Results 21 to 30 of about 25,693 (164)
Chemistry of heterocyclic compounds is one of the most popular sector in organic chemistry. Scientists allocate among them a class of derivatives of 1,2,4-triazole.
I. I. Aksyonova-Seliuk +2 more
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Syntheses of 1, 2, 4 Triazole Derivatives and their Biological Activity [PDF]
Cyclisation of [4‐(4‐oxo‐2‐phenyl‐4H‐quinazolin‐3‐yl)‐phenoxy]‐acetic acid‐N′‐(substituted phenyl)‐thiosemicarbazides with sodium metal in 99.0 % ethanol gave 3‐[4‐(4‐substituted phenyl‐5‐thioxo‐4,5‐dihydro‐1H‐1,2,4 triazol‐3‐ylmethoxy)‐ phenyl]‐2‐phenyl‐3H‐quinazolin‐4‐one .
Freddy H. Havaldar, Abhay R. Patil
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Evaluation Of Antioxidant Activity Of 1, 2, 4-Triazole Derivatives With Morpholine Moiety
The aim of the work was to study the antioxidant activity of 4-R-3- (morpholinomethyl)-4H-1,2,4-triazole-5-thioles and their alkyl derivatives in vitro using the method of non-enzymatic initiation of lipid peroxidation. Among the 45 compounds studied, 8 showed varying degrees of AOA.
SHCHERBYNA, Roman +5 more
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A series of novel compounds like 3[(phenyl substituted)-5-methyl-1(Benzosulphonylamine)]-1,3,4-triazole-2-ones II(a-f) were synthesized by treating 4-amino-1-phenyl-3-methyl-5-oxo-1,2,4-triazoles with benzene sulphonyl chloride using pyridine as solvent.
Mahabaleshwaraiah Neelgundmath +1 more
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SYNTHESIS AND ANTIBACTERIAL EVALUATION OF CERTAIN 1,2,4- TRIAZOLE AND THIAZOLID INONE DERIVATIVES
The synthesis of certain 3 - (4- chloro - 3,5 - đimethyl - phenoxy ) methyl 4-alkyl or aryl -5 mercapto - 1,2,4 - triazoles ( 5a - e) is described.
Awatef Farag +3 more
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Novel Syntheses of Some 1, 2, 4‐Triazoles as Potent Bacteriocidal Agents [PDF]
A facile syntheses of 4‐aryl‐5‐(isomeric pyridoyl)‐3H‐1, 2, 4‐triazoles as potent bacteriocidal agents are described. The newly synthesized compounds were characterized by spectral and elemental analyses. Some compounds were screened for their antibacterial activity against S. aureus, E. coli, B. subtilis and P.aeruginosa. All compounds carrying 1, 2,
Ram Janam Singh, Dharmendra Kumar Singh
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Several fluoro phenyl triazoles were synthesized using click chemistry between fluoro phenyl azides and phenyl acetylene. Under ultrasound irradiation, this synthetic procedure was performed with Cu (I) in the presence of 1,10-phenanthroline.
Elisa Leyva +3 more
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Syntheses, Characterization and Biological Activity of Some 1, 2, 4‐Triazole Derivatives [PDF]
Syntheses of a series of 3‐alkyl‐4‐ amino‐5‐ cyanomethyl‐4H‐1, 2, 4‐triazoles with active methylene groups are described. The newly synthesized compounds were characterized by spectral and elemental analyses. Some compounds were screened for their antibacterial activity against S. aureus, E. coli, B. subtilis and P. aeruginosa.
R. J. Singh, D. K. Singh
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Synthesis of New Bis-1,2,4-Triazole Derivatives
A series of new 1,2/1,3-bis[o-(N-methylidenamino-3-aryl-5-phenyl-4H-1,2,4-triazole-4-yl)phenoxy]ethane/propane derivatives 4 were prepared in good yields bytreatment of 4-amino-3-aryl-5-phenyl-4H-1,2,4-triazoles 2 with certain bis-aldehydes 1.Compounds 4
Hakan Bektas, Olcay Bekircan
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Introduction. Modern medicine is faced with the resistance of Candida spp. to antimycotics, due to changes in the expression and structure of the ERG11 gene, the molecular target of triazoles.
Yuri V. Nesvizhsky +9 more
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