Results 1 to 10 of about 59,616 (308)
Thiazole-driven heterocyclic hybrids as EGFR inhibitors: progress in synthesis and anticancer applications. [PDF]
RSC AdvDsouza A, Subrahmanyam VM, Shetty NS.
europepmc +2 more sources
Synthesis and Biological Evaluation of 2-Aminothiazole Analogues of Nα-Protected Amino Acids [PDF]
Iranian Journal of Chemistry & Chemical Engineering, 2023 Synthesis of 2-amino-thiazoles from Nα-protected bromomethyl ketones obtained from Nα-protected diazomethyl ketones has been reported in this study.N-protected amino acids were converted to diazomethylketones using (Benzotriazol-1-yloxy) tris ...
Lalithamba Haraluru Shankaraiah +3 more
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Molecules, 2021 Thiazole, a five-membered heteroaromatic ring, is an important scaffold of a large number of synthetic compounds. Its diverse pharmacological activity is reflected in many clinically approved thiazole-containing molecules, with an extensive range of ...
Anca-Maria Borcea +3 more
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Synthesis of Thiazole-2(3H)-thiones as Antimicrobial Agents Promoted by H3PW12O40-amino-functionalized CdFe12O19@SiO2 Nanocomposite [PDF]
Nanochemistry Research, 2022 H3PW12O40-amino-functionalized CdFe12O19@SiO2 nanocomposite has been utilized as an effective nanocatalyst for the preparation of thiazole-2(3H)-thiones by three-component reactions of CS2, 2-bromoacetophenone or 2-bromo-1-(4-methoxyphenyl) ethenone, and
Hossein Shahbazi-Alavi +1 more
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Synthesis and Structural Confirmation of the Thiazole Alkaloids Derived from Peganum harmala L.
Applied Sciences, 2021 Peganumal A and B are thiazole alkaloids isolated from the seeds of Peganum harmala L. Thiazole moieties are rarely found in natural products, but diverse compounds possessing thiazole moieties have attracted attention owing to their broad range of ...
Myeonghyeon Sim +2 more
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5-Chloro-6-oxo-6H-xantheno[4,3-d]thiazole-2-carbonitrile
Molbank, 2022 Xanthones and benzothiazoles are important classes of heterocyclic compounds with versatile biological activities. Herein, we describe a straightforward and scalable synthesis of 5-chloro-6-oxo-6H-xantheno[4,3-d]thiazole-2-carbonitrile, a thiazole-fused ...
Konstantinos Paraskevas +3 more
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In Vitro Inhibition Effects of 2-Amino Thiazole Derivatives on Lactoperoxidase Enzyme Activity
Cumhuriyet Science Journal, 2022 Lactoperoxidase (LPO E.C. 1.11.1.7) is a member of the peroxidase family and is an important glycoprotein containing heme group in its structure and showing the antimicrobial effect on disease causing microorganisms in the digestive system of newborn ...
Işıl Nihan Korkmaz
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Molecules, 2022 For many decades, the thiazole moiety has been an important heterocycle in the world of chemistry. The thiazole ring consists of sulfur and nitrogen in such a fashion that the pi (π) electrons are free to move from one bond to other bonds rendering ...
Mohammed F. Arshad +15 more
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Thiazole antibiotics target FoxM1 and induce apoptosis in human cancer cells. [PDF]
PLoS ONE, 2009 Forkhead box M1 (FoxM1) oncogenic transcription factor represents an attractive therapeutic target in the fight against cancer, because it is overexpressed in a majority of human tumors.
Uppoor G Bhat +2 more
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Phytopathology Research, 2019 Rice bacterial blight (BB), caused by Xanthomonas oryzae pv. oryzae (Xoo), is one of the most destructive diseases in rice-growing regions worldwide. Zinc thiazole is a novel bactericide and has been applied for BB control for 10 years.
Xian Chen +5 more
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