Results 121 to 130 of about 2,089 (211)

Concise syntheses of 7-anilino-indoline-N-benzenesulfonamides as antimitotic and vascular disrupting agents

, 2014
[[abstract]]Described herein is the development of a novel series of 7-anilino-indoline-N-benzenesulfonamides, derived from ABT751 (1), as potent anticancer agents.
Mehndiratta, S;Chiang, YF;Lai, MJ;Lee, HY;Chen, MC;Kuo, CC;Chang, CY;Chang, JY;Liou, JP
core   +1 more source

Synthesis of a new fluorophore: wavelength-tunable bisbenzo[f]isoindolylidenes. [PDF]

Chem Sci, 2023
Ye C, Huang R, Chiou MF, Wang B, Li D, Bao H.   +5 more
europepmc   +1 more source

Theoretical investigation on the molecular structure, Infrared, Raman and NMR spectra of para-halogen benzenesulfonamides, 4-X-C6H4SO2NH2 (X = Cl, Br or F)

, 2009
In the present study, the structural properties of para-halogen benzenesulfonamides, 4-XC6H4SO2NH2 (4-chlorobenzenesulfonamicle (I). 4-bromobenzenesulfonamide (II) and 4-fluorobenzenesulfonamide (III)) have been studied extensively utilizing ab initio ...
Çoruh, Ali
core   +1 more source

Radiosynthesis of three [11C]ureido-substituted benzenesulfonamides as PET probes for carbonic anhydrase IX in tumors

, 2011
Three ureido-substituted benzenesulfonamides 1a–c have been developed as potent inhibitors for carbonic anhydrase IX, which is overexpressed in hypoxic tumors. In this study, we labeled these unsymmetrical ureas 1a–c using [11C]phosgene ([11C]
福村 利光, Fujinaga, Masayuki, 460067, Asakawa, Chiharu, 460066, 460065, 460064, 由井 譲二, Kumata, Katsushi, 460069, 460068, 460070, 河村 和紀, Yamasaki, Tomoteru, 460052, Zhang, Ming-Rong, 張 明栄, 460071, Yui, Joji, 熊田 勝志, Ogawa, Masanao, Kawamura, Kazunori, Xie, Lin, 460056, 460055, 460054, 460053, 460059, 460058, 浅川 千春, 460057, 460063, 460062, 藤永 雅之, 460061, 460060, 小川 政直, 謝 琳, Fukumura, Toshimitsu, 山崎 友照   +39 more
core  

Reaction of normal and pseudo 2-formylbenzenesulfonyl chlorides with amines: experimental and theoretical studies on the structure of 2-formyl benzenesulfonamides in solid, solution and gas phases

, 1994
The reaction of 2-formylbenzenesulfonyl chloride 1 and its pseudo isomer 2 with primary amines give either the corresponding sulfonamido Schiff bases or the corresponding 2-formylbenzenesulfonamide depending on the concentration of the amine used.
Rajeev, Kallanthottathil G., Bhatt, M. Vivekananda, Shashidhar, Srikantiah M., Pius, Kuruvilla   +3 more
core   +1 more source

Quantum chemical modelling of acidity constatns of secondary benzenesulfonamides.

, 2017
Various sulfonamides are used in medicine as drug components. Depending on the properties of these compounds, they can be used as antibacterial agents, drug carriers, etc.
Ananičienė, Kristina,
core  

Benzenesulfonamide compounds for somatic embryogenesis in plants

, 2014
Benzenesulfonamide compounds potentiate 2,4-D induced embryogenesis in plants. In particular, 4-chloro-N-methyl-N-(2-methylphenyl) benzenesulfonamide and analogs induce somatic embryogenesis in plants. Methods of inducing somatic embryogenesis comprise exposing selected plant tissues, e.g. seed embryos, to auxins, e.g.
Fiers, M.A., Boutilier, K.A.
openaire   +1 more source

In-vitro high-throughput library screening-Kinetics and molecular docking studies of potent inhibitors of α-glucosidase. [PDF]

PLoS One, 2023
Ali M, Malik K, Zaidi A, Farooq U, Bukhari SM, Majeed Z, Mahnashi MH, Nawazish S, Abdulwahab A, Alshaibari KS.   +9 more
europepmc   +1 more source

Design and Synthesis of Bis-Triazole-Linked Benzenesulfonamides as Selective Carbonic Anhydrase IX/XII Inhibitors with Chemosensitizing Activity. [PDF]

J Med Chem
Roshdy E, Kilic A, Mustafa M, Celik I, Sarı ZB, Simsek E, Nocentini A, Giovannuzzi S, Supuran CT, Özensoy Güler Ö, Winum JY, Abe M.   +11 more
europepmc   +1 more source

Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. [PDF]

J Enzyme Inhib Med Chem, 2023
Badawi WA, Rashed M, Nocentini A, Bonardi A, Abd-Alhaseeb MM, Al-Rashood ST, Veerakanellore GB, Majrashi TA, Elkaeed EB, Elgendy B, Gratteri P, Supuran CT, Eldehna WM, Elagawany M.   +13 more
europepmc   +1 more source