Results 101 to 110 of about 14,599 (204)

Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E₂ and Leukotriene Biosynthesis Inhibitors. [PDF]

ACS Med Chem Lett, 2023
Potenza M, Giordano A, Chini MG, Saviano A, Kretzer C, Raucci F, Russo M, Lauro G, Terracciano S, Bruno I, Iorizzi M, Hofstetter RK, Pace S, Maione F, Werz O, Bifulco G.   +15 more
europepmc   +1 more source

Design, Synthesis, Antibacterial Evaluations and In Silico Studies of Novel Thiosemicarbazides and 1,3,4-Thiadiazoles. [PDF]

Molecules, 2022
Janowska S, Khylyuk D, Andrzejczuk S, Wujec M.   +3 more
europepmc   +1 more source

Eco-Friendly Synthesis of 3-Aryl-2,3-dihydro-1,3,4-thiadiazoles Based on Benzofuran and Chromone Moieties

, 2020
International audienceIn consideration of green and efficient organic chemical methodology, we reported here a green, an efficient and convenient procedure for synthesis of 3-aryl-2,3-dihydro-1,3,4-thiadiazoles based on benzofuran as well as chromone ...
Abdel-Aziem, Anhar, Kirsch, Gilbert, El-Sawy, Eslam   +2 more
core   +1 more source

1,3,4-Thiadiazoles Effectively Inhibit Proliferation of Toxoplasma gondii. [PDF]

Cells, 2021
Węglińska L, Bekier A, Dzitko K, Pacholczyk-Sienicka B, Albrecht Ł, Plech T, Paneth P, Paneth A.   +7 more
europepmc   +1 more source

New 1,3,4-thiadiazoles as potential anticancer agents: pro-apoptotic, cell cycle arrest, molecular modelling, and ADMET profile. [PDF]

RSC Adv, 2023
Hekal MH, Farag PS, Hemdan MM, El-Sayed AA, Hassaballah AI, El-Sayed WM.   +5 more
europepmc   +1 more source

Exploring the Antiparasitic Activity of Tris-1,3,4-Thiadiazoles against Toxoplasma gondii-Infected Mice. [PDF]

Molecules, 2022
Almutairi TM, Rezki N, Aouad MR, Hagar M, Bakr BA, Hamed MT, Hassen MK, Elwakil BH, Moneer EA.   +8 more
europepmc   +1 more source

Synthesis and Preliminary Anticancer Activity Assessment of N-Glycosides of 2-Amino-1,3,4-thiadiazoles. [PDF]

Molecules, 2021
Żurawska K, Stokowy M, Kapica P, Olesiejuk M, Kudelko A, Papaj K, Skonieczna M, Szeja W, Walczak K, Kasprzycka A.   +9 more
europepmc   +1 more source

Synthesis of 1,3,4-Thiadiazoles: Review

INTERNATIONAL JOURNAL OF SCIENTIFIC RESEARCH IN ENGINEERING AND MANAGEMENT
Abstract Molecules with 1,3,4-thiadiazole ring structures have potential biological relevance. These organic molecules have potentially reported for their medicinal importance. In this review, different strategies for the synthesis of biologically important molecules of 1,3,4-thiadiazole ring are briefly summarized and an attempt has been made with ...
openaire   +1 more source

2-Amino-1,3,4-thiadiazoles as Glutaminyl Cyclases Inhibitors Increase Phagocytosis through Modification of CD47-SIRPα Checkpoint. [PDF]

ACS Med Chem Lett, 2022
Park E, Song KH, Kim D, Lee M, Van Manh N, Kim H, Hong KB, Lee J, Song JY, Kang S.   +9 more
europepmc   +1 more source

Synthesis of 2-acylamino, 2-aroylamino and ethoxycarbonyl imino-1,3,4-thiadiazoles as antitumor agents

, 2007
2-Amino-1,3,4-thiadiazoles compounds (2a-e) were obtained from the reaction of thiosemi carbazide with 2-cyanomethoxyphenoxyacetonitriles (1). Mono acylamino, mono aroylamino and diethoxycarbonylimino-1,3,4-thiadiazole compounds (3a-e, 4a-e, 5a-c) were ...
Er, Mustafa, Unver, YASEMİN, Sancak, KEMAL   +2 more
core