Results 101 to 110 of about 21,202 (267)

Synthesis of Some 2, 6-Disubstituted 4-Amidopyridines and -Thioamidopyridines, and Their Antimycobacterial and Photosynthesis-Inhibiting Activity

Molecules, 2000
A group of 26 new 2-halogeno-6-alkylsulfanyl- and 2,6-bis-alkylsulfanyl-4-amidopyridines and corresponding thioamidopyridines was synthesised. Some of the amidopyridines and all thioamidopyridines were tested for their antimycobacterial activity against ...
Miroslav Miletin, Jiri Hartl, Z. Odlerova, Martin Dolezal, K. Kralova, Milos Machacek   +5 more
doaj   +1 more source

Antibacterial and Antibiofilm Activity of 8‐Hydroxyquinoline Derivatives Against Mycobacterium and Staphylococcus Species

Chemistry &Biodiversity, Volume 22, Issue 12, December 2025.
Synthesis of 8‐hydroxyquinoline derivatives (QD 1‐12) from different analogues of 8‐hydroxyquinoline (HQ 1‐4). The derivatives and parent compounds were evaluated for antibacterial and antibiofilm activity against Mycobacterium tuberculosis, Mycobacterium smegmatis, methicillin‐resistant Staphylococcus aureus and methicillin‐sensitive Staphylococcus ...
Namrita Lall, Anna‐Mari Kok, Carel B. Oosthuizen, Surjeet Verma, François Chassagne, Phuc H. Vo, Khanh‐Van Ho, Chung‐Ho Lin, Cassandra L. Quave, Danielle Twilley   +9 more
wiley   +1 more source

Synthesis of N,N’-Diarylalkanediamides and Their Antimycobacterial and Antialgal Activity

Molecules, 2000
A set of N,N'-diarylalkanediamides was synthesized. The compounds were tested for their antimycobacterial and antialgal activity. The antimycobacterial activity of N,N'-diarylalkanediamides depends on the lipophilicity of the respective acid ...
Zbynek Svoboda, Jiri Janota, Milan Slosarek, Zelmira Odlerova, Katarina Kralova, Jiri Kunes, Karel Waisser, Lenka Kubicova   +7 more
doaj   +1 more source

Study of antibacterial, antimycobacterial, antifungal, and antioxidant activities of Foeniculum vulgare: A review [PDF]

, 2016
Foeniculum vulgare (fennel) belong to Apiaceae family has been used in traditional medicine for many therapeutic purposes. The aim of this study was to overview its therapeutic effects than its nutritive and industrial effects.
Kiani, S., Miraj, S.
core  

2-Substituted agelasine analogs : synthesis and biological activity, and structure and reactivity of synthetic intermediates [PDF]

, 2011
2-Substituted N-methoxy-9-methyl-9H-purin-6-amines were synthesized either from their corresponding 6-chloro-9-methyl-9H-purines or 2-chloro-N-methoxy-9-methyl- 9H-purin-6-amine.
Bohlin, Lars, Burman, Robert, Charnock, Colin, Felth, Jenny, Gorbitz, Carl Henrik, Gundersen, Lise-Lotte, Larsson, Rolf, Roggen, Heidi, Tamm, Toomas   +8 more
core   +1 more source

Recent Advances in Isatin–Thiazole Hybrids: Synthesis, Structural Design, and Biological Application

Chemistry &Biodiversity, Volume 22, Issue 12, December 2025.
ABSTRACT Isatin–thiazole hybrids are considered privileged chemical scaffolds due to their broad spectrum of pharmacological properties, making them attractive candidates for drug development. As a result, isatin–thiazole derivatives have emerged as a prominent class of hybrid heterocycles and have been the focus of extensive research in recent years ...
Isadora M. G. Andrade, Edson de O. Lima Filho, Caio F. Valadão, Luana da S. M. Forezi, Fernando de C. da Silva   +4 more
wiley   +1 more source

In Silico Structure-Activity Study of Selected Triterpenoids as Potential Inhibitors of Mycolic Acid Transporter of Mycobacterial MmpL3 Receptor Protein

Sciences of Phytochemistry
Structural features of the triterpenoid skeleton that are necessary for antimycobacterial activity are not well understood. Following the isolation of the triterpenoids ergosterol-5,8-endoperoxide, 6β-hydroxykulactone, 12β-hydroxykulactone, (24R)-24,25 ...
Mohamed Said Rajab
doaj   +1 more source

Bioprospecting of Labdane‐Type Diterpenes From Austroeupatorium laetevirens: Molecular Networking, Structural Elucidation, and Biological Activity Evaluation

Chemistry &Biodiversity, Volume 22, Issue 12, December 2025.
ABSTRACT Labdane‐type diterpenes are the main specialized metabolites in the Austroeupatorium genus, known for diverse biological activities. This study employed molecular networking to facilitate the identification of labdanes in Austroeupatorium laetevirens, alongside isolation, structural elucidation, and evaluation of anti‐Mycobacterium ...
Francielli A. P. Valeze, Maria Eduarda V. de Souza, Beatriz P. Moreno, Bianca D. B. Sahm, Andressa L. Ieque, Cleverton S. Fernandes, Regiane B. L. Scodro, Leticia V. Costa‐Lotufo, Marta R. B. do Carmo, Andrea N. L. Batista, João M. Batista Junior, Ernani A. Basso, Maria H. Sarragiotto, Debora C. Baldoqui   +13 more
wiley   +1 more source

Tricks to translating TB transcriptomics. [PDF]

, 2015
Transcriptomics and other high-throughput methods are increasingly applied to questions relating to tuberculosis (TB) pathogenesis. Whole blood transcriptomics has repeatedly been applied to define correlates of TB risk and has produced new insight into ...
Coussens, AK, Deffur, A, Wilkinson, RJ
core   +1 more source

The Impact of Essential Oils From Aromatic Plants on Microbial Dynamics and Nutrition in Lacto‐Fermented Systems

Food Science &Nutrition, Volume 13, Issue 12, December 2025.
Bioactive compounds found in essential oils (EOs), which are obtained by distilling certain plants, have been shown to inhibit pathogenic microorganisms and also support the growth of probiotic bacteria. In this context, EO nutraceuticals have properties that can improve the shelf life and sensory properties of products.
Ibrahim Canbey, Tulay Ozcan, Ozan Gurbuz
wiley   +1 more source