Results 141 to 150 of about 26,717 (273)

Deconvolution of the On-Target Activity of Plasmepsin V Peptidomimetics in <i>Plasmodium falciparum</i> Parasites. [PDF]

ACS Infect Dis
Su W, Nguyen W, Siddiqui G, Dziekan JM, Marapana D, Penington JS, Mehra S, Razook Z, McCann K, Ngo A, Jarman KE, Barry AE, Papenfuss AT, Gilson PR, Creek DJ, Cowman AF, Sleebs BE, Dans MG.   +17 more
europepmc   +1 more source

Potent peptidomimetics [PDF]

Nature Biotechnology, 1999
openaire   +1 more source

Retraction Note: Thiazole-valine peptidomimetic (TTT-28) antagonizes multidrug resistance in vitro and in vivo by selectively inhibiting the efflux activity of ABCB1. [PDF]

Sci Rep
Wang YJ, Patel BA, Anreddy N, Zhang YK, Zhang GN, Alqahtani S, Singh S, Shukla S, Kaddoumi A, Ambudkar SV, Talele TT, Chen ZS.   +11 more
europepmc   +1 more source

Role of Structural Modifications in Peptidomimetic Compounds as Potential Antimicrobial Agents against <i>Staphylococcus aureus</i> and <i>Streptococcus pyogenes</i>: Balancing Bioavailability, Safety, and Antimicrobial Activity. [PDF]

ACS Omega
Dzierżyńska M, Sawicka J, Łada K, Gajewicz-Skretna A, Deptuła M, Chernobrovkin A, Pogorzelska A, Grubb A, Zubarev RA, Pikuła M, Kasprzykowski F, Rodziewicz-Motowidło S.   +11 more
europepmc   +1 more source

Application of Doebner-type aminoazole based heterocycle acides in Ugi 4CR [PDF]

, 2018
Chebanov, V. A., Kolomiets, O. V., Murlykina, M. M., Sakhno, Y. I., Tsygankov, A. V.   +4 more
core  

Novel macrocyclic peptidomimetics targeting the insulin-regulated aminopeptidase (IRAP): design, synthesis and evaluation. [PDF]

RSC Med Chem
Olaniran Håkansson E, Balestri LJI, Puthiyaparambath S, Moes S, Henschel H, Sköld C, Hallberg M, Larhed M, Skillinghaug B, Odell LR.   +9 more
europepmc   +1 more source

Machine Learning-Guided Repositioning of a SARS-CoV-2-Targeting Molecular Series as Cruzain Inhibitors. [PDF]

ChemMedChem
Lameiro RF, Barbosa LF, Cardoso ER, Ho BS, Martins FCP, de Melo BC, Rosini F, Shamim A, Souza PM, de Souza WF, Montanari CA.   +10 more
europepmc   +1 more source

A Polyproline Type II Peptidomimetic Disrupts a Grb2 SH3C Domain Protein-Protein Interaction Implicated in Breast Cancer. [PDF]

Chembiochem
Luccarelli J, Simister PC, Hamilton AD, Feller SM, Thompson S.   +4 more
europepmc   +1 more source

High-Affinity Peptidomimetic Inhibitors of the DCN1-UBC12 Protein-Protein Interaction.

Journal of Medicinal Chemistry, 2018
Haibin Zhou, Weihua Zhou, Bing Zhou, Liu Liu, Ting‐Rong Chern, Krishnapriya Chinnaswamy, Jianfeng Lu, D. Bernard, Chao-Yie Yang, Shasha Li, Mi Wang, J. Stuckey, Yi Sun, Shaomeng Wang   +13 more
semanticscholar   +1 more source

Bacterial resistance and susceptibility to antimicrobial peptides and peptidomimetics [PDF]

, 2017
Citterio, Linda
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