Results 221 to 230 of about 125,963 (338)

Discovery of the first M5-selective and CNS penetrant negative allosteric modulator (NAM) of a muscarinic acetylcholine receptor: (S)-9b-(4-chlorophenyl)-1-(3,4-difluorobenzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one (ML375).

Journal of Medicinal Chemistry, 2013
P. Gentry, M. Kokubo, T. Bridges, Nathan R Kett, J. Harp, Hyekyung P. Cho, Emery Smith, Peter S. Chase, P. Hodder, C. Niswender, J. Daniels, P. Conn, M. Wood, C. Lindsley   +13 more
semanticscholar   +1 more source

Endogenous muscarinic acetylcholine receptor signaling blunts α₁-adrenergic vasoconstriction during higher-intensity handgrip exercise in humans. [PDF]

Am J Physiol Regul Integr Comp Physiol
Terwoord JD, Dinenno FA, Richards JC, Hearon CM.   +3 more
europepmc   +1 more source

Sexually dimorphic muscarinic acetylcholine receptor modulation of contextual fear learning in the dentate gyrus. [PDF]

Neurobiol Learn Mem, 2021
Yavas E, Trott JM, Fanselow MS.
europepmc   +1 more source

Expression of Functional M2 Muscarinic Acetylcholine Receptor in Escherichia coli [PDF]

, 2000
Hiroyasu Furukawa, Tatsuya Haga
openalex   +1 more source

Voiding Behavior and Efferent Bladder Function Altered in Mice Following Social Defeat but Not Witness Trauma [PDF]

, 2020
Chess-Williams, Russ, McDermott, Catherine, Sellers, Donna J, West, Eliza   +3 more
core   +1 more source

Acetylcholine autoexcites the release of proopiomelanocortin-derived peptides from melanotrope cells of Xenopus laevis via an M1 muscarinic receptor.

, 1996
F. J. Van Strien, Eric W. Roubos, Hubert Vaudry, Bruce G. Jenks   +3 more
openalex   +2 more sources

Investigation of Muscarinic Acetylcholine Receptor M₃ Activation in Atomistic Detail: A Chemist's Viewpoint. [PDF]

ChemMedChem
Drabek M, Emmerich R, Djulic N, Bünemann M, Schlitzer M, Kolb P.   +5 more
europepmc   +1 more source

Disentangling bias between G_q, GRK2, and arrestin3 recruitment to the M₃ muscarinic acetylcholine receptor. [PDF]

Elife, 2021
Flöser A, Becker K, Kostenis E, König G, Krasel C, Kolb P, Bünemann M.   +6 more
europepmc   +1 more source

Differential effects of hypoxia on ligand binding properties of nicotinic and muscarinic acetylcholine receptors on cultured bovine adrenal chromaffin cells.

, 1991
Ken Lee, Kunio Koshimura, Tetsuya Ohue, Soichi Miwa   +3 more
openalex   +1 more source

Inhibition of acetylcholine muscarinic M₁ receptor function by the M₁‐selective ligand muscarinic toxin 7 (MT‐7) [PDF]

, 2000
Maria C. Olianas, Carlo Maullu, Abdu Adem, Ezra Mulugeta, Evert Karlsson, Pierluigi Onali   +5 more
openalex   +1 more source