Results 91 to 100 of about 5,322 (210)

Synthesis and biological evaluation of 4-(1H-imidazol-2-yl)-2-(pyrimidin-5-yl)oxazoles as potent anticancer agents

open access: yesResults in Chemistry
A new series of aryl derivatives of 4-(1H-imidazol-2-yl)-2-(pyrimidin-5-yl)oxazoles 11a–j were synthesised and their structures were characterized by analytical techniques.
Divya Komirishetti, Vasantha Mittapelli
doaj   +1 more source

A new route to functionalised oxazoles

open access: yes, 1996
Functionalised oxazoles 4 are prepared from amides 1 by rhodium cartenoid N-H insertion reaction to give beta-carbonyl amides 3 followed by cyclodehydration with triphenylphosphine-iodine-triethylamine.
Bagley, M C   +4 more
core   +2 more sources

Design, synthesis, molecular docking, anti-inflammatory and antioxidant activity of novel 2-(1-(4-(4-chlorophenyl)thiazol-2-yl)-1H-pyrazol-4-yl)benzo[d]oxazoles

open access: yesActa Chimica Slovenica
A series of novel 2-(1-(4-(4-chlorophenyl)thiazol-2-yl)-1H-pyrazol-4-yl)benzo[d]oxazoles 5 were synthesized from 2-[(E)-{1-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-1H-pyrazol-4-yl}(hydroxyimino)methyl]phenol 4 through Beckmann rearrangement.
Nirmala Darekar   +7 more
doaj   +1 more source

A Method for Iodination of Oxazoles at C-4 via 2-Lithiooxazoles

open access: yes, 2016
A Method for Iodination of Oxazoles at C-4 via 2 ...
Leza M. Luchetta (3045975)   +1 more
core   +1 more source

Reactions between Weinreb Amides and 2-Magnesiated Oxazoles:  A Simple and Efficient Preparation of 2-Acyl Oxazoles

open access: yes, 2016
Treatment of oxazole or 5-aryl oxazoles with i-PrMgCl smoothly generates the corresponding 2-Grignard reagents, which react with Weinreb amides to provide exclusively 2-acyl oxazole ...
Christopher M. Mapes (2250142)   +2 more
core   +1 more source

Síntesis de 3-amino-1,2-oxazoles y 3-amino-4,5-dihidro-1,2-oxazoles a partir de nitrilos α,β-insaturados y cetooximas

open access: yes, 2017
Se estudió la preparación general de 3-amino-1,2-oxazoles partiendo de nitrilos α,β-insaturados y cetooximas. Se aislaron y caracterizaron las oximas O-alquiladas resultantes de la reacción de adición y se estudió su conversión a los 3-amino-4,5-dihidro ...
Soria, Olivia   +4 more
core  

Reaction of Oxazoles with Dienophiles

open access: yesChemical and Pharmaceutical Bulletin, 1966
Naito, Takeo, Yoshikawa, Toru
openaire   +3 more sources

Modular Approach for Photoinduced Cycloaddition Enabling the Synthesis of Diverse Bioactive Oxazoles

open access: yes
The synthesis of bioactive oxazoles is often inefficient, and the reported methods remain largely unexplored for complex derivatives. To circumvent this issue, we have utilized a metal-free, photomediated [3 + 2] cycloaddition reaction between diazo ...
Ghosh, Ankan   +3 more
core   +1 more source

Home - About - Disclaimer - Privacy