Convenient procedure for in situ cyclization of hydrazinecarbodithioate potassium salts to 1,3,4-oxadiazole-2(3H)-thiones under normal phase micellar media catalysis promoted by sodium dodecyl sulfate (SDS) as an anionic surfactant is reported.
Ayhan YILDIRIM
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Recent advancements in oxadiazole-based anticancer agents [PDF]
Oxadiazole ring system occupies a significant position among heterocyclic templates for medicinal compounds due to its wide spectrum of biological activities.
Ahmad, Matloob +6 more
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Synthesis, characterization and antioxidant activity of 1,3,4-oxadiazoles bearing an indole ring [PDF]
1,3,4-oxadiazoles have been widely studied by many researchers in various fields. Due to its heterocyclic structure, 1,3,4-oxadiazoles possess of many biological and pharmacological activities such as antibacterial, anticancer, antiinflammatory ...
Kong, Kian Liang
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Synthesis, Reactions and Antioxidant Activity of 5-(3', 4'-dihydroxy-tetrahydrofuran-2'-yl)-2-methyl-3-carbohydrazide [PDF]
In this manuscript, we describe the synthesis of the carbohydrazide 2. Acid-catalyzed condensation with several carbonyl compounds to afford the corresponding carbohydrazide derivatives 3-12.
Mohamed El Sadek +4 more
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Efficient synthesis of new oxadiazole-thiazole hybrids using (diacetoxyiodo)benzene [PDF]
85-92An efficient synthesis of some new 2-aryl-5-(2'-(4-nitrophenylamino)thiazol-4'-yl)-1,3,4-oxadiazoles 7a-e, has been accomplished through oxidative cyclization of 2-(4-nitrophenylamino)-N'-(substituted benzylidene) thiazole-4-carbohydrazides 6a-e ...
Aggarwal, Ranjana +2 more
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Synthetic Approaches to 1,3,4-Oxadiazole-Containing Boronic Derivatives
1,3,4-Oxadiazoles containing boronic acid moieties are promising as a highly versatile class of compounds with significant utility across various scientific domains.
Barbara Wołek, Agnieszka Kudelko
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Cross Linking and Degradation Mechanisms in Model Sealant Candidates [PDF]
Model compounds were investigated as to which type of heterocyclic ring is the most advantageous for curing sealants based on perfluoroalkylether chains. The relative thermal, thermal oxidative, hydrolytic, and fuel stability of potential crosslinks were
Ito, T. I. +4 more
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Biological evaluation of 1,3,4-oxadiazoles bis-substitute derivatives as potential anticancer agents [PDF]
Cancer is a major health problem and causes substantial morbidity and mortality worldwide.In order to identify new potent antitumor agents with good specificity and low toxicity, a series of 12 new 1,3,4-oxadiazole bis-substitute molecules were tested on
NIEDDU, Valentina
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Toxicological Evaluation of Anti-Scrapie Trimethoxychalcones and Oxadiazoles
An altered form of the cellular prion protein, the PrPScor PrPRes, is implicated in the occurrence of the still untreatable transmissible spongiform encephalopathies.
CLAUDIA P. FIGUEIREDO +10 more
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2-(5-[4-диметиламинофенил]-2-оксазолил)-бензойная кислота как флуоресцентный сенсор влаги в органических растворителях [PDF]
Проведен сравнительный анализ спектрально-люминесцентных свойств синтезированой 2-(5-[4-ди-метиламинофенил]-2-оксазолил)-бензойной кислоты в предварительно осушенных органических растворителях разной полярности.
Вульфова, Д.А. +4 more
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