Results 151 to 160 of about 1,479 (165)

Monastrol, a 3,4-dihydropyrimidin-2(1 H )-thione, as structural scaffold for the development of modulators for GHB high-affinity binding sites and α 1 β 2 δ GABA A receptors

European Journal of Medicinal Chemistry, 2017
The α4βδ subtype of the γ-aminobutyric acid (GABA) type A receptors (GABAARs) has been shown to be implicated in high-affinity binding of the neuromodulator γ-hydroxybutyric acid (GHB), but may not be the only GHB high-affinity binding sites.
Anas Al-Khawaja, Petrine Wellendorph, Bente Frølund   +2 more
exaly   +2 more sources

Monastrol analogs: A synthesis of pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screening

Bioorganic and Medicinal Chemistry Letters, 2010
A synthesis of novel pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged pyrazolo-, tetrazolo-, benzimidazo-, and thiazolopyrimidines via Hantzsch- and Biginelli-like condensations has been developed.
Jan Svetlik, Lucia Veizerová, Thomas U Mayer   +2 more
exaly   +2 more sources

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Design, Docking Studies, and Anticancer Activity of Newly Synthesized Monastrol Analogues Bearing Ligustrazine Moiety

Russian Journal of General Chemistry, 2022
Ashraf M Mohamed, Abd El-Galil E Amr, Amr A E   +2 more
exaly  

Design, Synthesis, and Biological Screening for Cytotoxic Activity of Monastrol Analogues

Polycyclic Aromatic Compounds, 2022
Shahab Bohlooli, Saghi Sepehri
exaly  

Synthesis and differential antiproliferative activity of Biginelli compounds against cancer cell lines: Monastrol, oxo-monastrol and oxygenated analogues

Bioorganic Chemistry, 2006
Dennis Russowsky, Romulo F S Canto, Angelo De Fátima   +2 more
exaly  

Fatty-monastrol derivatives and its cytotoxic effect against melanoma cell growth

Bioorganic Chemistry, 2017
Marcelo G Montes D'Oca, Ana Paula De Souza Votto   +1 more
exaly  

Synthesis and biological evaluation of conformationally flexible as well as restricted dimers of monastrol and related dihydropyrimidones

European Journal of Medicinal Chemistry, 2011
Ahmed Kamal, M Shaheer Malik, Sistla Ramakrishna   +2 more
exaly  

Differential effects of monastrol in two human cell lines

Cellular and Molecular Life Sciences, 2004
Larisa Gheber
exaly  

Transient exposure to the Eg5 kinesin inhibitor monastrol leads to syntelic orientation of chromosomes and aneuploidy in mouse oocytes

Mutation Research - Genetic Toxicology and Environmental Mutagenesis, 2004
John B Mailhes
exaly  

Discovery of coumarin–monastrol hybrid as potential antibreast tumor-specific agent

European Journal of Medicinal Chemistry, 2013
Koneni V Sashidhara, Srinivasa Rao Avula, Gopala Reddy Palnati   +2 more
exaly