Results 21 to 30 of about 1,345 (190)

Crystal structure of 3-((3,4-dichloroisothiazol-5-yl)methoxy)benzo[d] isothiazole 1,1-dioxide, C11H6Cl2N2O3S2

open access: yesZeitschrift für Kristallographie - New Crystal Structures, 2023
C11H6Cl2N2O3S2, triclinic, P1‾ (no. 2), a = 6.974(3) Å, b = 8.132(3) Å, c = 12.349(5) Å, α = 86.123(4)°, β = 78.299(4)°, γ = 85.715(4)°, V = 682.9(4) Å3, Z = 2, R gt(F) = 0.0410, wR ref(F 2) = 0.1058, T = 296(2) K.
Cong Huang   +4 more
doaj   +1 more source

2-(3-Methylbut-2-en-1-yl)-1,2-benzisothiazol-3(2H)-one 1,1-dioxide

open access: yesActa Crystallographica Section E, 2009
In the title compound, C12H13NO3S, a saccharin derivative, the dihedral angle between the aromatic and isothiazole rings is 2.91 (12)°. The planar 3,3-dimethylallyl group [maximum deviation = 0.0086 (16) Å]
Hafiz Mubashar-ur-Rehman   +4 more
doaj   +1 more source

Synthesis and Biological Activity of Novel Comenic Acid Derivatives Containing Isoxazole and Isothiazole Moieties

open access: yesNatural Product Communications, 2018
Methyl 5-hydroxy-4-oxo-4 H -pyran-2-carboxylate was synthesized by esterification of methanol with comenic acid under acidic catalysis. The obtained ester was alkylated with 3-(chloromethyl)-5-phenylisoxazole and 4,5-dichloro-3-(chloromethyl)isothiazole ...
Alexey V. Kletskov   +9 more
doaj   +1 more source

Electrospinning of pyrazole-isothiazole derivatives: nanofibers from small molecules [PDF]

open access: yes, 2019
We investigate the electrospinning of small molecules, specifically designed peptide derivatives of the pyrazole-isothiazole scaffold. Such non-natural peptides enhance the spectrum of fundamental materials used for electrospinning.
Eleta-Lopez, Aitziber   +11 more
core   +1 more source

The N’-Substituted Derivatives of 5-Chloro-3-Methylisothiazole-4-Carboxylic Acid Hydrazide with Antiproliferative Activity

open access: yesMolecules, 2019
Thanks to the progress in oncology, pharmacological treatment of cancer is gaining in importance and in the near future anti-cancer chemotherapeutics are expected to be the main method of treatment for cancer diseases.
Izabela Jęśkowiak   +6 more
doaj   +1 more source

A Mixture of D-Amino Acids Enhances the Biocidal Efficacy of CMIT/MIT Against Corrosive Vibrio harveyi Biofilm

open access: yesFrontiers in Microbiology, 2020
Biocides are widely used for the mitigation of microbial contamination, especially in the field of the aviation fuel industry. However, the long-term use of biocide has raised the concerns regarding the environmental contamination and microbial drug ...
Xiaomeng Liu   +15 more
doaj   +1 more source

Synthesis, Fungicidal Activity and Plant Protective Properties of 1,2,3-Thiadiazole and Isothiazole-Based N-acyl-N-arylalaninates

open access: yesMolecules, 2023
The addition of active groups of known fungicides, or systemic acquired resistance inducers, into novel compound molecules to search for potential antifungal compounds is a popular and effective strategy.
Tatiana A. Kalinina   +6 more
doaj   +1 more source

A novel synthesis of fused isothiazole ring systems [PDF]

open access: yes, 1994
The reaction of aromatic and heteroaromatic aldehydes with bis(trimethylsilyl)sulfide leads to the corresponding thioaldehydes, which, through a fine tuning of the reaction conditions, are trapped both intermolecularly and intramolecularly, thus ...
Capperucci, Antonella   +5 more
core   +1 more source

Thienoisothiazoles. I. The synthesis of Thieno[2,3-c]isothiazole and some of its derivatives

open access: yes, 1982
.Thieno[2,3-c]isothiazole-3-carboxylic acid was the compound obtained by the reaction of ethyl-3-cyano-5,5-diethoxy-2-oxopentanoate with phosphorus pentasulfide, previously assumed to yield thieno[3,4-d]isothiazole-4-carboxylic acid. The parent thieno[2,
HD Krebs, FC James
core   +1 more source

Chemistry of polyhalogenated nitrobutadienes, 10: Synthesis of highly functionalized heterocycles with a rigid 6-amino-3-azabicyclo[3.1.0]hexane moiety

open access: yesBeilstein Journal of Organic Chemistry, 2012
The nitropolychlorobutadienes 3, 4 are valuable building blocks for various amination and successive heterocyclization products. Nucleophilic substitution reactions of the partially protected, bioactive amines 1, 2 with either vinyl, imidoyl or carbonyl ...
Viktor A. Zapol’skii   +3 more
doaj   +1 more source

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