Results 71 to 80 of about 1,246 (203)
A highly divergent synthesis of regioisomeric thiohydantoins and pseudothiohydantoins spiro-fused to a pharmacologically valuable pyrrole-2-one fragment involving the reaction of [e]-fused 1H-pyrrole-2,3-diones with thioureas was developed.
Aleksandr I. Kobelev +5 more
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2-(Alkyl-1-yl)-1H-imidazol-5(4H)-ones 5a–n were synthesized via nucleophilic substitution of the methylsulfanyl group of the corresponding 2-(methylthio)-1H-imidazol-5(4H)-ones 3a–c with suitably substituted secondary amines.
Edward R. Biehl +2 more
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Synthesis, antimicrobial and anticancer activities of some 2-thiohydantoin derivatives [PDF]
641-648The vital organic compound 3-[(2-hydroxy-3-methoxybenzylidene)- amino]-2-thiohydantoin 3 has been prepared via the reaction of 2-hydroxy-3-methoxybenzaldehyde 1 with thiosemicarbazide to give N-[(2-hydroxy-3-methoxybenzylidene) amino]thiourea 2 ...
Abubshait, Samar A
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The acid dissociation constants of potential bioactive fused ring thiohydantoin-pyrrolidine compounds were determined by potentiometric titration in 20% (v/v) ethanol-water mixed at 25±0.1°C, at an ionic background of 0.1 mol/L of NaCl using the ...
Yahya Nural +5 more
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Progress on the Chemical Constituents Derived from Glucosinolates in Maca (Lepidium meyenii)
Maca (Lepidium meyenii Walp.), a famous food supplement, has drawn an unprecedented international interest over the last two decades. It was assumed that glucosinolates, macamides, macaenes, and alkaloids are the main bioactive components of Maca before.
Yan-Jie Huang +2 more
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HYDANTOINS: THE SYNTHESIS OF 2-THIOHYDANTOIN. [SEVENTH PAPER.] [PDF]
n ...
Johnson, Treat B., Nicolet, Ben H.
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Apoptotic Effects of Some Thiohydantoin Derivatives
WOS: 000282700000017Objectives: The aim of this study is to investigate the effects of newly synthesized 3-phenly-and 3-(4-methoxyphenyl)-2-thiohydantoin derivatives on 5RP7 ve CO25 cell apoptosis.
Akalın Çiftçi, Gülsen +1 more
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Synthesis of Thiohydantoin-Castanospermine Glycomimetics as Glycosidase Inhibitors
The preparation of bicyclic carbohydrate mimics related to (+)-castanospermine incorporating a thiohydantoin moiety is reported. The synthetic approach is compatible with molecular diversity-oriented strategies and involves alpha-azidoesters, built at the C-5/C-6 segment in gluco- or galactofuranose scaffolds, as the key precursors.
Aguilar Moncayo, Matilde +3 more
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P.G. Department of Chemistry, Sambalpur University. Jyoti Vihar, Burla. Sambalpur-768 019, Orissa. India E-mail : dhruba_dash@yahoo.co.in Manuscript received 15 October 2008, revised 27 April 2009, accepted 18 May 2009 A few complexes of the type [ML2]
D. C. Dash +4 more
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