Green Chemistry Letters and Reviews, 2016 A simple and eco-friendly method for the synthesis of novel imidazo[2,1-b][1,3]thiazin derivatives has been developed via the one-pot, three-component and solvent-free reaction of thiohydantoins, aromatic aldehyde and 5,5-dimethylcyclohexane-1,3-dione in
Mohammad Mehdi Ghanbari
doaj +1 more source
Inhibition of iodine organification and regulation of follicular size in rat thyroid tissue in vitro [PDF]
, 2018 The factors mediating the accumulation of thyroglobulin are of great importance to the understanding of the pathogenesis of human and experimentally induced colloid goiters.
Büchler, Markus +8 more
core
Synthesis and crystal structure of (S)-5-isopropyl-5-methyl-2-thiohydantoin [PDF]
, 2013 (S)-5-Isopropyl-5-methyl-2-thiohydantoin was synthesized by one-pot reaction of α-methyl-L-valine and thiourea in the absence of solvent. The crystal structure of this compound has been determined from single crystal X-ray diffraction data.
Fujinami, Shuhei +8 more
core +1 more source
A természet szénhidrátkémikusai: enzimatikus glikozilezések = Nature's carbohydrate chemists: enzymatic glycosylation [PDF]
, 2009 Oligoszacharidok enzimekkel történő előállítása egy igen vonzó alternatív módszer a konvencionális kémiai megközelítés mellett, mert védő csoportok használata nélkül a célvegyület képződését eredményezi.
Bajza, István +3 more
core
مجلة بغداد للعلومRecently, some prostate cancer patients have acquired resistance to the second -generation drugs (anzalutamide and apalutamide) prescribed for the treatment of this disease due to the emergence of the F876L mutation, which represents a challenge
Qusay Hussein Hays +1 more
doaj +1 more source
New 5-ylidene rhodanine derivatives based on the dispacamide A model.
, 2014 International audienceA practical approach for the preparation of ([Formula: see text]) 5-ylidene rhodanine derivatives bearing the (4,5-dihalogeno-pyrrol-2-yl)carbamoyl fragment of dispacamide A is reported.
Bazureau, Jean-Pierre +6 more
core +4 more sources
One-Pot High-throughput Synthesis of N3-Substituted 5-Arylidene-2-Thiohydantoin Amides and Acids. [PDF]
Tetrahedron Lett, 2022 Whitely C, Li Y.
europepmc +1 more source
IN VITRO STUDIES ON THE ANTIDIABETIC ACTIVITY OF 2-THIOHYDANTOIN USING α-amylase AND α-GLUCOSIDASE [PDF]
, 2019 Objective: The aim of the present study was to investigate the inhibitory effect of 2-thiohydantoin on the enzymes α-amylase and α-glucosidase in vitro as an antidiabetic therapeutic approach to reduce gastrointestinal glucose production.
DEVIKA PT, UMA S
core +1 more source
Novel imidazolium-thiohydantoin hybrids and their Mn(iii) complexes for antimicrobial and anti-liver cancer applications. [PDF]
RSC Adv, 2022 Ismail LA +7 more
europepmc +1 more source
Reactions with 5-Arylazo- and 5-Arylidene-4-thiohydantoin Derivatives [PDF]
, 1979 5-Arylazo-3-phenyl-4-thiohydantoins (IIa-g) have been prepared and then treated with primary aromatic amines to afford the corresponding 5-arylazo-4-arylimino-3-phenyl hydantoins (VIIa-c).
A. F. A. Shalaby +2 more
core +1 more source