Results 151 to 160 of about 3,510,874 (207)

Bridging BET bromodomain and immune checkpoint inhibitors through generative bioorganic frameworks for next-generation cancer immunotherapy. [PDF]

RSC Med Chem
Diab MK, Yassen ASA, Fahmy SA, Ashour HF, Nafie MS.   +4 more
europepmc   +1 more source

Reversible control of CAR T cells through PROTAC compound targeting bromodomain mutant. [PDF]

Mol Ther Oncol
Kim Y, Lee DY, Choi JU, Jeun M, Lee HK, Choi SU, Park CH.   +6 more
europepmc   +1 more source

Unusual backfolded binding poses of BAZ2A bromodomain binders. [PDF]

Acta Crystallogr D Struct Biol
Dalle Vedove A, Cazzanelli G, D'Agostino VG, Vargas Rosales PA, Caflisch A, Lolli G.   +5 more
europepmc   +1 more source

Development of a Lysine-Reactive Targeted Covalent Inhibitor for the P300/CBP-Associated Factor Bromodomain Through Structure-Based Design. [PDF]

ChemMedChem
Ede RR, Peterson KE, Begyinah RK, Tom IP, Ochoada JM, Sneddon MS, Tiu AKY, Fischer M, Shelat AA, Pomerantz WCK.   +9 more
europepmc   +1 more source

The bromodomain protein Bdf3 is sufficient to activate expression of a procyclin gene in bloodstream stage African trypanosomes. [PDF]

mSphere
Kim EJ, Goroza EL, Tan AY, Lin JJ, Saucedo KC, Tanizawa F, Smith JE, Schulz D.   +7 more
europepmc   +1 more source

Targeting the Androgen Receptor and Associated Cofactors in Prostate Cancer: Novel Approaches and Future Perspectives. [PDF]

Int J Mol Sci
Dziubańska-Kusibab PJ, Jourdan T, Haendler B.   +2 more
europepmc   +1 more source

Fragment-Based Discovery of BRD4-BD2 Selective Binders: Biophysical Validation and Structural Insights for Domain-Selective Inhibitor Design. [PDF]

ACS Omega
Baskaran SP, Subramani YV, Bairy SG, Prasad TK, Kumar V, Sridhar A, Padmanabhan B, Kamariah N.   +7 more
europepmc   +1 more source

NanoBRET Tracer Development for Class I Bromodomain Target Engagement in Live Cells. [PDF]

Bioconjug Chem
Sneddon MS, Tsou CJ, Fu X, Shelat AA, Pomerantz WCK.   +4 more
europepmc   +1 more source

Structural insights into histone mimicry by the small hepatitis delta antigen. [PDF]

J Biol Chem
Hu H, Lv M, Wang X, Shang X, Wu Q, Chen Y, Zhou Y, Huang Q, Jiang T, Qin S, Huang X, Zhang Z, Xu G, Liu Y.   +13 more
europepmc   +1 more source

Cis and trans regulatory mechanisms of extrachromosomal DNA segregation. [PDF]

Nat Cell Biol
Xie Y, Lim JYS, Liu W, Gilbreath C, Sun X, Qiao K, Kim YJ, Wu S.   +7 more
europepmc   +1 more source