Synthesis of di(Imdazolium) and di(Pyrazolium) Salts as Precursors for N-heterocyclic Dicarbene Complexes [PDF]
, 2001 Alpha,omega-bis(pyrazol-1-yl)alkanes and alpha,omega-bis(imidazol-1-yl)alkanes with spacers consisting of four to ten methylene groups have been prepared from pyrazole, 3,5-dimethylpyrazole or imidazole and corresponding dibromoalkanes in a superbasic ...
Tatiana V. Goncharova +12 more
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Studies with Arylhydrazono-3-oxopropanals:A novel route to synthesis of substituted pyrazoles, oxoalkanonitrile and glyoxalonitrile containing sulfa drug moieties [PDF]
, 2008 Coupling of enaminones 1 with diazonium salts gave thehydrazonopropanals 3a-h. Compound 3 react with ω-bromoacetophenone or α-chloroacetanilide to yield 5 and 8. These compounds were cyclized smoothly into 6 and 9 respectively.
Abdel Hafiz, I.S. +4 more
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THE REACTIONS OF THE FORMAMIDINES. IX. THE SYNTHESIS OF 5-PHENYL-4-PYRAZOLE CARBOXYLIC ACID. [PDF]
, 1921 F. B. Dains, Wang Long
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Synthesis and biological evaluation of novel pyrazole derivatives as urease inhibitors [PDF]
, 2011 Studies on enzyme inhibition remain an important area of pharmaceutical research since these studies have led to the discoveries of drugs useful in a variety of physiological conditions.
Bole, S.B. +5 more
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Synthesis and biological evaluation of tetrahydropyridinepyrazoles ('PFPs') as inhibitors of STAT3 phosphorylation [PDF]
, 2013 The transcription factor STAT3 is constitutively overexpressed in many human tumors and hence represents a putative target for anticancer drug design. In this work, we describe the synthesis and biological evaluation of a novel chemotype, pyridine-fused ...
Andreas Bender, . +11 more
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Studies on Pyrazolones. X. Reactions of Pyrazole Blue with Cyanoacetamide and Malononitrile. [PDF]
, 1956 Gunnel Westöö +4 more
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SASH: Student Academic Showcase and Honors 2018 [PDF]
, 2017 A celebration of scholarship and creative activities for undergraduate and graduate students held in April, 2018 at the Roger Williams University campus in Bristol, Rhode ...
Roger Williams University
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Co-crystalization and in vitro biological characterization of 5-Aryl-4-(5-substituted-2-4-dihydroxyphenyl)-1,2,3-thiadiazole Hsp90 inhibitors [PDF]
, 2012 A potential therapeutic strategy for targeting cancer that has gained much interest is the inhibition of the ATP binding and ATPase activity of the molecular chaperone Hsp90.
Chrisostomos Prodromou +7 more
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Pyrazole Studies. XI. Oxidation by Air of 1:4-Disubstituted Pyrazolidine-3:5-diones. [PDF]
, 1958 Stig Veibel +5 more
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