Results 41 to 50 of about 6,253 (217)

Synthesis of novel 4-thiazolidinone derivatives via one-pot three-component reaction of maleimide, thiosemicarbazide, and Meldrum’s acid

, 2022
The synthesis of novel thiazolidinone derivatives via the three-component reaction has been developed involving the reaction of thiosemicarbazide with maleimide and Meldrum’s acid in a single pot.
Naouel Boufroua (6679082), Sophie Poulain-Martini (13842422), Samia Achouche-Bouzroura (13842425), Elisabet Dunach (640263), Nadia Sadou (13842419)   +4 more
core   +1 more source

Synthesis of Benzimidazole–Based Analogs as Anti Alzheimer’s Disease Compounds and Their Molecular Docking Studies

Molecules, 2020
We synthesized 10 analogs of benzimidazole-based thiosemicarbazide 1 (a–j) and 13 benzimidazole-based Schiff bases 2 (a–m), and characterized by various spectroscopic techniques and evaluated in vitro for acetylcholinesterase (AchE) and ...
Bushra Adalat, Fazal Rahim, Muhammad Taha, Foziah J. Alshamrani, El Hassane Anouar, Nizam Uddin, Syed Adnan Ali Shah, Zarshad Ali, Zainul Amiruddin Zakaria   +8 more
doaj   +1 more source

Aminooxy-, Hydrazide-, and Thiosemicarbazide-Functionalized Saccharides:  Versatile Reagents for Glycoconjugate Synthesis

, 2016
Aminooxy-, Hydrazide-, and Thiosemicarbazide-Functionalized Saccharides:  Versatile Reagents for Glycoconjugate ...
Lisa A. Marcaurelle (1342419), Elena C. Rodriguez (3001716), Carolyn R. Bertozzi (187405)   +2 more
core   +1 more source

Synthesis and Characterization of Novel Corrosion Inhibitor Derived from Oleic Acid: 2-Amino 5-Oleyl-1,3,4-Thiadiazol (AOT)

International Journal of Electrochemical Science, 2012
Novel corrosion inhibitor as a green chemical product namely derivative, 2-amino 5-oleyl-1,3,4-thiadiazol (AOT) was synthesized by cyclization of oleic acid. The new corrosion inhibitor was characterized by FT-IR and NMR spectroscopical methods.
Sutiana Junaedi, Abdul Amir H. Kadhum, Ahmed A. Al-Amiery, Abu Bakar Mohamad, Mohd Sobri Takriff   +4 more
doaj   +1 more source

Pharmacophore Mapping Approach for Drug Target Identification: A Chemical Synthesis and in Silico Study on Novel Thiadiazole Compounds [PDF]

Journal of Clinical and Diagnostic Research, 2017
Introduction: Compounds containing thiadiazole moiety are cognized to possess with variety of clinical and therapeutic activity. Finding a suitable drug target for newly synthesized compounds remain a major bottle neck in current high throughout ...
Rohan J. Meshram, Vijay B. Baladhye, Rajesh N. Gacche, Bhausaheb K. Karale, Rajendra B. Gaikar   +4 more
doaj   +1 more source

Design, Synthesis, Antibacterial Evaluations and In Silico Studies of Novel Thiosemicarbazides and 1,3,4-Thiadiazoles

Molecules, 2022
The emergence of drug-resistant bacterial strains continues to be one of the major challenges of medicine. For this reason, the importance of searching for novel structures of antibacterial drugs chemically different from the currently known antibiotics ...
Sara Janowska, Dmytro Khylyuk, Sylwia Andrzejczuk, Monika Wujec   +3 more
doaj   +1 more source

1,1,4-Derivatives of Thiosemicarbazide—New Non-Staining Antiozonants

, 1973
In the nature of non-staining antiozonants, a new class of compounds, 1,1,4-derivatives of thiosemicarbazide, are proposed. The mechanism of reaction of thiosemicarbazide derivatives with ozone is analogous to the mechanism of this reaction with thiourea
L. K. Zolotarevskaya, A. M. Lipkin, A. E. Grinberg, L. G. Angert   +3 more
core   +1 more source

Determination of the Lipophilicity of Some New Derivatives of Thiosemicarbazide and 1,2,4-triazoline-5-thione with Potential Antituberculosis Activity [PDF]

, 2010
The chromatographic behavior of newly obtained derivatives of thiosemicarbazide and 1,2,4- triazoline-5-thione was determined. The lipophilicity was confirmed by the use of the Reversed Phase Thin-Layer Chromatography (RP-TLC) method.
Ginalska, Grażyna, Polak, Beata, Pitucha, Monika, Popiołek, Łukasz, Swatko-Ossor, Marta   +4 more
core   +1 more source

Engineering Halide Perovskites With Chalcogen‐Based Compounds: Insights Into Stability, Interfaces, and Device Integration

Carbon Energy, EarlyView.
Chalcogen‐based compounds are explored as versatile tools to enhance the stability and performance of halide perovskites. Their roles in defect passivation, ion migration suppression, and interface engineering are analyzed, along with impacts on device efficiency.
Atanu Jana, Deblina Das, Sourav Mal, Tarak Nath Mandal, Sangeun Cho   +4 more
wiley   +1 more source

Synthesis and Evaluation of Antimicrobial Activity of 1, 3, 4-Thiadiazole Analogues for Potential Scaffold

Journal of Pharmacopuncture, 2021
Objectives: Pathogenic microbes are causal agents for various types of severe and even lethal infectious diseases. Despite of development in medication, bacterial and fungal infections still persist to be a vital problem in health care.
Sagar Sahu, Tanesh Sahu, Gunjan Kalyani, Bina Gidwani   +3 more
doaj   +1 more source