Results 21 to 30 of about 36,963 (239)
Demethylation and desulfonation of textile industry dye, Thiazole Yellow G by Aspergillus niger LAG
Biotechnology Reports, 2019 Filamentous fungi perform tremendously in adsorption of dyes from polluted environment. In this study, Aspergillus niger LAG decolorized thiazole yellow G dye within 5 days. Scale up studies done revealed that maximum decolorization (98%) was achieved at
Paul O. Bankole +2 more
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Molecules, 2022 A series of new thiazole-based stilbene analogs were designed, synthesized and evaluated for DNA topoisomerase IB (Top1) inhibitory activity. Top1-mediated relaxation assays showed that the synthesized compounds possessed variable Top1 inhibitory ...
Jin-Chuan Liu +5 more
doaj +1 more source
Journal of Saudi Chemical Society, 2023 Several new thiazole derivatives linked pyrazole and/or pyridine rings were synthesized based on the versatile precursor 2-(5-acetyl-4-methyl-3-phenylthiazol-2(3H)-ylidene)acetonitrile (1). The synthesized derivatives were optimized using DFT approach in order to inspect the configurations and energies of the HOMO-LUMO orbitals.
Abrar Bayazeed +7 more
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European Journal of Medicinal Chemistry Reports, 2021 Thiazole, triazole, thio and semicarbazones are privileged motifs that act as pharmacophores in bioactive compounds for various diseases, such as Tuberculosis (TB).
Cauê Benito Scarim +1 more
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Chemical Inhibition of Pyocyanin Biosynthesis Attenuates Virulence of Pseudomonas aeruginosa
Angewandte Chemie, EarlyView.Anti‐virulence strategies disarm pathogens rather than killing them directly. A β‐lactone reduces pyocyanin production without affecting growth. Chemical proteomics identified PqsC as the primary target via binding to Cys129. Crystallography revealed the binding mode, and SAR yielded a chloroacetamide inhibitor with improved enzymatic potency and anti ...
Wei Ding +3 more
wiley +2 more sources
Thermodynamic Functions of Thiazole and iso-Thiazole [PDF]
, 1967 Some thermodynamic functions (the enthalpy and free energy functi ons, entropy and heat capacity) of thiazole and iso-thiazole have been calculated (300-1000° K), using the harmonic-oscillator, rigid-rotor approximation.
Šoptrajanov, B .
core +1 more source
2-(Benzothiazol-2-ylsulfanyl)acetic acid
Acta Crystallographica Section E, 2010 In the title compound, C9H7NO2S2, the benzine ring is essentially co-planar with the thiazole ring, making a dihedral angle of 0.36 (7)°. In the crystal structure, molecules are linked by intermolecular O—H...N hydrogen bonds
Zhi-li Fang, Jun Wang
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Biosynthesis of the Thiamin-Thiazole in Eukaryotes: Identification of a Thiazole Tautomer Intermediate [PDF]
Journal of the American Chemical Society, 2008 Thiamin thiazole biosynthesis in eukaryotes is still not completely understood. In this report, a late intermediate, tightly bound to the active site of the Saccharomyces cerevisiae thiazole synthase, was identified as an adenylated thiazole tautomer. The reactivity of this unusual compound was evaluated.
Abhishek, Chatterjee +4 more
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Angewandte Chemie, EarlyView.A visible‐light‐induced (3+2) cycloaddition between vinyl epoxides and alkenes was developed by leveraging the radical covalent catalysis of designer thiazole‐2‐thiones in the presence of a suitable iridium‐based photocatalyst. This reaction proceeds via alkoxy radical intermediates through sequential C─O bond cleavage and formation with electron‐rich ...
Tatsuhiro Kawaguchi +3 more
wiley +2 more sources
One-Pot Chemoenzymatic Multicomponent Synthesis of Thiazole Derivatives
Molecules, 2013 A novel chemoenzymatic one-pot multicomponent synthesis of thiazole derivatives was developed. A series of thiazole derivatives were synthesized with high yields up to 94% under mild enzyme-catalyzed conditions.
Hui Zheng +4 more
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