Results 91 to 100 of about 1,413 (178)

Design, Synthesis, and Structure-Activity Relationship Studies of (4-Alkoxyphenyl)glycinamides and Bioisosteric 1,3,4-Oxadiazoles as GPR88 Agonists. [PDF]

J Med Chem, 2020
Rahman MT, Decker AM, Langston TL, Mathews KM, Laudermilk L, Maitra R, Ma W, Darcq E, Kieffer BL, Jin C.   +9 more
europepmc   +1 more source

A novel and sustainable synthesis-functionalization strategy for the oxidative cyclization towards 2,5-disubstituted-1,3,4-oxadiazoles using bentonite-supported copper(i) iodide as a green catalyst. [PDF]

RSC Adv
Tran VQ, Tran DM, Tran MH, Tran PH, Nguyen HT.   +4 more
europepmc   +1 more source

SYNTHESIS OF 1,3,4-OXADIAZOLES AS SELECTIVE T-TYPE CALCIUM CHANNEL INHIBITORS. [PDF]

Heterocycles, 2020
Zhang M, Zou B, Gunaratna MJ, Weerasekara S, Tong Z, Nguyen TDT, Koldas S, Cao WS, Pascual C, Xie XS, Hua DH.   +10 more
europepmc   +1 more source

2:1 Adducts Arising from Reactions between Benzynes and 1,3,4-Oxadiazoles. [PDF]

Org Lett
Guzman AL, Kevorkian PV, Hoye TR.
europepmc   +1 more source

In Vitro and In Silico Evaluation of Anticancer Activity of New Indole-Based 1,3,4-Oxadiazoles as EGFR and COX-2 Inhibitors. [PDF]

Molecules, 2020
Sever B, Altıntop MD, Özdemir A, Akalın Çiftçi G, Ellakwa DE, Ellakwa DE, Tateishi H, Radwan MO, Ibrahim MAA, Otsuka M, Fujita M, Ciftci HI, Ali TFS.   +12 more
europepmc   +1 more source

Molecular Docking and In Vitro Studies of Synthesized Oxadiazole Derivatives as Urease Inhibitors

Journal of Mathematical and Fundamental Sciences
A novel sequence of 1,3,4-oxadiazoles (7a–h) was synthesized. The compounds were characterized by IR, ¹H NMR, and MS analyses. They were also examined to determine whether they could prevent urease from functioning.
Kamran Mehdi, Obaid-ur-Rahman Abid, Saqib Khan, Is Helianti, Muhammad Ikhlas Abdjan, Aleesha Aleesha, Muhammad Ali, Naseer Ahmed   +7 more
doaj  

2-(Difluoromethyl)-1,3,4-oxadiazoles: The Future of Selective Histone Deacetylase 6 Modulation? [PDF]

ACS Pharmacol Transl Sci
König B, Hansen FK.
europepmc   +1 more source

Synthesis of 1,3,4-oxadiazoles derivatives with antidepressant activity and their binding to the 5-HT_1A receptor. [PDF]

RSC Adv, 2020
Wang S, Qi L, Liu H, Lei K, Wang X, Liu R.   +5 more
europepmc   +1 more source

1,3,4-oxadiazoles as inhibitors of the atypical member of the BET family bromodomain factor 3 from Trypanosoma cruzi (TcBDF3). [PDF]

Front Microbiol
Alonso VL, Escalante AM, Rodríguez Araya E, Frattini G, Tavernelli LE, Moreno DM, Furlan RLE, Serra E.   +7 more
europepmc   +1 more source

Efficient Synthesis of Novel 1,3,4-Oxadiazoles Bearing a 4-N,N-Dimethylaminoquinazoline Scaffold via Palladium-Catalyzed Suzuki Cross-Coupling Reactions. [PDF]

Molecules, 2020
Wołek B, Werłos M, Komander M, Kudelko A.   +3 more
europepmc   +1 more source