Results 121 to 130 of about 14,599 (204)

Future Prospects in the Treatment of Parasitic Diseases: 2-Amino-1,3,4-Thiadiazoles in Leishmaniasis. [PDF]

Molecules, 2019
Serban G.
europepmc   +1 more source

Utility of 3-(2-oxo-2H-chromen-3-yl)-1-phenyl-1H-pyrazole-4-carbaldehyde in the synthesis of novel 1,3,4-thiadiazoles or 1,3-thiazoles and study their cytotoxic activity. [PDF]

Sci Rep
Abdel-Aziem A, Abdelhamid AO.
europepmc   +1 more source

Chitosan-MgO Nanocomposite: One Pot Preparation and Its Utility as an Ecofriendly Biocatalyst in the Synthesis of Thiazoles and [1,3,4]thiadiazoles. [PDF]

Nanomaterials (Basel), 2018
Riyadh SM, Khalil KD, Aljuhani A.
europepmc   +1 more source

Comparison of HPLC, HPTLC, and In Silico Lipophilicity Parameters Determined for 5-Heterocyclic 2-(2,4-Dihydroxyphenyl)-1,3,4-thiadiazoles. [PDF]

Molecules
Paw B, Śliwa R, Komsta Ł, Senczyna B, Karpińska M, Matysiak J.   +5 more
europepmc   +1 more source

ZnX2 (X = Cl, Br) catalyzed efficient regioselective synthesis of 1,3,4-oxadiazole and 1,3,4-thiadiazole rings and their antibacterial studies

, 2014
Oxadiazoles, thiadiazoles and their derivatives are important classes of heterocyclic compounds and have created great interest in synthetic organic and medicinal chemistry due to their versatile medicinal potential.
Rahman, Anisur, MD.
core  

Identification of the minimum PAR4 inhibitor pharmacophore and optimization of a series of 2-methoxy-6-arylimidazo[2,1-b][1,3,4]thiadiazoles. [PDF]

Bioorg Med Chem Lett, 2016
Temple KJ, Duvernay MT, Maeng JG, Blobaum AL, Stauffer SR, Hamm HE, Lindsley CW.   +6 more
europepmc   +1 more source

Aggregation-Modulated Excited-State Intramolecular Proton Transfer and Antifungal Potential of Selected 1,3,4-Thiadiazole Derivatives. [PDF]

Int J Mol Sci
Budziak-Wieczorek I, Rząd K, Koselski M, Górecki A, Kachel-Górecka M, Matwijczuk A, Gładyszewska B, Burg P, Okoń S, Matwijczuk A.   +9 more
europepmc   +1 more source

Structural design and cytotoxic profiling of a novel 1,3,4-thiadiazole derivative targeting MCF-7 and HCT-116 cell lines: synthesis, cytotoxicity, and <i>in silico</i> study. [PDF]

RSC Adv
Sayed M, Mohammed E, Aboubaker DH, El-Rashedy AA, Hassanien R, Tolba MS, Ahmed M.   +6 more
europepmc   +1 more source

An Imidazo[2,1-b][1,3,4]thiadiazole Derivative Inhibits the Virulence Factor α-Hemolysin by Blocking the Pullout of Its Stem Domain. [PDF]

ChemMedChem
Korotkov VS, Lukat P, Di Lucrezia R, Shekhar A, Degenhart C, Diestel R, Bilitewski U, Dinkel K, Blankenfeldt W, Brönstrup M.   +9 more
europepmc   +1 more source

Synthesis and characterization of FeCuAlO₄ as a reusable heterogeneous acidic nanocatalyst for preparation of 2-amino-1,3,4-thiadiazole derivatives in water. [PDF]

Sci Rep
Nikoo A.
europepmc   +1 more source