Results 41 to 50 of about 18,651 (251)

Synthesis and Antibacterial Evaluation of Novel Heterocyclic Compounds Containing a Sulfonamido Moiety

open access: yesMolecules, 2013
Aiming for the synthesis of new heterocyclic compounds containing a sulfonamido moiety suitable for use as antibacterial agents, the precursor ethyl {[4-N-(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenylazo}cyanoacetate was reacted with a variety of active ...
Eman A. El-Bordany   +2 more
doaj   +1 more source

Synthesis of 2,6-bis-(oxazolyl)pyridine ligands for luminescent Ln(III) complexes [PDF]

open access: yes, 2012
Submitted to the European Journal of Organic ChemistryNew bis-(oxazolyl)pyridine ligands for Ln(III) ions were prepared using a expeditious methodology from threonine and dipicolinic acid chloride.
Castanheira, Elisabete M. S.   +4 more
core   +1 more source

Helium nanodroplet infrared spectroscopy of oxazole-(water)n (n = 1,2) clusters

open access: yesAIP Advances, 2021
The mass-selective infrared (IR) spectra of oxazole-(D2O)n≤2 complexes embedded in helium droplets are recorded in the spectral range of 2565–2800 cm−1. The experimental IR spectra are assigned by comparing with quantum chemical calculations at the MP2/6-
Tarun Kumar Roy   +4 more
doaj   +1 more source

Computational Redesign of Bacterial Biotin Carboxylase Inhibitors Using Structure-Based Virtual Screening of Combinatorial Libraries

open access: yesMolecules, 2014
As the spread of antibiotic resistant bacteria steadily increases, there is an urgent need for new antibacterial agents. Because fatty acid synthesis is only used for membrane biogenesis in bacteria, the enzymes in this pathway are attractive targets for
Michal Brylinski, Grover L. Waldrop
doaj   +1 more source

2-(Naphthalen-1-yl)-4-(naphthalen-1-ylmethylidene)-1,3-oxazol-5(4H)-one

open access: yesActa Crystallographica Section E, 2011
In the title compound, C24H15NO2, the oxazole ring is oriented at dihedral angles of 10.09 (4) and 6.04 (4)° with respect to the mean planes of the naphthalene ring systems, while the two naphthalene ring systems make a ...
Cevher Gündoğdu   +4 more
doaj   +1 more source

Synthesis and biological activities of the tris-oxazole macrolactone analogs of mycalolides [PDF]

open access: yes, 2012
Mycalolides are tris-oxazole macrolides isolated from the marine sponge Mycale sp., which shows cytotoxic, antifungal, and actin-depolymerizing activities. To develop an efficient synthetic route of mycalolides and to evaluate its functional mechanism of
Ishitsuka Tomoya   +8 more
core   +1 more source

Methylation‐Induced Permanent Charge Polarization in Covalent Organic Frameworks for Visible Light‐Driven Water Decontamination and Disinfection

open access: yesAdvanced Science, EarlyView.
A targeted in situ methylation strategy is developed to engineer cationic centers in a quinoline‐linked COF (NQ‐COFS1‐Me), creating a strong built‐in electric field, which effectively suppresses excitonic effects and promotes charge separation. The optimized material demonstrates powerful photocatalytic ROS generation for rapid bacterial inactivation ...
Xuewen Peng   +7 more
wiley   +1 more source

Recent advances in direct C–H arylation: Methodology, selectivity and mechanism in oxazole series

open access: yesBeilstein Journal of Organic Chemistry, 2011
Catalytic direct (hetero)arylation of (hetero)arenes is an attractive alternative to traditional Kumada, Stille, Negishi and Suzuki–Miyaura cross-coupling reactions, notably as it avoids the prior preparation and isolation of (hetero)arylmetals ...
Cécile Verrier   +6 more
doaj   +1 more source

Design, synthesis and biological evaluation of 3-(2-aminooxazol-5-yl)-2H-chromen-2-one derivatives

open access: yesChemistry Central Journal, 2018
Background In view of wide range of biological activities of oxazole, a new series of oxazole analogues was synthesized and its chemical structures were confirmed by spectral data (Proton/Carbon-NMR, IR, MS etc.). The synthesized oxazole derivatives were
Saloni Kakkar   +6 more
doaj   +1 more source

Design and Synthesis of Oxazoline-Based Scaffolds for Hybrid Lewis Acid/Lewis Base Catalysis of Carbon–Carbon Bond Formation [PDF]

open access: yes, 2016
A new class of hybrid Lewis acid/Lewis base catalysts has been designed and prepared with an initial objective of promoting stereoselective direct aldol reactions.
Benoit, Adam R.   +6 more
core   +1 more source

Home - About - Disclaimer - Privacy