Results 31 to 40 of about 8,323 (256)
The Polymerization of Azetidines and Azetidine Derivatives [PDF]
Polymer Journal, 1980 The cationic ring-opening polymerization of azetidine, N-alkylazetidines and a number of azetidines carrying a second functional group is reviewed. Some of these monomers lead to “living” polymers. The rate constants for the polymerization of different azetidines are discussed and compared with the rate constants for the polymerization of other four ...
E J Goethals +4 more
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Frontiers in Chemistry, 2023 Azetidine is a prevalent structural motif found in various biologically active compounds. In this research paper, we report La(OTf)3-catalyzed intramolecular regioselective aminolysis of cis-3,4-epoxy amines to afford azetidines.
Yuse Kuriyama +2 more
doaj +1 more source
Synthesis of Azetidine-Based Beta-Amino Alcohols
Medical Sciences Forum, 2022 Beta-amino alcohols are versatile chemicals used as scaffolds in medicinal chemistry and they are key factors for the efficacy of numerous pharmaceutical products.
Linda Supe
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Azetidines. II. Some Functional Derivatives of Azetidines [PDF]
Bulletin of the Chemical Society of Japan, 1967 Abstract The sodium methoxide-catalyzed cyclization of methyl α-tosylamino-γ-chlorobutyrate gave methyl 1-tosylazetidine-2-carboxylate, which was then converted to the corresponding carboxylic acid and carbinol. 1-Acetyl-2,2,4,4-tetramethylazetidine-3-carboxylic acid was prepared by the photolysis of 1-acetyl-4-diazo-2,2,5,5 ...
Teng-yueh Chen +3 more
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Journal of Organic Chemistry, 2023 Four-membered heterocycles offer exciting potential as small polar motifs in medicinal chemistry but require further methods for incorporation. Photoredox catalysis is a powerful method for the mild generation of alkyl radicals for C–C bond formation ...
Maryne A. J. Dubois +10 more
semanticscholar +1 more source
Tetrahedron Green Chem, 2023 The synthesis of functionalized azetidines from azetines is poorly explored. Here, we report the safe and sustainable continuous flow hydrogenation of 2-azetines using ethyl acetate and CPME as environmentally responsible solvents.
Elena Graziano +6 more
doaj +1 more source
Defining stage-specific activity of potent new inhibitors of Cryptosporidium parvum growth in vitro [PDF]
, 2020 Currently, nitazoxanide is the only FDA-approved treatment for cryptosporidiosis; unfortunately, it is ineffective in immunocompromised patients, has varied efficacy in immunocompetent individuals, and is not approved in infants under 1 year of age ...
Funkhouser-Jones, Lisa J +2 more
core +2 more sources
Access to Azetidines via Gold Mediated Energy Transfer Photocatalysis.
Organic Letters, 2023 The area of energy transfer photocatalysis to generate four-membered rings is experiencing an unprecedented level of activity. Here, we report an operationally simple method toward azetidines from 2-isoxasoline-3-carboxylates and alkenes, using [Au(cbz ...
Sébastien G. Guillet +4 more
semanticscholar +1 more source
Synthesis of 2-Oxazolines from Ring Opening Isomerization of 3-Amido-2-Phenyl Azetidines
Molecules, 2021 Chiral 2-oxazolines are valuable building blocks and famous ligands for asymmetric catalysis. The most common synthesis involves the reaction of an amino alcohol with a carboxylic acid.
Xin Zhou, Baiyi Mao, Zhanbin Zhang
doaj +1 more source