Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta Praktiki, 2014 The creation and improvement of the original domestic medicines is anactual problem of medical and pharmaceutical industries. Chemistry of heterocyclicsystems attracts scientists all over the world, as it is associated with a number of properties of this
R. О. Shcherbyna +3 more
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SYNTHESIS, CHARACTERIZATION AND IN VITRO MICROBIAL EVALUATION OF REGIOISOMERS OF ALLYL PHENYL ETHERS DERIVED 1, 2, 4-TRIAZOLES [PDF]
, 2014 Objective: Synthesis and antimicrobial evaluation of regioisomers of allyl phenyl ethers derived 1, 2, 4-triazoles. Methods: A series of new 1,2,4-triazole derivatives of allyl phenyl ethers were synthesized by reacting a mixture of regio isomers 1-(3 ...
B., Kumar Aswamy +3 more
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MoleculesIncorporation of a trifluoromethyl group with 1,2,3-triazoles motifs was described. We explored a click reaction approach for regioselective synthesis of 1-susbstituted-4-trifluoromethyl-1,2,3-triazoles in which 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU ...
Tinghong Tang +5 more
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Acute toxicity of 5-(furan-2-yl, 2-metylfuran-3-yl)-4-amino-1,2,4-triazole-3-thiol alkyl derivatives
Zaporožskij Medicinskij Žurnal, 2017 The purpose of our work was the further exploration of the new 5-(furan-2-yl, 2-metylfuran-3-yl)-4-amino-1,2,4-triazole-3-thiol alkyl derivatives’ acute toxicity, setting some patterns of alkyl substituents influence by the Sulfur atom on the acute ...
D. M. Danilchenko, V. V. Parchenko
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SYNTHESIS, CHARACTERIZATION, AND EVALUATION OF ANTIFUNGAL PROPERTIES OF SUBSTITUTED BENZIMIDAZOLE ANALOG [PDF]
, 2018 Objective: The aim of the present study is to synthesize novel benzimidazole derivatives as potent antifungal agents.Methods: 2-chloromethyl-1H-benzimidazole has been synthesized by refluxing o-phenylenediamine with chloroacetic acid in the presence of ...
J, Anbhule Sachin, M, Vijey Aanandhi
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GREEN SYNTHESIS, DOCKING STUDIES AND ANTI DIABETIC ACTIVITY OF NOVEL AMINO FUSED TRIZOLE SCAFFOLD. [PDF]
In the present work, the green synthesis of novel amino fused triazole scaffold hybird heterocyclic derivatives have been carried out and substituted,and they were checked for docking scores against the DPP IV topoisomerase II enzyme.From that, ten
Senthil Kumar N, Subhashini D, Sumathi K
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Spectroscopic Study of some Schiff Bases Derived from Dibenzoylmethane [PDF]
, 2010 A series of Schiff bases 7-11 derived from dibenzoylmethane have been prepared. The UV, IR, 1H NMR and mass spectra revealed theses compounds were existed mainly as the keto-enamine tautomer in the solution.
A. Saeed, Bahjat, Al-Masoudi, Wasfi A.
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Angewandte Chemie, EarlyView.Bei vielen Pd‐katalysierten Kreuzkupplungen hat sich gezeigt, dass die Katalysatorleistung durch dessen Aktivierung begrenzt wird. Methylnaphthyl (MeNAP)‐Palladiumtrifluoracetat‐Dimere werden als leicht zu lagernde und handhabende Präkatalysatoren vorgestellt, die sich unter Reaktionsbedingungen schnell aktivieren, selbst wenn nur schwach ...
Sourav Manna +6 more
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Propanoyl(1Z)-N-(2,6-dimethylphenyl)-2-oxopropanehydrazonoate as inhibitor for corrosion of 6061 Al alloy15 % (v) SiC(p) composite in hydrochloric acid media [PDF]
, 2012 : The corrosion inhibition effect of Propanoyl(1Z)-N-(2,6-dimethylphenyl)-2-oxopropanehydrazonoate (PDOH) in the corrosion of 6061 Aluminium alloy-15%(v) SiC(p)Â composite in 0.5 and 1M hydrochloric acid medium at four different temperatures (30, 40, 50 ...
Herle, Ramadev +4 more
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NASA patent abstracts bibliography: A continuing bibliography. Section 1: Abstracts (supplement 41) [PDF]
s are provided for 131 patents and patent applications entered into the NASA scientific and technical information system during the period Jan. 1992 through Jun. 1992.
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