Results 81 to 90 of about 873 (170)

Solvent-modulated second harmonic generation in <i>N</i>-alkylated thiohydantoin derivatives: synthesis, characterization, and first-principle insights. [PDF]

RSC Adv
Ali MA, Qureshi MZ, Saleem RSZ, Mojzych M, Sharif A, Arshad M.   +5 more
europepmc   +1 more source

[3 + 2] Cycloaddition of thioformylium methylide with various arylidene-azolones in the synthesis of 7-thia-3-azaspiro[4.4]nonan-4-ones. [PDF]

Beilstein J Org Chem
Rudik DI, Tiushina IV, Sokolov AI, Smirnov AY, Romanenko AR, Korlyukov AA, Mikhaylov AA, Baranov MS.   +7 more
europepmc   +1 more source

In vitro assays identified thiohydantoins with anti-trypanosomatid activity and molecular modelling studies indicated possible selective CYP51 inhibition. [PDF]

Sci Rep
Camargo PG, Suzukawa HT, Pereira PML, Silva ML, Macedo F, Albuquerque MG, Rodrigues CR, Yamada-Ogatta SF, da Silva Lima CH, Bispo MLF.   +9 more
europepmc   +1 more source

Synthesis of Enantioenriched <i>gem</i>-Disubstituted 4-Imidazolidinones by Palladium-Catalyzed Decarboxylative Asymmetric Allylic Alkylation. [PDF]

Org Lett, 2021
Sercel ZP, Sun AW, Stoltz BM.
europepmc   +1 more source

Spirocyclic Thiohydantoin Antagonists of F877L and Wild-Type Androgen Receptor for Castration-Resistant Prostate Cancer. [PDF]

ACS Med Chem Lett, 2021
Zhang Z, Connolly PJ, Trabalón Escolar L, Rocaboy C, Pande V, Meerpoel L, Lim HK, Branch JR, Ondrus J, Hickson I, Bush TL, Bischoff JR, Bignan G.   +12 more
europepmc   +1 more source

<i>In vitro</i> anti-breast cancer study of hybrid cinnamic acid derivatives bearing 2-thiohydantoin moiety. [PDF]

Future Med Chem
Binjawhar DN, Al-Salmi FA, Alghamdi MA, Abu Ali OA, Fayad E, Rizzk YW, Ali NM, El-Deen IM, Eltamany EH.   +8 more
europepmc   +1 more source

[3+2]-Cycloaddition of azomethine ylides to 5-methylidene-3-aryl-2-сhalcogen-imidazolones: access to dispiro indolinone-pyrrolidine-imidazolones. [PDF]

R Soc Open Sci, 2022
Kukushkin ME, Kondratieva AA, Karpov NA, Shybanov DE, Tafeenko VA, Roznyatovsky VA, Grishin YK, Moiseeva AA, Zyk NV, Beloglazkina EK.   +9 more
europepmc   +1 more source

Design, eco-friendly synthesis, and molecular docking studies of isatin hybrids as promising therapeutic agents (anticancer, anticholinesterase inhibitor, α-glucosidase inhibitor, and anti-MRSA). [PDF]

RSC Adv
Seliem IA.
europepmc   +1 more source

Synthesis and Biological Evaluation of Novel Dispiro-Indolinones with Anticancer Activity. [PDF]

Molecules, 2023
Ivanenkov YA, Kukushkin ME, Beloglazkina AA, Shafikov RR, Barashkin AA, Ayginin AA, Serebryakova MS, Majouga AG, Skvortsov DA, Tafeenko VA, Beloglazkina EK.   +10 more
europepmc   +1 more source

Chiral Recognition of Chiral (Hetero)Cyclic Derivatives Probed by Tetraaza Macrocyclic Chiral Solvating Agents via ¹H NMR Spectroscopy. [PDF]

Anal Chem
Wang Y, Zhao H, Yang C, Fang L, Zheng L, Lv H, Stavropoulos P, Ai L, Zhang J.   +8 more
europepmc   +1 more source