Thiazole-induced rigidification in substituted dithieno-tetrathiafulvalene: The effect of planarisation on charge transport properties [PDF]
, 2015 © 2015 Taylor et al; licensee Beilstein-Institut.Two novel tetrathiafulvalene (TTF) containing compounds 1 and 2 have been synthesised via a four-fold Stille coupling between a tetrabromo-dithienoTTF 5 and stannylated thiophene 6 or thiazole 4.
Olena Avramchenko (7163237) +8 more
core +9 more sources
Synthesis and Biological Evaluation of 2-Aminothiazole Analogues of Nα-Protected Amino Acids [PDF]
Iranian Journal of Chemistry & Chemical Engineering, 2023 Synthesis of 2-amino-thiazoles from Nα-protected bromomethyl ketones obtained from Nα-protected diazomethyl ketones has been reported in this study.N-protected amino acids were converted to diazomethylketones using (Benzotriazol-1-yloxy) tris ...
Lalithamba Haraluru Shankaraiah +3 more
doaj +1 more source
Synthesis of Thiazole-2(3H)-thiones as Antimicrobial Agents Promoted by H3PW12O40-amino-functionalized CdFe12O19@SiO2 Nanocomposite [PDF]
Nanochemistry Research, 2022 H3PW12O40-amino-functionalized CdFe12O19@SiO2 nanocomposite has been utilized as an effective nanocatalyst for the preparation of thiazole-2(3H)-thiones by three-component reactions of CS2, 2-bromoacetophenone or 2-bromo-1-(4-methoxyphenyl) ethenone, and
Hossein Shahbazi-Alavi +1 more
doaj +1 more source
Synthesis and Structural Confirmation of the Thiazole Alkaloids Derived from Peganum harmala L.
Applied Sciences, 2021 Peganumal A and B are thiazole alkaloids isolated from the seeds of Peganum harmala L. Thiazole moieties are rarely found in natural products, but diverse compounds possessing thiazole moieties have attracted attention owing to their broad range of ...
Myeonghyeon Sim +2 more
doaj +1 more source
5-Chloro-6-oxo-6H-xantheno[4,3-d]thiazole-2-carbonitrile
Molbank, 2022 Xanthones and benzothiazoles are important classes of heterocyclic compounds with versatile biological activities. Herein, we describe a straightforward and scalable synthesis of 5-chloro-6-oxo-6H-xantheno[4,3-d]thiazole-2-carbonitrile, a thiazole-fused ...
Konstantinos Paraskevas +3 more
doaj +1 more source
In Vitro Inhibition Effects of 2-Amino Thiazole Derivatives on Lactoperoxidase Enzyme Activity
Cumhuriyet Science Journal, 2022 Lactoperoxidase (LPO E.C. 1.11.1.7) is a member of the peroxidase family and is an important glycoprotein containing heme group in its structure and showing the antimicrobial effect on disease causing microorganisms in the digestive system of newborn ...
Işıl Nihan Korkmaz
doaj +1 more source
Molecules, 2022 For many decades, the thiazole moiety has been an important heterocycle in the world of chemistry. The thiazole ring consists of sulfur and nitrogen in such a fashion that the pi (π) electrons are free to move from one bond to other bonds rendering ...
Mohammed F. Arshad +15 more
doaj +1 more source
Azole γ-Peptides Helix Switching via Heterocycle Substitutions. [PDF]
Angew Chem Int Ed EnglHeterocycle substitution in azole‐based γ‐amino acids enables control over the helical shape of heterocyclic γ‐peptides. S↔N permutation in thiazole residues switches a canonical 9‐helix into a flexible helix exhibiting discontinuous hydrogen bonding.
Chaise S +10 more
europepmc +3 more sources
Thiazole antibiotics target FoxM1 and induce apoptosis in human cancer cells. [PDF]
PLoS ONE, 2009 Forkhead box M1 (FoxM1) oncogenic transcription factor represents an attractive therapeutic target in the fight against cancer, because it is overexpressed in a majority of human tumors.
Uppoor G Bhat +2 more
doaj +1 more source
Ranking ligand affinity for the DNA minor groove by experiment and simulation [PDF]
, 2010 The structural and thermodynamic basis for the strength and selectivity of the interactions of minor-groove binders (MGBs) with DNA is not fully understood.
Wittayanarakul, Kitiyaporn +8 more
core +4 more sources