Half-Sandwich Nickelacarboranes Derived from [7-(MeO(CH2)2S)-7,8-C2B9H11]−
Inorganics, 2023 New carboranyl thioethers 1-MeO(CH2)nS-1,2-C2B10H11 (n = 2, 3) were prepared by the alkylation of the trimethylammonium salt of 1-mercapto-ortho-carborane with 1-bromo- 2-methoxyethane and 1-bromo-3-methoxypropane, respectively.
Dmitriy K. Semyonov +3 more
doaj +1 more source
Boron-containing delocalised lipophilic cations for the selective targeting of cancer cells [PDF]
, 2016 Correction for “Boron-containing delocalised lipophilic cations for the selective targeting of cancer cells” by Gianpiero Calabrese et al., Med. Chem. Commun., 2017, 8, 67–72.
Calabrese, Gianpiero +6 more
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“Free of Base” Sulfa-Michael Addition for Novel o-Carboranyl-DL-Cysteine Synthesis
Crystals, 2020 The sulfa-Michael addition reaction was applied for the two-step synthesis of o-carboranyl cysteine 1-HOOCCH(NH2)CH2S-1,2-C2B10H11 from the trimethylammonium salt of 1-mercapto-o-carborane and methyl 2-acetamidoacrylate.
Julia Laskova +5 more
doaj +1 more source
Chelating N-heterocyclic carbene-carboranes offer flexible ligand coordination to IrIII, RhIII and RuII: effect of ligand cyclometallation in catalytic transfer hydrogenation [PDF]
, 2016 Imidazolium salts linked by an ethyl tether to closo-dicarbadodecaboranes were reacted with [IrCp*Cl2]2, [RhCp*Cl2]2 or [Ru(p-cymene)Cl2]2 in the presence of Ag2O to prepare complexes of the type [MCp*(NHC)Cl2] (M = Ir, Rh; NHC = N-heterocyclic carbene ...
Aher +54 more
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Novel Isoniazid-Carborane Hybrids Active In Vitro against Mycobacterium tuberculosis
Pharmaceuticals, 2020 Tuberculosis (TB) is a severe infectious disease with high mortality and morbidity. The emergence of drug-resistant TB has increased the challenge to eliminate this disease.
Daria Różycka +9 more
doaj +1 more source
Pharmacokinetics of core-polymerized boron-conjugated micelles designed for boron neutron capture therapy for cancer [PDF]
, 2012 journal ...
Horiguchi Yukichi +8 more
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Applications of AFM in pharmaceutical sciences [PDF]
, 2016 Atomic force microscopy (AFM) is a high-resolution imaging technique that uses a small probe (tip and cantilever) to provide topographical information on surfaces in air or in liquid media.
Lamprou, Dimitrios, Smith, James R.
core +2 more sources
Thermally activated delayed fluorescence in neutral and cationic copper(I) complexes with the 2-(4-Thiazolyl)benzimidazole ligand [PDF]
, 2023 Cationic [Cu(P^P)(Htbz)]PF6 [P^P = xantphos, dpephos; Htbz = 2-(4-thiazolyl)benzimidazole] and the corresponding neutral complexes [Cu(P^P)(tbz)], obtained through deprotonation of the diimine ligand, have been synthesized with the aim of analyzing the ...
Alconchel, A., Crespo, O., Gimeno, M. C.
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Advances in Diclofenac Derivatives: Exploring Carborane-Substituted N-Methyl and Nitrile Analogs for Anticancer Therapy. [PDF]
ChemMedChemBy N‐methylation, the intramolecular lactam formation in carborane‐substituted diclofenac analogs is prevented, yielding a series of open‐chain derivatives alongside with their phenyl analogs exhibiting anticancer activity and thus offering a promising avenue for future drug development. This study explores the anticancer potential of N‐methylated open‐
Selg C +12 more
europepmc +2 more sources
Synthesis and Structural Characterization of p -Carboranylamidine Derivatives † [PDF]
, 2023 In this contribution, the first amidinate and amidine derivatives of p -carborane are described. Double lithiation of p -carborane ( 1 ) with n -butyllithium followed by treatment with 1,3-diorganocarbodiimides, R–N=C=N–R (R = i Pr, Cy (= cyclohexyl ...
Busse, Sabine +7 more
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