Results 131 to 140 of about 26,717 (273)

Editorial: Expansion of the Genetic Code: Unnatural Amino Acids and their Applications

Frontiers in Chemistry, 2022
Subhendu Sekhar Bag, Ishu Saraogi, Jiantao Guo   +2 more
doaj   +1 more source

A peptidomimetic with a chiral switch is an inhibitor of epidermal growth factor receptor heterodimerization

OncoTarget, 2017
Among different types of EGFR dimers, EGFR-HER2 and HER2-HER3 are well known in different types of cancers. Targeting dimerization of EGFR will have a significant impact on cancer therapies.
S. Kanthala, Yong-Yu Liu, Sitanshu S. Singh, Rushikesh Vilas Sable, Sandeep Pallerla, S. Jois   +5 more
semanticscholar   +1 more source

Solid-Phase Synthesis and Circular Dichroism Study of β-ABpeptoids

Molecules, 2019
The development of peptidomimetic foldamers that can form well-defined folded structures is highly desirable yet challenging. We previously reported on α-ABpeptoids, oligomers of N-alkylated β2-homoalanines and found that due to the presence ...
Ganesh A. Sable, Kang Ju Lee, Hyun-Suk Lim   +2 more
doaj   +1 more source

Interferon gamma peptidomimetic targeted to interstitial myofibroblasts attenuates renal fibrosis after unilateral ureteral obstruction in mice

OncoTarget, 2016
Renal fibrosis cannot be adequately treated since anti-fibrotic treatment is lacking. Interferon-γ is a pro-inflammatory cytokine with anti-fibrotic properties.
Fariba Poosti, Ruchi Bansal, S. Yazdani, J. Prakash, L. Beljaars, J. van den Born, M. D. de Borst, H. van Goor, J. Hillebrands, K. Poelstra   +9 more
semanticscholar   +1 more source

The Risk of Immune‐Mediated Skin Disease Under Dipeptidyl‐Peptidase IV Inhibitor: A Global Population‐Based Study

International Journal of Dermatology, Volume 65, Issue 2, Page 356-358, February 2026.
Noor Mruwat, Noga Givon‐Lavi, Ralf J. Ludwig, Khalaf Kridin   +3 more
wiley   +1 more source

Stem cells in chronic myeloid leukaemia [PDF]

, 2007
Holyoake, T., Pellicano, F.
core   +1 more source

Computer-aided design of amino acid-based therapeutics: a review

Drug Design, Development and Therapy, 2018
Tayebeh Farhadi,1 Seyed MohammadReza Hashemian1,2 1Chronic Respiratory Diseases Research Center (CRDRC), National Research Institute of Tuberculosis and Lung Diseases (NRITLD), Shahid Beheshti University of Medical Sciences, Tehran, Iran; 2Clinical ...
Farhadi T, Hashemian SM
doaj  

Vipegitide: a folded peptidomimetic partial antagonist of α2β1 integrin with antiplatelet aggregation activity

Drug Design, Development and Therapy, 2015
Tatjana Momic,1 Jehoshua Katzhendler,1 Ela Shai,2 Efrat Noy,3 Hanoch Senderowitz,3 Johannes A Eble,4 Cezary Marcinkiewicz,5 David Varon,2 Philip Lazarovici11School of Pharmacy Institute for Drug Research, Faculty of Medicine, The Hebrew University of ...
Momic T, Katzhendler J, Shai E, Noy E, Senderowitz H, Eble JA, Marcinkiewicz C, Varon D, Lazarovici P   +8 more
doaj  

Editorial: Contemporary Perspective on 5-HT2C Receptor Function and Its Pharmacological Targeting

Frontiers in Pharmacology, 2020
Philippe De Deurwaerdère, Abdeslam Chagraoui, Abdeslam Chagraoui, Kathryn A. Cunningham   +3 more
doaj   +1 more source

Evidence of an activity-enhancing conformational shift in Arabidopsis thaliana plant cysteine oxidase 4 induced by binding of substrate or substrate-mimics. [PDF]

J Biol Chem
Latter R, Hintzen JCJ, Shah LMN, Gunawardana DM, Sher RM, White MD, Mecinović J, Benesch JLP, Flashman E.   +8 more
europepmc   +1 more source