Results 161 to 170 of about 26,717 (273)

Antimicrobial activity of a short guanidine mimic immobilised on contact lenses. [PDF]

J Mater Sci Mater Med
Sara M, Kuppusamy R, Enninful G, Suresh D, Vasilev K, Mackenzie D, Dehghani F, Hui A, Wong EHH, Yasir M, Kumar N, Willcox M.   +11 more
europepmc   +1 more source

Tyr1-ψ[( Z)CF═CH]-Gly2 Fluorinated Peptidomimetic Improves Distribution and Metabolism Properties of Leu-Enkephalin.

ACS Chemical Neuroscience, 2018
Ryan A. Altman, K. Sharma, L. Rajewski, P. Toren, M. Baltezor, M. Pal, S. N. Karad   +6 more
semanticscholar   +1 more source

Thiazole peptidomimetics as chemical modulators of <i>KRAS</i> gene expression <i>via</i> G-quadruplex stabilization. [PDF]

RSC Chem Biol
Biswas D, Gorai A, Maiti S, Chaudhuri R, Pradhan S, Dash J.   +5 more
europepmc   +1 more source

Development of Peptidomimetic Inhibitors of the ERG Gene Fusion Product in Prostate Cancer.

Cancer Cell, 2017
Xiaoju Wang, Y. Qiao, I. Asangani, Bushra Ateeq, A. Poliakov, M. Cieslik, S. Pitchiaya, B. V. Chakravarthi, Xuhong Cao, Xiaojun Jing, Cynthia X Wang, I. Apel, Rui Wang, J. Tien, Kristin Juckette, Wei Yan, Hui Jiang, Shaomeng Wang, S. Varambally, A. Chinnaiyan   +19 more
semanticscholar   +1 more source

Integrated computational screen and validation of thalidomide-based PROTACs targeting SARS-CoV-2 main protease. [PDF]

RSC Med Chem
Guo LN, Li YH, Zhu RY, Su N, Shao ZY, Diao H.   +5 more
europepmc   +1 more source

Spectrum and activity of novel antimicrobial peptidomimetics [PDF]

, 2012
Hein-Kristensen, Line
core  

Functionalised peptidomimetic metallohelices [PDF]

Chapter 1 introduces small host-defence peptides in cancer therapy. The main mechanisms proposed in their interactions with membranes and intracellular targets are discussed. The biologically relevant peptide mimetics are also reviewed.\ud \ud Chapter 2 describes the synthesis and characterisation of alkyne derivatives of metallohelices.
openaire  

Structures of Zika virus NS2B‐NS3 protease in complex with peptidomimetic inhibitors

Antiviral Research, 2018
W. W. Phoo, Zhenzhen Zhang, M. Wirawan, E. Chew, Alvin Bing Liang Chew, Jenny Kouretova, T. Steinmetzer, D. Luo   +7 more
semanticscholar   +1 more source

AlphaFold-Guided Discovery of an Overlapping MYC/Miz-1 Interface Enables Peptidomimetic Disruption of MYC/MAX. [PDF]

ChemMedChem
Ellenbroek BD, Tirtosentono ASS, Pomplun SJ.   +2 more
europepmc   +1 more source

Ultrashort Cationic Self-assembled Peptides/Peptidomimetic Nanomaterials [PDF]

, 2014
Gilmore, B. F., Laverty, G., McCloskey, A. P.   +2 more
core