Results 121 to 130 of about 12,547 (208)

Antibacterial, antifungal and antimycobacterial activities of some substituted thiosemicarbazides and 2,5-disubstituted-1,3,4-thiadiazoles [PDF]

, 2001
In this research, some 1-[4-(acetylamino)benzoyl]-4-substituted thiosemicarbazides and 5-[4-(acetylamino)phenyl]-2-substitutedamino-1,3,4-thiadiazoles were screened for antibacterial, antifungal and antimycobacterial activities.

core   +1 more source

A SIMULATION APPROACH FOR NOVEL 1,3,4 THIADIAZOLE ACETAMIDE MOIETIES AS POTENT ANTIMYCOBACTERIAL AGENTS [PDF]

Objective: To design novel series of 1,3,4 thiadiazoles and to evaluate their anti-mycobacterial potency via In silico modeling. Methods: In silico modeling comprising of Lipinski rule evaluation, ADMET prediction, Molecular docking and Simulation ...
MATHEWS, SANTHOSH M., VARGHESE, SAIRA SUSAN   +1 more
core  

In vitro and in silico insights into antimicrobial and anticancer activities of novel imidazo[2,1-b][1,3,4]thiadiazoles. [PDF]

Sci Rep
Dwarakanath D, Nayak YN, Kulal A, Pandey S, Pai KSR, Gaonkar SL.   +5 more
europepmc   +1 more source

Design, synthesis and biological evaluation of non-glucosidal based 1,3,4-thiadiazoles as SGLT-2 inhibitors. [PDF]

Future Med Chem
Sharma S, Kumar S, Gupta J, Mittal A, Khurana N.   +4 more
europepmc   +1 more source

Future Prospects in the Treatment of Parasitic Diseases: 2-Amino-1,3,4-Thiadiazoles in Leishmaniasis. [PDF]

Molecules, 2019
Serban G.
europepmc   +1 more source

Utility of 3-(2-oxo-2H-chromen-3-yl)-1-phenyl-1H-pyrazole-4-carbaldehyde in the synthesis of novel 1,3,4-thiadiazoles or 1,3-thiazoles and study their cytotoxic activity. [PDF]

Sci Rep
Abdel-Aziem A, Abdelhamid AO.
europepmc   +1 more source

Chitosan-MgO Nanocomposite: One Pot Preparation and Its Utility as an Ecofriendly Biocatalyst in the Synthesis of Thiazoles and [1,3,4]thiadiazoles. [PDF]

Nanomaterials (Basel), 2018
Riyadh SM, Khalil KD, Aljuhani A.
europepmc   +1 more source

Assessment of the Microbiological Potential and Spectroscopic Properties of New Imino-1,3,4-Thiadiazoles Showing the ESIPT Effect Strongly Enhanced by Aggregation. [PDF]

Molecules
Chruściel E, Ślusarczyk L, Gładyszewska B, Karcz D, Luchowski R, Nucia A, Ociepa T, Nowak M, Kowalczyk K, Włodarczyk A, Gagoś M, Okoń S, Matwijczuk A.   +12 more
europepmc   +1 more source

Comparison of HPLC, HPTLC, and In Silico Lipophilicity Parameters Determined for 5-Heterocyclic 2-(2,4-Dihydroxyphenyl)-1,3,4-thiadiazoles. [PDF]

Molecules
Paw B, Śliwa R, Komsta Ł, Senczyna B, Karpińska M, Matysiak J.   +5 more
europepmc   +1 more source

Identification of the minimum PAR4 inhibitor pharmacophore and optimization of a series of 2-methoxy-6-arylimidazo[2,1-b][1,3,4]thiadiazoles. [PDF]

Bioorg Med Chem Lett, 2016
Temple KJ, Duvernay MT, Maeng JG, Blobaum AL, Stauffer SR, Hamm HE, Lindsley CW.   +6 more
europepmc   +1 more source