Results 11 to 20 of about 14,086 (252)

Palladium(II) Complexes of NS Donor Ligands Derived from Steroidal Thiosemicarbazones as Antibacterial Agents [PDF]

open access: yesMolecules, 2010
We have investigated the antibacterial activity of some new steroidal thiosemicarbazones and their Pd(II) metal complexes were prepared by the reaction of the thiosemicarbazones with [Pd(DMSO)2Cl2].
Abdullah M. Asiri, Salman A. Khan
doaj   +2 more sources

A novel class of thiosemicarbazones show multi-functional activity for the treatment of Alzheimer's disease. [PDF]

open access: yesEuropean journal of medicinal chemistry, 2017
Over 44 million people live with Alzheimer's disease (AD) worldwide. Currently, only symptomatic treatments are available for AD and no cure exists. Considering the lack of effective treatments for AD due to its multi-factorial pathology, development of ...
Duraippandi Palanimuthu   +8 more
semanticscholar   +2 more sources

Antifungal activities of thiosemicarbazones and semicarbazones against mycotoxigenic fungi [PDF]

open access: yesCiência e Agrotecnologia, 2014
Mycotoxigenic fungi can compromise the quality of food, exposing human and animal health at risk. The antifungal activity of eight thiosemicarbazones (1-8) and nine semicarbazones (9-17) was evaluated against Aspergillus flavus, A. nomius, A.
Rojane de Oliveira Paiva   +4 more
doaj   +2 more sources

Synthesis, characterization, antibacterial activity of thiosemicarbazones derivatives and their computational approaches: Quantum calculation, molecular docking, molecular dynamic, ADMET, QSAR

open access: yesHeliyon, 2023
The thiosemicarbazones and their derivatives have been recognized as antimicrobial agents against human pathogenic bacteria and fungi. Regarding these prospective, this study was designed to address the new antimicrobial agents from thiosemicarbazones ...
Mahbub Alam   +6 more
doaj   +2 more sources

Electrochemical Behavior of Some Substituted Thiosemicarbazones and their Reaction Products with Tetracyanoethylene [PDF]

open access: yesInternational Journal of Electrochemical Science, 2008
The electrochemical behavior of substituted thiosemicarbazones has been investigated. It is found that the cyclic voltammetry of all substitutions is different; this can be attributed to the nature of terminal aldehydic group.
S.A.M. Refaey, A.A. Hassan and H.S. Shehata
doaj   +3 more sources

Thiosemicarbazones with tyrosinase inhibitory activity [PDF]

open access: yesMedChemComm, 2019
Thiosemicarbazones reveal strong anti-tyrosinase activity.
Katarzyna Hałdys, Rafał Latajka
openaire   +3 more sources

Structural Studies of 2,6-Diacetyl- and 2,6-Diformylpyridine Bis(thiosemicarbazones) [PDF]

open access: yesJournal of the Brazilian Chemical Society, 2002
Although a large number of crystal structures of heterocyclic thiosemicarbazones have recently appeared in the literature, few structures of heterocyclic bis(thiosemicarbazones) or their metal complexes have been reported.
Brown Christine A.   +4 more
doaj   +3 more sources

Transalkylidation reaction: green, catalyst-free synthesis of thiosemicarbazones and solving the NMR conflict between their acyclic structure and intramolecular cycloaddition products

open access: yesGreen Chemistry Letters and Reviews, 2019
A series of arylidene thiosemicarbazides have been prepared by a new method, which was titled as transalkylidation. This method is an effective, fast, green and clean method. The mechanism of this reaction has been discussed.
Mohamed A. El-Atawy   +3 more
doaj   +2 more sources

StructureActivity Relationships of Di-2-pyridylketone 2Benzoylpyridine, and 2Acetylpyridine Thiosemicarbazones for Overcoming Pgp-Mediated Drug Resistance [PDF]

open access: yes, 2016
Multidrug resistance (MDR) mediated by P-glycoprotein (Pgp) represents a significant impediment to successful cancer treatment. The compound, di-2-pyridylketone 4,4-dimethyl-3-thiosemicarbazone (Dp44mT), has been shown to induce greater cytotoxicity ...
Duraippandi Palanimuthu   +11 more
core   +5 more sources

Para-Substituted Thiosemicarbazones as Cholinesterase Inhibitors: Synthesis, In Vitro Biological Evaluation, and In Silico Study

open access: yesACS Omega, 2023
The current research reports the synthesis of 14 para-substituted thiosemicarbazone derivatives in good to excellent yields using standard procedures. Initially, 4-ethoxybenzaldehyde (1) and 4-nitrobenzaldehyde (2) were refluxed with thiosemicarbazide in
Momin Khan   +8 more
semanticscholar   +1 more source

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