Results 121 to 130 of about 19,712 (214)

Expeditious synthesis and biological evaluation of new C-6 1,2,3-triazole adenosine derivatives A1 receptor antagonists or agonists.

, 2010
International audienceThe synthesis of new C-6 1,2,3-triazole adenosine derivatives via microwave assisted 1,3-dipolar cycloaddition as key step is described.
Attolini, Mireille, Berthault, Aurélie, By, Youlet, Carrega, Louis, Chouraqui, Gaëlle, Commeiras, Laurent, Condo, Jocelyne, Gaudel-Siri, Anouk, Guieu, Régis, Mathew, Smitha C, Parrain, Jean-Luc, Rodriguez, Jean, Ruf, Jean, Virolleaud, Marie-Alice   +13 more
core   +5 more sources

Synthèse, dérivation et évaluation de pharmacophores hybrides Alcynyl-TriAzolyCarbinols N-glycosylés [PDF]

, 2014
La fonction alcényl-alcynylcarbinol (AAC) est un pharmacophore clé rencontré dans des produits naturels extraits d'éponges marines, les pétrosiacétylènes, aux propriétés biologiques multiples, en particulier une cytotoxicité remarquable sur les cellules ...
Oukessou, Mohamed
core  

Cycloaddition reactions of heterocyclic azides with 2-cyanoacetamidines as a new route to C,N-diheteroarylcarbamidines

Beilstein Journal of Organic Chemistry
A novel and efficient base-catalyzed, transition-metal-free method for the synthesis of diheterocyclic compounds connected by an amidine linker, including apart from the common 1,2,3-triazole ring, either an additional pyrimidinedione, 4-nitroimidazole ...
Pavel S. Silaichev, Tetyana V. Beryozkina, Vsevolod V. Melekhin, Valeriy O. Filimonov, Andrey N. Maslivets, Vladimir G. Ilkin, Wim Dehaen, Vasiliy A. Bakulev   +7 more
doaj   +1 more source

Current progress of 1,2,3-triazole hybrids as EGFR inhibitors for cancer therapy - a literature review. [PDF]

RSC Adv
Khasawneh HEN, Hassan HM, Alharbi AA, Almagharbeh WT, Al-Aouadi RFA, Kaur K, Maranan R, Farhan HM, Hashem H, Hassan MM, Bräse S, Al-Emam A.   +11 more
europepmc   +1 more source

Mitochondrial Dysfunction Induced by a Novel Salicylate-Based 1,2,3-Triazole Salt With Potent Antileishmanial Activity. [PDF]

Chem Biol Drug Des
De Oliveira BA, de Oliveira Lemos AS, Bastos JPRC, Antinarelli LMR, de Freitas ALR, Ribeiro RGM, da Silva Neto AF, Coimbra ES, Da Silva AD.   +8 more
europepmc   +1 more source

Design, Synthesis and Antiproliferative Activity Studies of Novel 1,2,3-Triazole-Urea Hybrids. [PDF]

Drug Des Devel Ther
Gao E, Zhang H, Guo Y, Wang X, Mao L, Peng L, Xu G, Yao X, Li S, Long H, Wang T, Wu H.   +11 more
europepmc   +1 more source

New Copper (II) Complexes Based on 1,4-Disubstituted-1,2,3-Triazole Ligands with Promising Antileishmanial Activity. [PDF]

Pharmaceutics
Nascimento JPC, Faganello NL, Freitas KF, Pinto LMC, das Neves AR, Carvalho DB, Arruda CCP, Silva SM, Almeida RCF, Júnior AM, Back DF, Pizzuti L, Saba S, Rafique J, Baroni ACM, Casagrande GA.   +15 more
europepmc   +1 more source

Anticoronavirus Activity of Uridine Glycoconjugates Containing a 1,2,3-Triazole Moiety. [PDF]

J Med Chem
Graul M, Brzuska G, Wisniewska E, Dominska M, Strakova P, Ruzek D, Pastuch-Gawolek G, Krol E.   +7 more
europepmc   +1 more source

Highly Stable and Active Catalyst for Sabatier Reactions [PDF]

Highly active Ru/TiO2 catalysts for Sabatier reaction have been developed. The catalysts have shown to be stable under repeated shutting down/startup conditions.
Brooks, Kriston P., Hu, Jianli
core   +1 more source

Design and synthesis of 1,2,3-triazole thiadiazole hybrids with in vitro and in silico evaluation of their anti-inflammatory and anti-alzheimer activities. [PDF]

Sci Rep
Rabee AR, Abdel-Hamid H, Soliman SM, Ashraf S, Sobhy AA, Ghareeb DA, Saad AK, Hagar M.   +7 more
europepmc   +1 more source