Results 91 to 100 of about 8,698 (205)

Effects of a Thiosemicarbazide Camphene Derivative on Trichophyton mentagrophytes

Molecules, 2009
Thiosemicarbazides are compounds known for their biological activity, particularly their antimicrobial properties, which include activity against fungi.
Cleuza Conceição da Silva, Benedito Prado Dias Filho, Tânia Ueda-Nakamura, Ana Paula Barbosa da Silva, Mirian Ueda Yamaguchi, Celso Vataru Nakamura   +5 more
doaj   +1 more source

Synthesis, antitubercular activity and mechanism of resistance of highly effective thiacetazone analogues [PDF]

, 2013
Defining the pharmacological target(s) of currently used drugs and developing new analogues with greater potency are both important aspects of the search for agents that are effective against drug-sensitive and drug-resistant Mycobacterium tuberculosis ...
A Alahari, A Alahari, A Banerjee, A Bhatt, AE Grzegorzewicz, AK Ojha, AR Baulard, C Vilcheze, CK Stover, D Fegan, D Fegan, Derek Craig, E Dubnau, E Sacco, Emilie Vialla, F Wang, FM Shahab, G Lutfalla, Geoffrey D. Coxon, JA Caminero, Jean Louis Herrmann, JM Belardinelli, JR Wei, K Takayama, L Kremer, Laila Gannoun-Zaki, Laurent Kremer, LE Bermudez, LG Dover, LS Kremer, MA Espinal, MS Glickman, N Slama, P Nunn, PT Davidson, R Mondal, R Veyron-Churlet, R Veyron-Churlet, RM Corrales, Rosa Milagros Corrales, S Cantaloube, TD Bugg, V Rao, VK Sambandamurthy, Y Rombouts   +44 more
core   +3 more sources

Synthetic Strategies to Access Fluorinated Azoles

European Journal of Organic Chemistry, Volume 28, Issue 47, December 15, 2025.
This review highlights recent synthetic strategies for introducing fluorine groups (mono‐, di‐, and trifluoromethylation) into 11 major azole classes, identifying research gaps to inform future innovations in materials science, medicinal chemistry, and biomedical research.
Mohammed K. Abd El‐Gaber, Mario Djugovski, Tzu‐Yu Huang, Sweta Adhikari, Sudeshna Roy   +4 more
wiley   +1 more source

Design, Synthesis, In Silico Absorption, Distribution, Metabolism, and Elimination and Molecular Docking Studies of Thiazole‐Based Furan Derivatives, and Their Biological Evaluation for Alzheimer Disease Therapy

ChemistryOpen, Volume 14, Issue 12, December 2025.
GA: Oxidative stress plays a critical role in Alzheimer's disease (AD) by promoting Aβ plaque accumulation and tau pathology, accelerating neurodegeneration. Elevated reactive oxygen species contribute to cognitive decline through extensive oxidative damage.
Abdüllatif Karakaya, Ulviye Acar Çevik, Betül Kaya, Bilge Çiftçi, Adem Necip, Mesut Işık, Şükrü Beydemir, Yusuf Özkay, Zafer Asım Kaplancıklı   +8 more
wiley   +1 more source

(3aR,6R)-3,3,6-Trimethyl-3,3a,4,5,6,7-hexahydro-2H-indazole-2-carbothioamide

IUCrData, 2016
The title compound, C11H19N3S, was prepared by the reaction of (R)-pulegone with thiosemicarbazide in acidic medium, using ethanol as solvent. The molecule is built up from fused six and five-membered rings.
Abdellah N'Ait Ousidi, My Youssef Ait Itto, Aziz Auhmani, Abdelkhalek Riahi, Sylviane Chevreux, Moha Berraho   +5 more
doaj   +1 more source

Enhancing Open‐Circuit Voltage and Fill Factor in Sn‐Based Perovskite Solar Cells: Challenges and Opportunities for Sustainable Photovoltaics

SusMat, Volume 5, Issue 6, December 2025.
This review summarizes advances in tin (Sn)‐based perovskite solar cells, a promising lead‐free alternative. It examines the main causes of Voc and fill factor losses, including Sn2+ oxidation, undercoordinated sites, and deep‐level traps. Strategies such as molecular coordination, surface passivation, compositional tuning, interface engineering, and ...
Padmini Pandey, Jun Ryu, Han‐Gyun Lim, Jincheol Kim, Dong‐Won Kang   +4 more
wiley   +1 more source

3-(4-Bromophenyl)-1-carbamothioyl-5-(2-carbamothioylhydrazinyl)-4,5-dihydro-1H-pyrazole-5-carboxylic Acid

Molbank
The reaction of 4-(4-bromophenyl)-2,4-dioxobutanoic acid with thiosemicarbazide, in a ratio of 1:2, when boiled in ethanol gives 3-(4-bromophenyl)-1-carbamothioyl-5-(2-carbamothioylhydrazinyl)-4,5-dihydro-1H-pyrazole-5-carboxylic acid with a good yield ...
Anastasia A. Andreeva, Maksim V. Dmitriev, Andrey N. Maslivets   +2 more
doaj   +1 more source

Copper(II) Complexes with Highly Water-Soluble L- and D-Proline Thiosemicarbazone Conjugates as Potential Inhibitors of Topoisomerase IIα [PDF]

, 2013
Two proline-thiosemicarbazone bioconjugates with excellent aqueous solubility, namely 3-methyl-(S)-pyrrolidine-2-carboxylate-2-formylpyridine thiosemicarbazone (L-Pro-FTSC or (S)-H2L) and 3-methyl-(R)-pyrrolidine-2-carboxylate-2-formylpyridine ...
Arion Vladimir B., Bacher Felix, Bognár Gabriella M., Enyedy Éva Anna, Kiss Tamás, Klapproth Erik, Nagy Nóra Veronika, Novak Maria S., Rockenbauer Antal, Trondl Robert   +9 more
core   +1 more source

1,2-Dibenzoylthiosemicarbazide

Molbank
When 1-benzoylthiosemicarbazide (2) or thiosemicarbazide (1) were treated with benzoyl chloride in a basic medium, a mixture of two compounds was obtained: 1,2-dibenzoylthiosemicarbazide (3) and 1,4-dibenzoylthiosemicarbazide (4).
Burcă Ion, Badea Valentin, Todea Anamaria, Bercean Vasile-Nicolae   +3 more
doaj   +1 more source

Design, Synthesis, and Fungicidal Activity of Novel Thiosemicarbazide Derivatives Containing Piperidine Fragments

Molecules, 2017
In order to discover novel eco-friendly lead compounds for plant pathogenic fungi control, a series of benzaldehyde thiosemicarbazide derivatives with a piperidine moiety have been designed and synthesized.
Xuebo Zhang, Peng Lei, Tengda Sun, Xiaoyu Jin, Xinling Yang, Yun Ling   +5 more
doaj   +1 more source