Results 71 to 80 of about 7,765 (231)
Biosynthetic Studies of Aziridine Formation in Azicemicins
, 2016 Biosynthetic Studies of Aziridine Formation in ...
Hung-wen Liu (1279131) +1 more
core +1 more source
Stereocontrolled Synthesis of 1,2- and 1,3-Diamine Building Blocks from Aziridine Aldehyde Dimers
, 2016 Vicinal aziridine-containing diamines have been obtained with high syn-stereoselectivity from readily available aziridine aldehyde dimers in the Petasis borono-Mannich reaction.
Jeffrey D. St. Denis (1724728) +3 more
core +2 more sources
European Journal of Organic Chemistry, Volume 29, Issue 22, 9 June 2026.Glycomimetics with triazoline and aziridine groups were synthesised via diastereoselective Huisgen cycloaddition from glycosyl azides. Density functional theory was applied to define the mechanism for BF3 promoted aziridine formation. Triazoline and aziridine derivatives were synthesised by diastereo‐ and regioselective Huisgen cycloaddition of 2,3,4,6‐
Aaron McCormack +4 more
wiley +1 more source
Aziridine Lithiation Using Lewis Acid Activation
, 2016 Aziridine Lithiation Using Lewis Acid ...
Edwin Vedejs (1264683) +1 more
core +1 more source
On Differences between Racemic and Enantiomerically Pure Forms of Aziridine-2-Carboxamide
Synthesis, X-ray and cytotoxicity studies of (S)- and (R)-aziridine-2-carboxamide (Leakadine) are described. X-Ray data of the enantiomerically pure form are compared with those for racemic aziridine-2-carboxamide in order to explain the 21 oC large ...
Meikas, A. +7 more
core +1 more source
Electrophilic Iodination of Heterocyclic Compounds. Recent Advances 2008–2025: Part II
European Journal of Organic Chemistry, Volume 29, Issue 22, 9 June 2026.Electrophilic iodination using molecular iodine and iodide sources represents an efficient approach for accessing valuable iodinated organic compounds. This review highlights recent advances in the iodination of heterocyclic compounds from 2008 to 2025, emphasizing the role of heteroaryl iodides as important synthetic intermediates for biologically ...
Njomza Ajvazi, Stojan Stavber
wiley +1 more source
A Study on the Biological Activity of Optically Pure Aziridine Phosphines and Phosphine Oxides
MoleculesA series of optically pure aziridine phosphines and their corresponding phosphine oxides were synthesized through established chemical methodologies. The compounds were systematically investigated for their biological properties. Notably, all synthesized
Aleksandra Kowalczyk +4 more
doaj +1 more source
Aziridine-Mediated Ligation and Site-Specific Modification of Unprotected Peptides
, 2016 A synthesis of aziridine-containing peptides via the Cu(II)-promoted coupling of unprotected peptide thioacids and N–H aziridine-2-carbonyl peptides is reported.
Ryan Joseph (1831123) +3 more
core +1 more source
Beilstein Journal of Organic Chemistry, 2011 A novel synthetic methodology has been developed for the synthesis of diethyl 5-alkyl/aryl/heteroaryl substituted 3,4-dihydro-2H-pyrrole-4,4-dicarboxylates (also called 2-substituted pyrroline-4,5-dihydro-3,3-dicarboxylic acid diethyl esters) by iodide ...
Satish S. More +4 more
doaj +1 more source
5-Azido-4-dimethylamino-1-methyl-1,2,4-triazolium Hexafluoridophosphate and Derivatives
Crystals, 2016 5-Azido-4-(dimethylamino)-1-methyl-1,2,4-triazolium hexafluoridophosphate was synthesized from the corresponding 5-bromo compound with NaN3. Reaction with bicyclo[2.2.1]hept-2-ene yielded a tricyclic aziridine, addition of an N-heterocyclic carbene ...
Gerhard Laus +2 more
doaj +1 more source