Results 101 to 110 of about 1,246 (203)

An efficient synthesis of imidazo[2,1-b][1,3]thiazins via a one-pot, three-component and solvent-free reaction

Green Chemistry Letters and Reviews, 2016
A simple and eco-friendly method for the synthesis of novel imidazo[2,1-b][1,3]thiazin derivatives has been developed via the one-pot, three-component and solvent-free reaction of thiohydantoins, aromatic aldehyde and 5,5-dimethylcyclohexane-1,3-dione in
Mohammad Mehdi Ghanbari
doaj   +1 more source

Biological potential of new molecular hybrids of thiohydantoin and zingerone derivatives

, 2022
Molecular hybridization is one of the most valuable structure modification tools currently used in drug construction. The concept of hybridization is usually achieved via chemical connection of two or more biologically active pharmacophoric moieties to ...
Virijevic, Katarina, Šmit, Biljana, Stanić, Petar, Muškinja, Jovana   +3 more
core  

1H NMR study of interactions between cisplatin and N-allyl-2-thiohydantoin type ligand

, 2018
cis-Diamminedichloridoplatinum(II) or cisplatin, cis-[PtCl2(NH3)2], is the one of most widely used anticancer drug. Its effectiveness against various cancer types is well established.
Živković, Marija, Šmit, Biljana, Soldatović, Tanja, Stanić, Petar, Ašanin, Darko   +4 more
core  

Study of the Anticancer and Antimicrobial Biological Activity of a New Series of Thiohydantoin Derivatives

مجلة بغداد للعلوم
        Recently, some prostate cancer patients have acquired resistance to the second -generation drugs (anzalutamide and apalutamide) prescribed for the treatment of this disease due to the emergence of the F876L mutation, which represents a challenge
Qusay Hussein Hays, Dakhil Zughayir Mutlaq   +1 more
doaj   +1 more source

Modification of intracellular free calcium in cultured F2408 embryo fibroblasts by 3-sub substituted-2-thiohydantoin derivatives

, 2004
WOS: 000221424800004PubMed ID: 151099823-substituted-2-thiohydantoin derivatives were synthesized and their Structures elucidated by IR, H-1-NMR spectroscopy and elemental analysis.
Benkli, Kadriye, Akalın, G, Kaplancıklı, Zafer Asım, Seller, Zerrin   +3 more
core   +1 more source

One-Pot High-throughput Synthesis of N3-Substituted 5-Arylidene-2-Thiohydantoin Amides and Acids. [PDF]

Tetrahedron Lett, 2022
Whitely C, Li Y.
europepmc   +1 more source

An electrospray ionization study of some novel alkylamine thiohydantoin amino acid derivatives

, 1995
An electrospray ionization-mass spectrometric (ES-MS) study of some novel alkylamine thiohydantoin amino acid derivatives is presented. The alkylamine derivatives are being developed as part of an on-going effort to couple an Edmanlike protein sequencer ...
Lee, Terry D., Bailey, Jerome M., Basic, Cecilia   +2 more
core   +1 more source

Novel imidazolium-thiohydantoin hybrids and their Mn(iii) complexes for antimicrobial and anti-liver cancer applications. [PDF]

RSC Adv, 2022
Ismail LA, Zakaria R, Hassan EM, Alfaifi MY, Shati AA, Elbehairi SEI, El-Bindary AA, Elshaarawy RFM.   +7 more
europepmc   +1 more source

Antidiabetic Potential of Novel 1,3,5-Trisubstituted-2-Thioxoimidazloidin-4-One Analogues: Insights into α-Glucosidase, α-Amylase, and Antioxidant Activities. [PDF]

Pharmaceuticals (Basel), 2022
Khirallah SM, Ramadan HMM, Aladl HAA, Ayaz NO, Kurdi LAF, Jaremko M, Alshawwa SZ, Saied EM.   +7 more
europepmc   +1 more source

Spiroleiferthione A and Oleiferthione A: Two Unusual Isothiocyanate-Derived Thioketone Alkaloids from Moringa oleifera Lam. Seeds. [PDF]

Pharmaceuticals (Basel), 2023
Jiang Y, Liu R, Huang L, Huang Q, Liu M, Liu S, Li J.   +6 more
europepmc   +1 more source