Comptes Rendus. Chimie, 2022 In our previous research, some screened 1,3-thiazole fragments were found to be potent by inhibiting LPS-induced TNF$\alpha $ and IL-8 release with IC50 values in the $\mu $M range without cytotoxic activity.
Modrić, Marina +7 more
doaj +1 more source
closo‐Carboranylanaloga von β‐Arylethylaminen: Direkte Synthese aus Alkenen mittels EnT‐Katalyse
Angewandte Chemie, EarlyView.Eine Strategie zur direkten Synthese von closo‐Carboranylanaloga medizinisch relevanter β‐Arylethylamine aus Alkenen wird vorgestellt. Die Reaktion basiert auf der erstmaligen Erzeugung von closo‐Carboranylradikalen mittels Energietransfer‐(EnT)‐Katalyse und ihren besonderen mechanistischen Merkmalen.
Fritz Paulus +8 more
wiley +1 more source
Molecules, 2020 Thiazole derivatives attract the attention of scientists both in the field of organic synthesis and bioactivity research due to their high biological activity.
Birutė Sapijanskaitė-Banevič +4 more
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InCl3-assisted synthesis and cytotoxic studies of some novel heteroaryl thiazoles [PDF]
, 2013 Heteroaryl thiazoles were synthesized by the Hantzsch reaction of various α-bromoketones with aryl thioureas using InCl3 as a catalyst in a shorter reaction time. The synthesized compds.
Boggavarapu Chand, S.G. +5 more
core
Neuere heterocyclische Zwischenprodukte für die Azokupplung durch Cyclisierung von Nitrilen
CHIMIA, 1980 Two types of syntheses of heteroaromatic amines by cyclization of nitriles are described. It is dealt with the cyclization of nitriles by elemental sulphur yielding thiophenes and thiazoles and with some reactions of the resulting 2-amino-thiophene-3 ...
Karl Gewald
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Reactivity of [Re\u3csub\u3e2\u3c/sub\u3e(CO)\u3csub\u3e8\u3c/sub\u3e(MeCN)\u3csub\u3e2\u3c/sub\u3e] with Thiazoles: Hydrido Bridged Dirhenium Compounds Bearing Thiazoles in Different Coordination Modes [PDF]
, 2007 Reactions of the labile compound [Re2(CO)8(MeCN)2] with thiazole and 4-methylthiazole in refluxing benzene afforded the new compounds [Re2(CO)7{μ-2,3-η2-C3H(R)NS}{η1-NC3H2(4-R)S}(μ-H)] (1, R = H; 2, R = CH3), [Re2(CO)6{μ-2,3-η2-C3H(R)NS}{η1-NC3H2(4-R)S}2(
Ahmed, Faruque +8 more
core +1 more source
Antimicrobial activity, synergism and inhibition of germ tube formation by Crocus sativus-derived compounds against Candida spp [PDF]
, 2016 The limited arsenal of synthetic antifungal agents and the emergence of resistant Candida strains have prompted the researchers towards the investigation of naturally occurring compounds or their semisynthetic derivatives in order to propose new ...
ANGIOLELLA, Letizia +4 more
core +2 more sources
ChemInform Abstract: Bioactive Thiazole and Benzothiazole Derivatives
ChemInform, 2015 AbstractReview: [90 refs.
Rouf, Abdul, Tanyeli, Cihangir
openaire +5 more sources
Nova Biotechnologica et Chimica, 2018 Substituted thiophene-2-carbaldehydes 1a-dwere utilized in the synthesis of symmetrically substituted thiazolo[5,4-d]thiazoles 3a-d. Bis(5,4-d)thiazoles with thiophene core at the termini are the most employed in the chemistry of materials but exhibit ...
Tokárová Zita, Biathová Anna
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closo‐Carboranyl Analogs of β‐Arylethylamines: Direct Synthesis from Alkenes via EnT‐Catalysis
Angewandte Chemie International Edition, EarlyView.A strategy to directly synthesize closo‐carboranyl analogs of medicinal chemically important β‐arylethylamines from alkenes is reported. This reaction is enabled by the first formation of closo‐carboranyl radicals by energy transfer (EnT) catalysis and its unique mechanistic features.
Fritz Paulus +8 more
wiley +1 more source