Results 161 to 170 of about 24,568 (261)

A covalent chemical probe for Chikungunya nsP2 cysteine protease with antialphaviral activity and proteome-wide selectivity. [PDF]

Sci Rep
Ghoshal A, Tse EG, Hossain MA, Asressu KH, Merten EM, Sears JD, Howell S, Perveen S, Burdick J, Morales NL, Martinez SA, Law I, Davenport BJ, Morrison TE, Streblow ZJ, Streblow DN, Mordant AL, Webb TS, Cabrera A, Herring LE, Arrowsmith CH, Pearce KH, Moorman NJ, Heise MT, Couñago RM, Brown PJ, Willson TM.   +26 more
europepmc   +1 more source

In Vitro Evaluation of ¹¹C‐Labeled (S)‐Nicotine, (S)‐3‐Methyl‐5‐(1‐Methyl‐2‐Pyrrolidinyl)isoxazole, and (R,S)‐1‐Methyl‐2‐(3‐Pyridyl)azetidine as Nicotinic Receptor Ligands for Positron Emission Tomography Studies

, 1998
Wiebke Sihver, Karl‐Johan Fasth, Mattias Ögren, Håkan Bivehed, Mats Bergström, Agneta Nordberg, Yasuyoshi Watanabe, Bengt Långström   +7 more
openalex   +1 more source

Oxazole and isoxazole-containing pharmaceuticals: targets, pharmacological activities, and their SAR studies. [PDF]

RSC Med Chem
Li S, Mei Y, Jiang L, Yang X, Zeng W, Du Y.   +5 more
europepmc   +1 more source

Synthesis of C-xylopyranosyl- and xylopyranosylidene-spiro-heterocycles as potential inhibitors of glycogen phosphorylase [PDF]

, 2019
Bokor, Éva, Czibere, Beáta, Czifrák, Katalin, Docsa, Tibor, Gergely, Pál, Koppány, Csenge, Kulcsár, László, Kun, Sándor, Somsák, László, Szilágyi, Enikő, Tóth, Marietta   +10 more
core   +1 more source

Novel Isoxazole-Based Antifungal Drug Candidates. [PDF]

Int J Mol Sci
Bąchor U, Brożyna M, Junka A, Chmielarz MR, Gorczyca D, Mączyński M.   +5 more
europepmc   +1 more source

Protein Kinase Cγ Associates Directly with the GluR4 α-Amino-3-hydroxy-5-methyl-4-isoxazole Propionate Receptor Subunit [PDF]

, 2003
Susana S. Correia, Carlos B. Duarte, Carlos Faro, Euclides Pires, Ana Luı́sa Carvalho   +4 more
openalex   +1 more source

Synthesis, characterization, molecular docking and pharmacological evaluation of isoxazole derivatives as potent anti-inflammatory agents. [PDF]

Heliyon
Sonu, Yt K, Gautam GK, Mishra AK, Parveen BR, Kumar A, Singh M, Singh H.   +7 more
europepmc   +1 more source

Facile Construction and Divergent Transformation of Polycyclic Isoxazoles: Direct Access to Polyketide Architectures. [PDF]

, 2003
Jeffrey W. Bode, Yoshifumi Hachisu, Tomoo Matsuura, Keisuke Suzuki   +3 more
openalex   +1 more source

Light-Induced, Lysine-Targeting Irreversible Covalent Inhibition of the Human Oxygen Sensing Hydroxylase Factor Inhibiting HIF (FIH). [PDF]

J Am Chem Soc
Wu Y, Li Z, Kaur S, Zhang Z, Yue J, Tumber A, Zhang H, Song Z, Yang P, Dong Y, Yang F, Li X, Schofield CJ, Zhang X.   +13 more
europepmc   +1 more source

Crystal structure of (3aS,4R,5S,6R,6aS)-4,5,6-tris-benzoyloxy-l-methylhexahydro- cyclopent(c)isoxazole, C28H25NO7

, 1997
S. Henkel, M. Kleban, V. Jäger
openalex   +1 more source