Results 11 to 20 of about 126 (118)
Passerini-type reaction of boronic acids enables α-hydroxyketones synthesis
Multicomponent reactions enable the rapid construction of diverse molecular scaffolds with modularity and step economy. In this work, the authors report the use of boronic acids as carbon nucleophiles in a Passerini-type three-component coupling reaction
Kai Yang +5 more
doaj +1 more source
O‐Arylative Passerini Reactions. [PDF]
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
El Kaim, Laurent +2 more
openaire +2 more sources
A carboxylic acid, an aldehyde, and an isonitrile were combined in a single step (Passerini reaction) under mechanochemical activation to produce several α‐acyloxycarboxamide derivatives in high to excellent yields within 15 min of milling ...
Dr. Sodeeq Aderotimi Salami +3 more
doaj +1 more source
Plant-Derived Triterpenoid Functionalization: Synthesis of α-Acyloxycarboxamides
The application of isocyanide-based multicomponent reactions (IMCRs) for triterpenoid functionalization has been little reported. Triterpenoids and their derivatives are an important class of natural products of interest in medicinal chemistry due to ...
Fidel Rodriguez-Lopez +3 more
doaj +1 more source
The Biginelli reaction was combined with the Passerini reaction for the first time in a sequential multicomponent tandem reaction approach. After evaluation of all possible linker components and a suitable solvent system, highly functionalized ...
Andreas C. Boukis +2 more
doaj +1 more source
Synthesis of phosphorous analogues of tri- and tetra-depsipeptides 4 involving the Passerini reaction of diethylisocyanmethylphosphonate 3 with carbonyl compounds 2 and N-protected glycine 1 is reported.
Janusz Rachoń
doaj +1 more source
A series of γ-lactone derivatives (E)-4-arylidene-5-oxotetrahydrofuran derivatives were synthesized via a tandem Passerini 3CC/SN cyclization microwave-assisted one-pot method efficiently starting from Baylis Hillman acids, aryl glyoxals and isocyanides,
Yun Dong +11 more
doaj +1 more source
Efficient Synthesis of Boron-Containing α-Acyloxyamide Analogs via Microwave Irradiation
In this report, a Passerini three-component reaction utilizing boron-containing carboxylic acids or aldehydes is discussed. The reaction was carried out in water and facilitated by the use of microwave irradiation.
Po-Shen Pan +6 more
doaj +1 more source
In this report, 19 boron-containing depsipeptides were synthesized via microwave-assisted Passerini three-component reaction (P-3CR) in an aqueous environment.
Shuo-Bei Qiu +11 more
doaj +1 more source
Passerini Reactions on Biocatalytically Derived Chiral Azetidines [PDF]
The purpose of this study was to explore a series of Passerini reactions on a biocatalytically derived enantiopure azetidine-2-carboxyaldehyde in order to obtain, in a diastereoselective manner, polyfunctionalised derivatives having the potential to be cyclized to chiral bridged bicyclic nitrogen heterocycles.
MONI, LISA +6 more
openaire +3 more sources

