Results 21 to 30 of about 7,689 (220)
Enantiomeric Separation of New Chiral Azole Compounds
Twelve new azole compounds were synthesized through an ene reaction involving methylidene heterocycles and phenylmaleimide, producing four oxazoles, five thiazoles, and one pyridine derivative, and ethyl glyoxylate for an oxazole and a thiazole compound.
Marziyeh E. Kenari +9 more
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Transition metal-mediated synthesis of oxazoles [PDF]
Among the synthetic methods for the formation of the oxazole ring, transition metal-mediated protocols are the most attractive in terms of selectivity, efficiency and mildness of reaction conditions.
Bresciani, Stefano +1 more
core +1 more source
A novel method for the synthesis of trisubstituted oxazoles via a one-pot oxazole synthesis/Suzuki–Miyaura coupling sequence has been developed.
Kohei Yamada +2 more
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Six 1,3-oxazoles were synthetized in moderate to good yields by Van Leusen reaction in a pressure reactor. The methodology allowed to decrease the reaction times reported in the literature from hours to 20 min.
Verónica G. García-Ramírez +4 more
doaj +1 more source
Naturally Occurring Oxazole-Containing Peptides [PDF]
Oxazole-containing peptides are mostly of marine origin and they form an intriguing family with a broad range of biological activities. Here we classify these peptides on the basis of their chemical structure and discuss a number of representatives of each class that reflect the extraordinary potential of this family as a source of new drugs.
Jessica T. Mhlongo +3 more
openaire +3 more sources
The rapid synthesis of oxazolines and their heterogeneous oxidation to oxazoles under flow conditions. [PDF]
A rapid flow synthesis of oxazolines and their oxidation to the corresponding oxazoles is reported. The oxazolines are prepared at room temperature in a stereospecific manner, with inversion of stereochemistry, from β-hydroxy amides using Deoxo-Fluor ...
Battilocchio, Claudio +6 more
core +2 more sources
Continuous multistep synthesis of 2-(azidomethyl)oxazoles
An efficient three-step protocol was developed to produce 2-(azidomethyl)oxazoles from vinyl azides in a continuous-flow process. The general synthetic strategy involves a thermolysis of vinyl azides to generate azirines, which react with bromoacetyl ...
Thaís A. Rossa +4 more
doaj +1 more source
Diazocarbonyl and Related Compounds in the Synthesis of Azoles
Diazocarbonyl compounds have found numerous applications in many areas of chemistry. Among the most developed fields of diazo chemistry is the preparation of azoles from diazo compounds.
Anton Budeev +3 more
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Sir John Cornforth AC CBE FRS: his synthetic work [PDF]
Sir John Cornforth’s work on the synthesis of cholesterol and penicillamine, on the chemistry of oxazoles, the stereochemistry of the synthesis of alkenes, the synthesis of abscisic acid and of dibenzophospholes as mimics of enzyme action, is ...
Abraham E.P. +15 more
core +1 more source
Gold Catalyzed Multicomponent Reactions beyond A3 Coupling
The preparation of complex architectures has inspired the search for new methods and new processes in organic synthesis. Multicomponent reactions have become an interesting approach to achieve such molecular diversity and complexity.
Renso Visbal +3 more
doaj +1 more source

