Synthesis and biological activity of 5-nitrofuran-containing (1,3,4-thiadiazol-2-yl)piperazine moieties as a new type of anti-Helicobacter pylori heterocycles [PDF]
Journal of the Serbian Chemical Society, 2011 In order to find new and potent drug candidates for the treatment of Helicobacter pylori infections‚ in this study attention was focused on the synthesis and anti-H.
ABBAS SHAFIEE +10 more
doaj
Molecules, 2002 3-(2-Furanyl)-4-amino-5-mercapto-1,2,4-triazole (1) was prepared from 2-furoic acid through a multi-step reaction sequence. Compound 1 reacted with aromatic acids in the presence of phosphorus oxychloride to give 3-(2-furanyl)-6-aryl-1,2,4-triazolo[3,4-b]
Zi-Yi Zhang +6 more
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One- Pot synthesis and reactions of Novel 5-(4-fluoro-phenyl)-3-(8-hydroxyquinolin-5- yl)-7-phenyl-5H-thiazolo[3,2-a]pyrimidine-6- carbonitrile as antimicrobial agents [PDF]
, 2018 The synthesis of 5-(4-fluoro-phenyl)-3-(8-hydroxyquinolin-5-yl)-7-phenyl-5H-thiazolo[3,2-a]pyrimidine-6-carbonitrile 4 was achieved by one-potthree-component synthesis using p-TSA (10 mol %) in refluxing CH3CN.
Abdelmohsen, S.A.
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Annals of Mechnikov's Institute, 2020 Introduction: The analysis of modern literature, including overseas one, showed that a lot of the scientific researches is devoted to finding and creating biologically active compounds on base 1,3,4-thiadiazole.
I Sych, L Perekhoda, Z Іеremina
doaj
Chemistry Central Journal, 2017 Background Pyrazolo[1,5-a]pyrimidines are purine analogues. They have beneficial properties as antimetabolites in purine biochemical reactions. This division compounds have attracted wide pharmaceutical interest because of their antitrypanosomal activity.
Nadia A. Abdelriheem +2 more
doaj +1 more source
Composite Materials with Magnetically Aligned Carbon Nanoparticles Having Enhanced Electrical Properties and Methods of Preparation [PDF]
Magnetically aligned carbon nanoparticle composites have enhanced electrical properties. The composites comprise carbon nanoparticles, a host material, magnetically sensitive nanoparticles and a surfactant.
Hong, Haiping +2 more
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Synthesis, Characterisation and Biological Activities of Nitrogen-Sulphur Ligands and Their Transition Metal Complexes [PDF]
, 2008 Synthetic compounds, especially those containing heterocyclic ring systems composed of nitrogen and sulphur have been of great interest due to their versatility as medicinal drugs.
Begum, Thahira
core
Reactions with hydrazonoyl halides 65: Synthesis of some new 1,3,4-thiadiazoles and triazolino[4,3-a]pyrimidines containing pyrazole moiety [PDF]
, 2011 2,3-Dihydro-1,3,4-thiadiazoles, and triazolino[4,3-a]pyrimidines containing pyrazole moieties were prepared from the reaction of alkyl 2-[1-(4-cyano-1,5-diphenyl-1H-pyrazol-3-yl)ethylidene]hydrazinecarbodithioate and pyrimidine-2-thione derivatives with ...
Abdelhamid, Abdou Osman +2 more
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3-(2-Fluorophenyl)-6-(phenoxymethyl)-1,2,4-triazolo[3,4-b][1,3,4]thiadiazole
Acta Crystallographica Section E, 2008 The crystal structure of the title compound, C16H11FN4OS, was synthesized in the course of our studies on 1,2,4-triazolo[3,4-b][1,3,4]thiadiazoles as inhibitors of p38 mitogen-activated protein kinase (MAPK). The three-dimensional data obtained were used
Stefan Laufer +2 more
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Synthesis and Anticancer Activity of 1,3,4-Thiadiazoles with 3-Methoxyphenyl Substituent. [PDF]
Molecules, 2022 Janowska S +7 more
europepmc +1 more source