Results 1 to 10 of about 22,631 (229)

Phytogenic silver, gold, and bimetallic nanoparticles as novel antitubercular agents [PDF]

International Journal of Nanomedicine, 2016
Richa Singh,1 Laxman Nawale,2 Manisha Arkile,2 Sweety Wadhwani,1 Utkarsha Shedbalkar,1 Snehal Chopade,1 Dhiman Sarkar,2 Balu Ananda Chopade1,3 1Department of Microbiology, Savitribai Phule Pune University, 2Combichem-Bioresource Center, Organic ...
Singh R, Nawale L, Arkile M, Wadhwani S, Shedbalkar U, Chopade S, Sarkar D, Chopade BA   +7 more
doaj   +7 more sources

Exploration of Piperidinols as Potential Antitubercular Agents [PDF]

Molecules, 2014
Novel drugs to treat tuberculosis are required and the identification of potential targets is important. Piperidinols have been identified as potential antimycobacterial agents (MIC < 5 μg/mL), which also inhibit mycobacterial arylamine N ...
Areej Abuhammad, Elizabeth Fullam, Sanjib Bhakta, Angela J. Russell, Garrett M. Morris, Paul W. Finn, Edith Sim   +6 more
doaj   +8 more sources

Causality assessment, severity and preventability of adverse drug reactions due to first-line antitubercular agents [PDF]

Pharmaciana, 2022
TB (Tuberculosis) is a common infectious disease affecting humans since very long time. Multidrug therapy with its associated adverse drug reactions is one of the major concerns for the management of TB.
Gunjan Upadhyay, Apexa B Shukla, Darshan J Dave   +2 more
doaj   +3 more sources

Synthesis, Characterization, and Biological Evaluation of New Derivatives Targeting MbtI as Antitubercular Agents [PDF]

Pharmaceuticals, 2021
Tuberculosis (TB) causes millions of deaths every year, ranking as one of the most dangerous infectious diseases worldwide. Because several pathogenic strains of Mycobacterium tuberculosis (Mtb) have developed resistance against most of the established ...
Matteo Mori, Giovanni Stelitano, Laurent R. Chiarelli, Giulia Cazzaniga, Arianna Gelain, Daniela Barlocco, Elena Pini, Fiorella Meneghetti, Stefania Villa   +8 more
doaj   +2 more sources

Dataset of 2-(2-(4-aryloxybenzylidene) hydrazinyl) benzothiazole derivatives for GQSAR of antitubercular agents [PDF]

Data in Brief, 2017
Fragment based Quantitative structure activity relationship (QSAR) analysis on reported 25 2-(2-(4-aryloxybenzylidene) hydrazinyl) benzothiazole dataset as antitubercular agents were carried out.
Amit S. Tapkir, Sohan S. Chitlange, Ritesh P. Bhole   +2 more
doaj   +2 more sources

Structure-Activity Relationships of Pyrazolo[1,5-<i>a</i>]pyrimidin-7(4<i>H</i>)-ones as Antitubercular Agents. [PDF]

ACS Infect Dis, 2021
Oh S, Libardo MDJ, Azeeza S, Pauly GT, Roma JSO, Sajid A, Tateishi Y, Duncombe C, Goodwin M, Ioerger TR, Wyatt PG, Ray PC, Gray DW, Boshoff HIM, Barry CE.   +14 more
europepmc   +3 more sources

Identification of benzothiazones containing a hexahydropyrrolo[3,4-c]pyrrol moiety as antitubercular agents against MDR-MTB. [PDF]

RSC Adv, 2020
Ma X, Han B, Wang A, Yang L, Huang M, Chowdhury K, Gu J, Zhang K, Lv K.   +8 more
europepmc   +3 more sources

Synthesis, antitubercular activity and mechanism of resistance of highly effective thiacetazone analogues [PDF]

, 2013
Defining the pharmacological target(s) of currently used drugs and developing new analogues with greater potency are both important aspects of the search for agents that are effective against drug-sensitive and drug-resistant Mycobacterium tuberculosis ...
A Alahari, A Alahari, A Banerjee, A Bhatt, AE Grzegorzewicz, AK Ojha, AR Baulard, C Vilcheze, CK Stover, D Fegan, D Fegan, Derek Craig, E Dubnau, E Sacco, Emilie Vialla, F Wang, FM Shahab, G Lutfalla, Geoffrey D. Coxon, JA Caminero, Jean Louis Herrmann, JM Belardinelli, JR Wei, K Takayama, L Kremer, Laila Gannoun-Zaki, Laurent Kremer, LE Bermudez, LG Dover, LS Kremer, MA Espinal, MS Glickman, N Slama, P Nunn, PT Davidson, R Mondal, R Veyron-Churlet, R Veyron-Churlet, RM Corrales, Rosa Milagros Corrales, S Cantaloube, TD Bugg, V Rao, VK Sambandamurthy, Y Rombouts   +44 more
core   +21 more sources

Identification of 2-(N-aryl-1,2,3-triazol-4-yl) quinoline derivatives as antitubercular agents endowed with InhA inhibitory activity. [PDF]

Front Chem
Sabt A, Abdulla MH, Ebaid MS, Pawełczyk J, Abd El Salam HA, Son NT, Ha NX, Vaali Mohammed MA, Traiki T, Elsawi AE, Dziadek B, Dziadek J, Eldehna WM.   +12 more
europepmc   +2 more sources

Review of Recent Advances in Thiazolidin-4-One Derivatives as Promising Antitubercular Agents (2021-Present). [PDF]

Molecules
Drzał W, Trotsko N.
europepmc   +2 more sources