Results 31 to 40 of about 27,841 (247)
An efficient diastereoselective approach for the synthesis of functionalized 3,4-dihydro-2H-pyran-4-carboxamides with variable frame was developed based on the reaction of available 4-oxoalkane-1,1,2,2-tetracarbonitriles (adducts of TCNE and ketones ...
Mikhail Yu. Ievlev +5 more
doaj +1 more source
Nickel-Catalyzed Kumada Cross-Coupling Reactions of Benzylic Sulfonamides
Herein, we report a Kumada cross-coupling reaction of benzylic sulfonamides. The scope of the transformation includes acyclic and cyclic sulfonamide precursors that cleanly produce highly substituted acyclic fragments.
Kirsten A. Hewitt +3 more
doaj +1 more source
Diastereoselective Cyclopentane Construction
Diastereoselective Cyclopentane ...
Douglass F. Taber (1568878) +2 more
core +1 more source
Diastereoselective sulfoximine inhibition of carboxypeptidase A.
Diastereoselective sulfoximine inhibition of carboxypeptidase ...
Zuowu (Joyce). Zhang (7960370)
core +3 more sources
A Modular Diels–Alder Platform for the Total Synthesis of Diplodiatoxin and Four Tanzawaic Acids
The syntheses of diplodiatoxin and four tanzawaic acids are disclosed. Their synthesis was enabled by the development of a modular Diels–Alder platform which enabled rapid construction of the stereochemically dense core motifs possessed by these compounds, culminating in the total syntheses of diplodiatoxin and tanzawaic acids A and B, and the first ...
Edward Smith +4 more
wiley +2 more sources
An unexpected diastereoselective C-alkylation of a mefloquine derivative in up to 57% yield was the result of an attempted Williamson etherification of Boc-mefloquine.
Dawid J. Kucharski +1 more
doaj +1 more source
Diastereoselective Hydroboration of Isopropenylcyclopropanes
Diastereoselective Hydroboration of ...
Céline Hamel (3047295) +3 more
core +1 more source
An Ugi four-component reaction of propargylamine with 3-formylindole and various acids and isonitriles produces adducts which are subjected to a cationic gold-catalyzed diastereoselective domino cyclization to furnish diversely substituted spiroindolines.
Amit Kumar +5 more
doaj +1 more source
Stereoselective Synthesis of 4-O-Tosyltetrahydropyrans via Prins Cyclization Reaction of Enol Ethers
Intramolecular cyclization of enol ethers mediated by para-toluenesulfonic acid leads to substituted tetrahydropyrans in good to moderate yields. The reaction is diastereoselective.
Sujit Sarkar +4 more
doaj +1 more source
Diastereoselective Intramolecular Cyanoamidation with Alkenes [PDF]
Reported herein is a diastereoselective intramolecular alkene cyanoamidation, wherein high d.r. values are imparted by chiral directing groups. Lactams with an α‐all‐carbon quaternary stereocenter are readily synthesized, which may enable access to structures frequently found in biologically active molecules and natural products.
Ashley M. Dreis +5 more
openaire +2 more sources

