Results 151 to 160 of about 1,246 (203)

On-Resin Synthesis and Late-Stage Functionalization of Macrocyclic Atosiban Mimetics via 5-Iodo-1,4-triazoles. [PDF]

Org Lett
Shepperson OA, Malone MA, Arnott KIM, Brown RJ, Jamieson AG.   +4 more
europepmc   +1 more source

Exploring novel Apalutamide analogues as potential therapeutics for prostate cancer: design, molecular docking investigations and molecular dynamics simulation. [PDF]

Front Chem
Gupta AK, Vaishnav Y, Jain SK, Annadurai S, Kumar N.   +4 more
europepmc   +1 more source

<i>In silico</i> targeting of <i>Enterococcus faecalis</i> proteins in endodontic infections: A systematic review. [PDF]

J Conserv Dent Endod
Geervani VS, Neelakantappa KK, Merwade S, Kumar RSM, Abhishek M, Manimozhi M.   +5 more
europepmc   +1 more source

Synthesis of Thiohydantoin. III

Synthesis of Thiohydantoin. III
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Solid-phase synthesis of branched thiohydantoin benzimidazolinethiones and branched thiohydantoin tetrahydroquinoxalinediones

Tetrahedron Letters, 2000
Abstract An efficient solid-phase synthesis method is described for branched thiohydantoin benzimidazolinethiones and branched thiohydantoin tetrahydroquinoxalinediones using 4-fluoro-3-nitrobenzoic acid.
Adel Nefzi, Marc A Giulianotti
exaly   +2 more sources

Thiohydantoin Nucleosides. Synthesis Approaches

Monatshefte Für Chemie, 2004
AbstractFor Abstract see ChemInform Abstract in Full Text.
Ahmed I Khodair, El Sayed H El Ashry, Najim A Al-Masoudi   +2 more
exaly   +2 more sources

Recent applications of hydantoin and thiohydantoin in medicinal chemistry

European Journal of Medicinal Chemistry, 2019
Hydantoin, imidazolidine-2,4-dione, is a non-aromatic five-membered heterocycle, which is considered a valuable, privileged scaffold in medicinal chemistry. The importance of the hydantoin scaffold in drug discovery has been reinforced by several medicines in clinical use, such as phenytoin, nitrofurantoin, and enzalutamide.
Seok-Ho Kim, Dongyun Shin
exaly   +3 more sources

Design, synthesis and evaluation of thiohydantoin derivatives as potent topoisomerase I (Top1) inhibitors with anticancer activity

European Journal of Medicinal Chemistry, 2015
DNA topoisomerase I is a potential chemotherapeutic target. Here, we designed and synthesized a library comprising of hydantoin and thiohydantoin derivatives and tested them against human and Leishmania Top1.
Chandramohan Bathula, Subhendu K Das, Rahul Agarwal   +2 more
exaly   +2 more sources

Crystal Structures and Conformations of 5-Benzyl-2-thiohydantoin and Its 1-Acetylated Derivative

Spectroscopy Letters, 2009
The crystal structures of 5-benzyl-2-thiohydantoin (5-BTH) and 1-acetyl-5-benzyl-2-thiohydantoin (1-Ac-5-BTH) have been determined by X-ray diffraction.
Ko-Ki Kunimoto, Soh-Ichi Kitoh, Akio Kuwae   +2 more
exaly   +3 more sources

Novel and efficient protocol for the syntheses of N-1 substituted thiohydantoin and a bicyclothiohydantoin under solvent-free conditions

Tetrahedron Letters, 2012
A novel approach for the synthesis of N-1 substituted thiohydantoin has been developed to give quantitative yields of the desired products. The efficient synthesis of bis-thiohydantoin derivative and bicyclothiohydantoin has extended scope and ...
M P Kaushik
exaly   +2 more sources