Results 61 to 70 of about 35,784 (226)
SYNTHESIS OF SOME NEW 2,4,6-TRISUBSTITUTEDTHIAZOLO-[5,4-d] PYRIMIDINE-5,7(4H,6H)-DIONES.
Zagazig Journal of Pharmaceutical Sciences, 1999 Reaction of 2,6-disubstitutedthiazolo5,4-dpyrimidin-7(6H)-ones 2 with ethyl chloroformate/ethanol mixture afforded 5-(ethoxycarbonylamino) -2-(substitutedthio) thiazole-4-(N-substituted)-carboxamides 4a-c.
Wahid Basyouni , Hanaa Hosni
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4-[Bis(thiazol-2-ylamino)methyl]phenol
Molbank, 2023 We have designed and synthesized novel bis-thiazole derivative. A 4-[bis(thiazol-2-ylamino)methyl]phenol was efficiently prepared in 71% yield by the reaction of 2-aminothiazole with 4-hydroxybenzaldehyde in ethanol for 24 h.
Joanna Cytarska, Anna Kolasa
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Antioxidants, 2023 The aim of the present research was to obtain a supramolecular complex between a strong antioxidant compound previously reported by our group, in order to extend its antioxidant activity.
Mihaela Mic +5 more
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Enhancing α7 nAChR function serves as a therapeutic strategy for cognitive disorders. Here, we report the synthesis and evaluation of 2-arylamino-thiazole-5-carboxylic acid amide derivatives 6–9 that as positive allosteric modulators (PAMs) activate ...
Han Wang (254423) +17 more
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A comprehensive review on thiazole derivatives as multifunctional therapeutics
Discover ChemistryThiazole, a versatile five-membered heterocyclic scaffold containing sulfur and nitrogen atoms, has emerged as a pivotal pharmacophore in medicinal chemistry due to its unique chemical properties and broad spectrum of biological activities.
Dattatray N. Thorat +5 more
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Acta Crystallographica Section E: Crystallographic Communications, 2020 The asymmetric unit of the title compound, C23H20N2OS, contains one slightly bent molecule. The naphthalene ring system and the thiazole ring are twisted with respect to each other, making a dihedral angle of 13.69 (10)°; the anisole ring is inclined to ...
Ropak A. Sheakh Mohamad +2 more
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Enantiomeric Separation of New Chiral Azole Compounds
Molecules, 2021 Twelve new azole compounds were synthesized through an ene reaction involving methylidene heterocycles and phenylmaleimide, producing four oxazoles, five thiazoles, and one pyridine derivative, and ethyl glyoxylate for an oxazole and a thiazole compound.
Marziyeh E. Kenari +9 more
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Thermodynamic Functions of Thiazole and iso-Thiazole [PDF]
, 1967 Some thermodynamic functions (the enthalpy and free energy functi ons, entropy and heat capacity) of thiazole and iso-thiazole have been calculated (300-1000° K), using the harmonic-oscillator, rigid-rotor approximation.
Šoptrajanov, B .
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Synthesis of oligonucleotides containing thiazole and thiazole N-oxide nucleobases
, 2002 [reaction: see text] The thiazole C-nucleoside analogue was synthesized by the Hantzsch cyclization method to form the thiazole ring and was then converted to the thiazole N-oxide C-nucleoside analogue by peracid oxidation of the heterocycle nitrogen ...
Fronczek, Frank R +6 more
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Molecules, 2007 A series of eight new azomethine derivatives were synthesized by reacting 2-formylphenoxyacetic acid with aromatic amines. The chemical structures of these compounds were confirmed by means of 1H-NMR, 13C-NMR, MS and elemental analysis.
George W. Weaver +4 more
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