Results 101 to 110 of about 2,854 (178)

The thiazolidinedione drug troglitazone inhibits Gq signaling through direct binding to the Gq alpha subunit through inhibition of GDP release. [PDF]

Mol Pharmacol
Issa NT, Shen T, Vizurraga A, Pronin A, Henry T, Wang Q, Kwarcinski FE, Schürer S, Badiavas E, Tall GG, Slepak VZ.   +10 more
europepmc   +1 more source

End-to-End Backbone Cyclization Enhances Passive Permeability of bRo5 Oligomeric Depsipeptides with Nonlinear Size Dependence. [PDF]

ACS Med Chem Lett
Thorpe MP, Hopkins CR, Johnston JN.
europepmc   +1 more source

Biosynthesis of the Fungal Cyclic Lipodepsipeptide Pleosporacin, a New Selective Inhibitor of the Phytopathogen Botrytis cinerea. [PDF]

Chembiochem
Wieder C, Wiechert R, Yemelin A, Sandjo LP, Thines E, Opatz T, Schüffler A.   +6 more
europepmc   +1 more source

Cyclic peptide inhibitors function as molecular glues to stabilize Gq/11 heterotrimers. [PDF]

Proc Natl Acad Sci U S A
Mühle J, Alenfelder J, Rodrigues MJ, Jürgenliemke L, Guixà-González R, Grätz L, Andres F, Bacchin A, Hennig M, Schihada H, Crüsemann M, König GM, Schertler G, Kostenis E, Deupi X.   +14 more
europepmc   +1 more source

Identification of Hoiamide A as an Inducer of Oxidative and Endoplasmic Reticulum Secretory Pathway Stress. [PDF]

J Nat Prod
Bonar SE, Mattos DR, Yu X, Neuhaus GF, Youssef DTA, Shaala LA, Gerwick WH, McPhail KL, Ishmael JE.   +8 more
europepmc   +1 more source

Antioxidant, Anti-Inflammatory and Anticancer Peptides from Extreme Marine Environments. [PDF]

Antioxidants (Basel)
Zakariya M, Montuori E, Kopp G, Coppola A, Giordano D, Bruno S, Lauritano C.   +6 more
europepmc   +1 more source

Amino acid analogues provide multiple plausible pathways to prebiotic peptides. [PDF]

J R Soc Interface
Zhang L, Ying J.
europepmc   +1 more source

Current issues in heartworm chemotherapy. [PDF]

Parasit Vectors
Geary TG.
europepmc   +1 more source

Beauvericin Induces Mitochondrial Apoptosis and Attenuates EMT-Associated Phenotypes and Angiogenic Signaling in Colorectal Cancer Cells <i>In Vitro</i>. [PDF]

J Microbiol Biotechnol
Kwon M, Jung HJ.
europepmc   +1 more source

Environmental metabolomics characterization of modern stromatolites and annotation of ibhayipeptolides. [PDF]

PLoS One
Neuhaus GF, Aron AT, Isemonger EW, Petras D, Waterworth SC, Madonsela LS, Gentry EC, Siwe Noundou X, Kalinski JJ, Polyzois A, Habiyaremye JC, Redick MA, Kwan JC, Dorrington RA, Dorrestein PC, McPhail KL.   +15 more
europepmc   +1 more source