloadditions of 3-Thioxo-[1,2,4]-Triazepin-5-one with Nitrilimines: An Experimental and Computational study [PDF]
, 2009 In this work the results of experimental and computational study of the title compounds and some ancillary compounds are reported. Two bicyclic pyrazol-1,3,4-thiadiazole derivatives were synthesized by reaction between 6-dimethylaminomethylene-3-thioxo-
Azzouzi, S. +7 more
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1,3,4-Thiadiazole: A Promising Pharmacophore
Oriental Journal Of Chemistry, 2023 Active pharmaceutical ingredients (A.P.I.) are made up of various heteroatomic moieties. Numerous heterocycle scaffolds are regarded as crucial structures. More frequently, presence of various heteroatoms viz. nitrogen, sulphur, halogens, and oxygen atoms at different position in 5- or 6-membered rings contributed them as valued source of therapeutic ...
Nidhi Chaudhary +3 more
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Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta Praktiki, 2020 Increased attention to thiadiazole and 1,2,4-triazole derivatives is determined by the extensive structural modification capabilities of heterocyclic system derivatives and their high pharmacological potential.
A. S. Hotsulia , S. O. Fedotov
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Recent synthetic strategies of medicinally important imidazothiadiazoles
Journal of Saudi Chemical Society, 2023 Imidazothiadiazole is a fundamental fused heterocyclic compound containing imidazole and thiadiazole ring systems. This versatile framework has significant applications in pharmaceutical chemistry and also possessed a remarkable biological profile.
Tooba Jabeen +6 more
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Assessment of pharmacological activity and bioavailability of the new derivative 1,3,4-thiadiazole [PDF]
, 2018 Acexazolamide is a new derivative of 1,3,4-thiadiazole and acexamic acid. In animal experiments, acute toxicity, pharmacological activity and bioavailability of acexazolamide were ...
Demidova, M. A. +2 more
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